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6-[2,6-dimethyl-4-(piperidin-1-ylmethyl)phenoxy]pyridine-3-carboxamide
6,6-dimethyl-5-oxo-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}thiomorpholine-3-carboxamide
6-[2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetyl]-N-[(1-phenylcyclopentyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
6-[(diethylamino)methyl]-N-methyl-N-(pyridin-2-ylmethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
ethyl 2-[({1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}carbamoyl)amino]acetate
5-[(4-methylpiperazin-1-yl)methyl]-N-[(2R)-1,1,1-trifluoro-3-methylbutan-2-yl]furan-2-carboxamide
N-methyl-2-oxo-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-1H,2H,5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
3-(4-fluorophenyl)-4-[3-(3-hydroxy-3-methylbut-1-yn-1-yl)benzoyl]piperazin-2-one
[2-methoxy-1-(pyridin-2-yl)ethyl](methyl)[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]amine
(2S,4R)-4-[(adamantan-2-yl)amino]-1-(2,2-diphenylethyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
(3aS,6aR)-3-[2-(4-fluorophenyl)ethyl]-5-[3-(1H-pyrazol-1-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
3,3-diethyl-1-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}urea
1-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}-3-(1-methylpiperidin-3-yl)propan-1-one
1-[(4-methoxyphenyl)methyl]-N-methyl-N-[(3-methylthiophen-2-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
3-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidine-1-carbonyl]-2,6-dimethyl-1,4-dihydropyridin-4-one
4-{3-[4-(2,3-dimethylphenyl)piperazine-1-carbonyl]piperidin-1-yl}-2-(2-methoxy-2-methylpropyl)-2,3-dihydro-1H-isoindole-1,3-dione
5-(4-methylphenyl)-4-[1-(2,3,4-trimethoxybenzoyl)piperidin-3-yl]pyrimidine
1-[1-(1-ethyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}[(4-methylphenyl)(pyridin-4-yl)methyl]amine
1-methyl-2-(morpholin-4-yl)-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-1H-1,3-benzodiazole-5-carboxamide
(2S,4S)-4-[2-(3,5-dimethyl-1H-pyrazol-1-yl)acetamido]-N-ethyl-1-(3-methylbut-2-en-1-yl)pyrrolidine-2-carboxamide
1-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}propane-1,2-dione
2-[1-cyclopropyl-2,5-dioxo-3-(4-phenylphenyl)pyrrolidin-3-yl]-N-methyl-N-(thiophen-3-ylmethyl)acetamide
1-[(6-methylpyridin-2-yl)methyl]-4-(2-methylpyridin-4-yl)-1,4-diazepane
N-[(2-fluorophenyl)methyl]-4-methyl-5-{1-[2-(morpholin-4-yl)ethyl]-1H-pyrazol-3-yl}-1,3-thiazol-2-amine
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-{[1-(2-methoxyethyl)piperidin-3-yl]methyl}acetamide
3-[N-benzyl-1-(8-chloroquinolin-2-yl)formamido]propanamide
N-(dicyclopropylmethyl)-N-methyl-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
(3aR,6aS)-5-[5-(3-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]-2-methyl-octahydropyrrolo[3,4-c]pyrrole-1,3-dione
3-methyl-6-[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]-2,3-dihydro-1,3-benzoxazol-2-one
N-cyclopentyl-4-[6-(piperazin-1-yl)pyridin-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
(3R,4R)-1-[1-(3-chloro-4-methylphenyl)piperidin-4-yl]-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
1-{4-[(3,4-difluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}-2-hydroxyethan-1-one
(2R,3S,6R)-3-(3,5-difluorophenyl)-5-(6-methylpyridine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
[(2S,4R,5R)-5-(2-fluorophenyl)-4-[({[5-(hydroxymethyl)furan-2-yl]methyl}amino)methyl]-1-methylpyrrolidin-2-yl]methanol
methyl 4-[ethyl({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)carbamoyl]benzoate
N-{1-[(4-fluorophenyl)methyl]piperidin-4-yl}-2-(pyridin-4-yl)pyrimidine-5-carboxamide
5-(3-acetylphenoxymethyl)-N-methyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1H-pyrazole-3-carboxamide
5-[(2S)-1-methanesulfonylpyrrolidin-2-yl]-3-(2-methoxyethyl)-1-(2-phenylethyl)-1H-1,2,4-triazole
2-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1H,2H,3H,4H,5H-pyrido[4,3-b]indole
1-methyl-N-{[8-({4-[methyl(phenyl)amino]phenyl}methyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-1H-pyrazole-5-carboxamide
1-(4-chlorophenyl)-N-({1-[3-(6-oxo-1,6-dihydropyridazin-3-yl)propanoyl]piperidin-3-yl}methyl)cyclopropane-1-carboxamide
1-[(4-fluorophenyl)methyl]-4-[3-(1H-pyrazol-4-yl)benzoyl]piperazine
7-methoxy-4-methyl-2-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonan-3-yl]quinazoline
2-methoxy-5-[(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)methyl]phenol
2-{2-[(4-methylphenyl)methyl]benzoyl}-2,7-diazaspiro[4.5]decan-6-one
2-[5-(5-ethyl-1,3-oxazol-4-yl)-3-(2-methylpropyl)-1H-1,2,4-triazol-1-yl]pyridine
2-[5-cyclopropyl-4-(4-phenylpiperazine-1-carbonyl)-1H-pyrazol-1-yl]-4-(5-methylfuran-2-yl)pyrimidine
3-(methoxymethyl)-1-(2-oxo-2-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-yl}ethyl)-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
7-(2,2-dimethylpropyl)-2-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one