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methyl 1-[3-(4-{[(3-cyclopentylpropyl)amino]methyl}phenoxy)-2-hydroxypropyl]piperidine-4-carboxylate
6-cyano-N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}pyridine-3-carboxamide
(furan-2-ylmethyl)(methyl)({4-methyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)amine
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[2-(2-ethoxyphenyl)ethyl]acetamide
methyl (2S,4R)-1-[(2,5-dimethylphenyl)methyl]-4-(2-methylpropanamido)pyrrolidine-2-carboxylate
1-[(3-methylphenyl)methyl]-4-(quinolin-6-yloxy)piperidine-4-carboxylic acid
[(2S,6S)-4-[(2,5-dimethylphenyl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
1-{pyrazolo[1,5-a]pyridine-3-carbonyl}-4-(pyrimidin-2-yl)piperazine-2-carboxylic acid
3-{5-[2-(1,1-dioxo-1λ6-thiolan-3-yl)ethyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
4-{[2-(4-methoxyphenyl)ethyl]amino}-5-methyl-N-(2-methylpropyl)thieno[2,3-d]pyrimidine-6-carboxamide
5-[1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)pyrrolidin-2-yl]-3-(propan-2-yl)-1,2,4-oxadiazole
3-(azepane-1-carbonyl)-N-[(3-fluorophenyl)methyl]-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-[(3-methoxyphenyl)methyl]piperazin-2-one
1-[3-(3-{[4-(propan-2-yl)phenyl]amino}piperidine-1-carbonyl)phenyl]pyrrolidin-2-one
ethyl 5-{[(4,6-dimethylpyrimidin-2-yl)amino]methyl}furan-2-carboxylate
1-cyclopentyl-3-(3-methoxyphenyl)-3-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]pyrrolidine-2,5-dione
methyl (2S)-2-{[4-(dimethylamino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]amino}propanoate
methyl 3-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]-9-(oxan-2-ylmethoxy)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
5-butyl-1'-[3-(5-methylfuran-2-yl)butyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-cyclohexyl-4-[5-(methoxymethyl)furan-2-amido]piperidine-1-carboxamide
7-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
2-(methylsulfanyl)-3-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]pyridine
(2R)-2-({4-[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}amino)-3-methylbutan-1-ol
2-amino-3-ethyl-N-(2-methoxyethyl)-N-[(2-methylphenyl)methyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
5-ethyl-N-{[4-(3-methylpiperidin-1-yl)phenyl]methyl}-1,2-oxazole-3-carboxamide
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-(methylsulfanyl)benzamide
N-[2-(3-methoxyphenyl)phenyl]-1-[(2-methylphenyl)methyl]piperidine-4-carboxamide
4-chloro-3-{[4-(5-fluoropyrimidin-2-yl)piperazin-1-yl]methyl}-1-methyl-1H-indazole
2-[1-(2H-1,3-benzodioxol-5-ylmethyl)-2,5-dioxo-3-phenylpyrrolidin-3-yl]-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]acetamide
3,5-dichloro-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-(prop-2-en-1-yloxy)benzamide
5-(1H-imidazol-2-yl)-1-(oxolan-2-ylmethyl)-4-phenyl-1H-imidazole
4-(4-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}piperazin-1-yl)phenol
N,1,3-trimethyl-N-[2-(2-methylpiperidin-1-yl)ethyl]-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-(2H-1,3-benzodioxol-5-yl)-5-{spiro[2.3]hexane-1-carbonyl}-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
1-{1'-[5-(methoxymethyl)furan-2-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
dimethyl({[3-methyl-7-(1-methyl-1H-indole-2-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}sulfamoyl)amine
2-[3-({[2-(4-hydroxy-3-methoxyphenyl)ethyl]amino}methyl)-2-methyl-1H-indol-1-yl]acetamide
N,1-dimethyl-N-[1-(pyridin-3-yl)ethyl]-1H-imidazole-2-carboxamide
2-methyl-4-(4-{[4-(4H-1,2,4-triazol-4-yl)piperidin-1-yl]methyl}phenyl)butan-2-ol
3-({ethyl[(trimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)benzonitrile
N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-N,1-dimethyl-5-phenyl-1H-pyrrole-2-carboxamide
(1R,7S)-6-(4-fluoropiperidine-1-carbonyl)-3-(pyridin-3-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
1-(4-chlorophenyl)-3-cyclopropyl-5-(1-methanesulfonylpyrrolidin-2-yl)-1H-1,2,4-triazole
11-[3-ethoxy-4-hydroxy-5-(prop-2-en-1-yl)phenyl]-4,6,10,12-tetraazatricyclo[7.3.0.03,7]dodeca-1,3(7),8,10-tetraen-5-one
2-butoxy-1-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}ethan-1-one
(3S,5R)-1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-5-(cyclopropylcarbamoyl)piperidine-3-carboxylic acid
N-(isoquinolin-5-ylmethyl)-N-methyl-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]acetamide
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-methyl-N-(oxan-4-yl)propanamide
4-(4-methoxyphenoxy)-1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidine
2-{[1-(3,3-dimethylcyclohexyl)piperidin-4-yl]oxy}-4-methoxy-N-(2-methoxyethyl)benzamide