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4-(1H-pyrazol-3-yl)-N-{1-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}benzamide
1-ethyl-4-{[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}-1H-pyrrole-2-carbonitrile
7-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]-2-oxa-7-azaspiro[4.5]decane
N-({7-[(2E)-3-(2,3-difluorophenyl)prop-2-enoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-3-carboxamide
3-[(2-ethylbutyl)amino]-5-(methylsulfamoyl)-N-[3-(methylsulfanyl)phenyl]benzamide
1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-4-(4-methyl-5-{[2-(piperidin-1-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)piperidine
4-(5-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}thiophen-2-yl)-2-methylbut-3-yn-2-ol
2-(3,3-diphenylpiperidine-1-carbonyl)pyridine
N-[(4-methyl-1,3-thiazol-2-yl)methyl]-1-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
1-(4-fluorophenyl)-4-[1-(4-methoxybenzoyl)piperidin-3-yl]piperazine
2-{[5-(4-methylphenyl)-1H-pyrazol-3-yl]formamido}-3-phenylpropanoic acid
3-ethyl-4-{5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carbonyl}piperazin-2-one
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)propanamide
1-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}-3-(pyrrolidine-1-carbonyl)piperidine
3-{[2-(pyrazin-2-yl)ethyl]sulfamoyl}-N-(pyrrolidin-3-yl)benzamide
2-{1-[(4-methoxy-3-methylphenyl)methyl]-4-(quinolin-6-ylmethyl)piperazin-2-yl}ethan-1-ol
(2S)-1-{5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}pyrrolidine-2-carboxamide
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(3-chlorophenyl)methyl]-4-{[(2E)-2-methyl-3-phenylprop-2-en-1-yl]amino}pyrrolidine-2-carboxamide
methyl 2-(1-{2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxyphenyl}-N-methylformamido)acetate
ethyl 1-ethyl-5-[3-(thiophen-3-yl)-1H-pyrazole-5-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2,3-dimethyl-6-[4-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]quinoxaline
1-[(3,5-dimethylphenyl)methyl]-4-(3-methyl-1,2-oxazole-5-carbonyl)piperazin-2-one
(5S,9aS,9bS)-5-(3-chloro-4-hydroxy-5-methoxyphenyl)-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-{[cycloheptyl(pyridin-3-ylmethyl)amino]methyl}-N-methylbenzene-1-sulfonamide
4-{5-[2-(pyridin-3-yl)pyrrolidine-1-carbonyl]-1H-pyrazol-3-yl}phenol
N-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2,2-dimethyl-4-oxo-3,4-dihydro-2H-pyran-6-carboxamide
(1S,5R)-6-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-{4-[7-(methylsulfanyl)-3-{[(thiophen-2-ylmethyl)amino]methyl}quinolin-2-yl]piperazin-1-yl}ethan-1-one
7-[(3,4-difluorophenyl)methyl]-2-(4,4,4-trifluorobutyl)-2,7-diazaspiro[4.5]decan-6-one
N-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-methyl-5-{1-[2-(thiophen-2-yl)ethyl]-1H-pyrazol-3-yl}-1,3-thiazol-2-amine
1-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-[(2-methylphenyl)sulfanyl]ethan-1-one
(3S,4R)-N,N-dimethyl-4-(4-methylphenyl)-1-[4-(trifluoromethyl)benzoyl]pyrrolidin-3-amine
N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-methylpropanamide
1-{[1-(3-chloro-4-fluorophenyl)-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]methyl}piperidin-3-ol
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
4-{3-[(1-propylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}benzonitrile
4-[(2S,4S,6R)-4-acetamido-6-(4-fluoro-3-methoxyphenyl)oxan-2-yl]benzoic acid
N-[(3-chloro-2-fluorophenyl)methyl]-4-(2-oxopyrrolidin-1-yl)butanamide
methyl 3-(7-chloro-2-{[(2S)-2-acetamidopropanamido]methyl}-2,3-dihydro-1-benzofuran-5-yl)benzoate
N-methyl-N-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)-2-(1H-1,2,3,4-tetrazol-1-yl)pyridine-4-carboxamide
1-(2-methoxyacetyl)-N-[2-(5-methylfuran-2-yl)ethyl]piperidine-4-carboxamide
1-benzoyl-4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-{2-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}-1,2-dihydropyrimidin-2-one
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-ethyl-N-[(3S,4R)-4-hydroxyoxolan-3-yl]-1H-pyrazole-3-carboxamide
4-[(3,5-dimethoxyphenyl)methyl]-1-(2-methylphenyl)piperazin-2-one
2-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one
2-[3-(dimethylamino)propyl]-9-[(3-methyl-1,2-oxazol-5-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
2-(1H-pyrazol-1-yl)-1-(4-{[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)ethan-1-one
[(4S)-4-amino-5-[4-(4-methylphenoxy)piperidin-1-yl]-5-oxopentyl]urea
4-{[6-(dimethylamino)pyrimidin-4-yl]amino}-1λ6-thiane-1,1-dione