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3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]propanamide
N-(4-{1-[1-(3-cyanopyridin-2-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}phenyl)acetamide
1-(2,6-dimethylpyridin-4-yl)-4-[(3-methyl-1-phenyl-1H-pyrazol-4-yl)methyl]piperazine
3-(3-hydroxyquinoxalin-2-yl)-1-{4-[(pyridin-2-yl)amino]piperidin-1-yl}propan-1-one
(1r,4r)-4-({[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}amino)cyclohexan-1-ol
(4aS,8aR)-1-(2-aminoethyl)-6-(1-phenylcyclopropanecarbonyl)-decahydro-1,6-naphthyridin-2-one
(2S,4R)-4-amino-N,N-diethyl-1-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]pyrrolidine-2-carboxamide
3-(1,4-diazepane-1-carbonyl)-N-(2-methoxybutyl)benzene-1-sulfonamide
(1S,5R)-N-(furan-2-ylmethyl)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
2-cyclopropyl-N-[(3-methoxy-2-propoxyphenyl)methyl]pyrimidine-5-carboxamide
2-{[1-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-4-yl]oxy}-4-methoxy-N-(2-methoxyethyl)benzamide
4-benzyl-1-{[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperidine
3-{[7-(oxane-2-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}pyridine
6-(4-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperazin-1-yl)-9H-purine
2-[4-(furan-2-carbonyl)piperazin-1-yl]-2-[4-(methylsulfanyl)phenyl]acetic acid
4-ethyl-5-methyl-6-[3-(morpholin-4-yl)azetidin-1-yl]pyrimidin-2-amine
(2S)-2-amino-3-(1H-imidazol-4-yl)-N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}propanamide
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-6-methyl-2-oxo-1,2-dihydroquinoline-4-carboxamide
methyl 3-[2-(dimethylamino)benzoyl]-7-oxo-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(4-fluorobenzoyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[2-methyl-1-(pyridin-2-yl)propyl]-4-pentanamidobenzamide
4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-[2-(methylsulfanyl)ethyl]benzamide
3-methyl-8-[3-(pyridin-2-yl)propanoyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-ethyl-1-methyl-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-1H-indole-3-carboxamide
5-(furan-2-yl)-3-{[2-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-1H-imidazol-1-yl]methyl}-1,2,4-oxadiazole
1-methyl-9-(prop-2-en-1-yl)-4-(quinolin-4-ylmethyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
2-methoxy-N-({5-[2-methyl-2-(pyrrolidin-1-ylmethyl)propyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide
7-methyl-3-[6-(propan-2-yl)-1H-indole-2-carbonyl]-3,7,11-triazaspiro[5.6]dodecan-12-one
3-[2-(2,6-difluorophenyl)ethyl]-1-(5-methyl-1,2-oxazole-3-carbonyl)piperidine
(4aS,8aR)-6-(4-cyclobutyl-6-methylpyrimidin-2-yl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
methyl (2S,4R)-1-[(3-methylthiophen-2-yl)methyl]-4-(2-phenylbenzamido)pyrrolidine-2-carboxylate
7-{[4-(methylsulfanyl)phenyl]methyl}-3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
2-{3-[2-(2-fluorophenyl)ethyl]piperidine-1-carbonyl}-5-methylpyrazine
N-[2-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)propyl]-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
5-chloro-2-[3-(2-methylpiperidin-1-yl)azetidine-1-carbonyl]phenol
2-benzyl-N-[3-(1H-pyrazol-1-yl)propyl]-1,3-benzoxazole-5-carboxamide
1-benzyl-4-(3-phenyl-1H-pyrazole-5-carbonyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
5-{4-[(2-fluorophenyl)methyl]piperidine-1-carbonyl}-2-(methylsulfanyl)pyrimidine
1-[(3-chlorophenyl)methyl]-N-cyclohexyl-N-[2-(dimethylamino)ethyl]-1H-1,2,3-triazole-4-carboxamide
4-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-1-(3-methoxyphenyl)piperazin-2-one
1-(2H-1,3-benzodioxole-5-carbonyl)-3-[3-(propan-2-yloxy)benzoyl]piperidine
(2S,4R)-4-(benzylamino)-1-(2,2-diphenylethyl)-N-methylpyrrolidine-2-carboxamide
1-[(2E)-3-(pyridin-3-yl)prop-2-enoyl]-4-{[2-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
1-(4-fluorophenyl)-N-{[(3S,4S)-3-hydroxypiperidin-4-yl]methyl}-3,5-dimethyl-1H-pyrazole-4-carboxamide
4-ethyl-3-({1-[(3-hydroxyphenyl)methyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-3-{[(5-methylthiophen-2-yl)methyl]amino}benzamide
N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-2-hydroxy-N-methyl-4-(methylsulfanyl)butanamide
N-ethyl-4,4,4-trifluoro-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}butanamide
1-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-{2-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
methyl 2-(5-{1-[(2-hydroxy-5-methylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-3-yl)acetate