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1-[3-(dimethylamino)phenyl]-3-[4-(pyrrolidin-1-yl)butyl]urea
N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-3-(1H-pyrazol-1-yl)benzamide
N-[(1-benzylpyrrolidin-3-yl)methyl]-2,3-dihydro-1H-indene-2-carboxamide
2-({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(pyridin-2-ylmethyl)amino)butan-1-ol
N-[(2S)-1-hydroxy-4-(methylsulfanyl)butan-2-yl]-5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carboxamide
2-(4-{4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}pyrimidin-5-yl)acetic acid
(4aS,8aR)-6-(1-aminocyclobutanecarbonyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
8-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[(2-ethyl-6-methylpyridin-3-yl)oxy]-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]acetamide
N-[(1s,4s)-4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]cyclohexyl]adamantane-1-carboxamide
2-(2,3-dihydro-1H-isoindol-2-yl)-N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methylacetamide
1-cyclopentyl-5-oxo-N-{2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl}pyrrolidine-3-carboxamide
2-[1-cyclopentyl-3-(3-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-[(3,4-dimethoxyphenyl)methyl]-N-methylacetamide
(4aS,8aR)-1-(3-aminopropyl)-6-(1-benzofuran-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
2-(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-N,N,5-trimethylpyrimidin-4-amine
(4aR,8aS)-6-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1-{[3-(trifluoromethyl)phenyl]methyl}-decahydro-1,6-naphthyridin-2-one
N-(2-oxo-2,3-dihydro-1H-indol-5-yl)-1-benzothiophene-2-carboxamide
8-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
3-ethyl-1-methyl-N-{[3-methyl-7-(2-phenylacetyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-1H-pyrazole-5-carboxamide
1-(3-chloro-4-methoxyphenyl)-N-methyl-5-oxo-N-(1H-pyrazol-3-ylmethyl)pyrrolidine-3-carboxamide
N-({4-methoxy-3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)-2-(1H-pyrazol-1-yl)acetamide
3-(3-hydroxyquinoxalin-2-yl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}propanamide
5-cyclopropyl-1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-N-(pyridin-2-ylmethyl)-1H-pyrazole-4-carboxamide
4-({2-[5-methyl-6-(4H-1,2,4-triazol-4-yl)pyridin-3-yl]phenyl}methyl)morpholine
N-(1-{1-[(4-ethylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
5-[5-(pyrrolidine-1-carbonyl)furan-2-yl]-1,2,3,4-tetrahydroisoquinoline
N-(5-{[ethyl(oxan-2-ylmethyl)carbamoyl]amino}-2-methylphenyl)cyclopentanecarboxamide
{4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenyl}methanamine
(1-{[methyl({[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl})amino]methyl}cyclobutyl)methanol
1-ethyl-5-{4-[2-(pyridin-4-yl)ethyl]piperazin-1-yl}-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
1-(but-3-enoyl)-N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]piperidine-2-carboxamide
(1-{[1-(6-chloropyridazin-3-yl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)methanol
7-[(2,3-difluorophenyl)methyl]-2-(6-oxo-1,6-dihydropyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
4-[(4-fluorophenyl)methyl]-1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
1-(2-hydroxyethyl)-4-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}-1,4-diazepan-6-ol
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-(5-propyl-1,2-oxazole-3-carbonyl)piperidin-3-yl]piperazine
5-[3-(3-methoxyphenoxymethyl)piperidine-1-carbonyl]-2-methylpyrimidin-4-ol
(1S,4S)-2-{2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxybenzoyl}-2-azabicyclo[2.2.1]heptane
3-(2,3-dihydro-1H-inden-2-yl)-8-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-1-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2R,3R,6R)-5-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
(2-oxo-2-{6-[(1-phenylethyl)sulfamoyl]-1,2,3,4-tetrahydroisoquinolin-2-yl}ethyl)urea
4-(4-methyl-3-phenylpiperazine-1-carbonyl)-6-(2-methylpropyl)-1,2-dihydropyrimidin-2-one
(1S,5R)-6-benzyl-3-[3-(3-methoxyphenyl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}-4-phenylpiperidine-4-carbonitrile
N-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
N-[(3,4-dimethoxyphenyl)methyl]-3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(pyridin-2-ylmethyl)benzamide
methyl 2-(4-{[(1R,5S,6R)-3-(diethylcarbamoyl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl}-2-oxopiperazin-1-yl)acetate
2-[2-(thiophen-2-yl)ethyl]-1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperidine
4-[2-(4-chloro-1H-pyrazol-1-yl)acetyl]-1-[(3,5-dimethylphenyl)methyl]piperazin-2-one
2-[4-(dimethyl-1,3-thiazole-5-carbonyl)piperazin-1-yl]-4-phenylpyrimidine