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3-({[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(prop-2-en-1-yl)amino)-1λ6-thiolane-1,1-dione
N-methyl-N-(2-phenyl-1-{1-[3-(trifluoromethyl)benzoyl]piperidin-4-yl}ethyl)-2-(1H-pyrazol-1-yl)acetamide
2-[(4-chlorophenyl)methyl]-8-[2-(4-methyl-1H-pyrazol-1-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
4'-(3-methylbutyl)-1-(oxolane-3-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
4-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-[2-(4-fluorophenyl)morpholin-4-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
2-[4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-yl]-2-azaspiro[4.4]nonane
7-(3-chlorophenyl)-4-(2-methoxyethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-{[1-(1,4-dithiepan-6-yl)pyrrolidin-3-yl]methyl}benzamide
(1-methyl-4-{[4-(methylsulfanyl)phenyl]methyl}piperazin-2-yl)methanol
8-(3-cyclopentylpropyl)-2,8-diazaspiro[4.5]decan-3-one
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-1-[(4-hydroxyphenyl)methyl]-N5-[2-(1-methylpyrrolidin-2-yl)ethyl]piperidine-3,5-dicarboxamide
1-(diethylamino)-3-[5-({[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)amino}methyl)-2-methoxyphenoxy]propan-2-ol
2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]-N-{[4-(morpholin-4-yl)phenyl]methyl}acetamide
2-cyclopropyl-1-[2-(3,4-dimethoxyphenyl)ethyl]-N-[(2-fluorophenyl)methyl]-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
3-(3-{[2-(dimethylamino)ethyl](methyl)amino}piperidine-1-carbonyl)-6-methoxy-1,4-dihydroquinolin-4-one
(1S,5R)-3-cyclobutanecarbonyl-6-(1-methyl-1H-indole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-[1-(1-benzylpiperidin-4-yl)piperidin-4-yl]-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-({1-[2-(morpholin-3-yl)acetyl]piperidin-4-yl}oxy)benzoic acid
(4aS,7aR)-1-benzyl-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(1-benzyl-4-cycloheptylpiperazin-2-yl)ethan-1-ol
1-[(1R,5R)-6-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
1-(6-fluoro-2-oxo-1,2,3,4-tetrahydroquinolin-8-yl)-3-methyl-3-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}urea
3-hydroxy-N-({1-[(4-methoxyphenyl)methyl]pyrrolidin-3-yl}methyl)benzamide
1-ethyl-4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]piperidine
N-benzyl-2,4-dimethyl-N-(1,3-thiazol-2-ylmethyl)-1,3-thiazole-5-carboxamide
1-{2-[2-(4-fluorophenyl)piperidin-1-yl]-2-oxoethyl}-3-methoxy-1,2-dihydropyridin-2-one
N-(oxolan-2-ylmethyl)-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
1-[3-(4-fluorophenoxy)propyl]-4-(3-propyl-1H-pyrazole-5-carbonyl)piperazine
2-{5-[2-(difluoromethoxy)phenyl]-4-phenyl-1H-imidazol-1-yl}-N-methylbutanamide
(3S,5R)-5-[(4-fluorophenyl)carbamoyl]-1-(3-methylbenzoyl)piperidine-3-carboxylic acid
methyl 3-{[5-(2-methylphenyl)-1,2,4-triazin-3-yl]amino}propanoate
N-[2-(2-methylphenyl)ethyl]-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
2-(1-benzyl-3-oxopiperazin-2-yl)-N-(2-hydroxyethyl)-N-propylacetamide
2-[2,5-dioxo-3-phenyl-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]-N-(2-hydroxy-2-phenylethyl)-N-methylacetamide
1-(2H-1,3-benzodioxole-5-carbonyl)-3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidine
1-[7-(1,3-benzothiazol-2-yl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(3,5-dimethyl-1H-pyrazol-1-yl)ethan-1-one
1-[5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]-4-(4-methylpyridin-2-yl)piperazine
N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]quinoline-3-carboxamide
3-[3-methyl-1-(2-methylphenyl)-1H-1,2,4-triazol-5-yl]-1λ6-thiolane-1,1-dione
2-amino-N-(1H-indol-5-ylmethyl)-4-phenylpyrimidine-5-carboxamide
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-(pyridin-3-yl)acetamide
4-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-methyl-6-(propan-2-yl)pyrimidine
1-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-5-phenylpentan-1-one
4-{1-[(4-methoxyphenyl)methyl]-1H-1,2,4-triazol-5-yl}butanoic acid
9-{2-methylthieno[3,2-d]pyrimidin-4-yl}-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
3-(1,3-benzothiazol-2-yl)-N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]propanamide
1-(2-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}phenyl)ethan-1-one
1-methyl-1'-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
1-[7-(5-chloropyridin-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(3,4,5-trimethoxyphenyl)ethan-1-one