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1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[3-(pyridin-4-yl)propyl]piperidine-3-carboxamide
methyl 5-[(4-methylpentan-2-yl)amino]-3-(oxolane-3-amido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-{1-[(4-methoxyphenyl)methyl]piperidin-4-yl}-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
5-benzyl-4-(1-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}piperidin-3-yl)-2-methylpyrimidine
ethyl 1-(cyclopropylmethyl)-5-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-(pyridin-2-yl)-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
3-cyclopropyl-1-[4-(dimethylamino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]propan-1-one
3-[2-(2H-1,3-benzodioxol-5-ylmethyl)-5-oxopyrrolidin-2-yl]-N-[(2-benzyl-1,3-thiazol-4-yl)methyl]propanamide
2-(propan-2-yloxy)-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}propanamide
N-[3-(1H-imidazol-1-yl)propyl]-9-methoxy-7-oxo-3-{[4-(propan-2-yl)phenyl]methyl}-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2,3,6-trimethyl-4-[4-(4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]quinoline
N-{1-[1-(pyridine-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2H-1,3-benzodioxole-5-carboxamide
(1R,7S)-3-[(3-methoxyphenyl)methyl]-N-methyl-4-oxo-N-[2-(1H-pyrazol-1-yl)ethyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
methyl 3-[(4-acetamidophenyl)methyl]-9-[(4-fluorophenyl)methoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
8-[3-(2-methoxyphenyl)benzoyl]-2,8-diazaspiro[4.5]decan-3-one
1-(7-methanesulfonyl-4-methylquinazolin-2-yl)-N-[(1R)-1-(3-methoxyphenyl)ethyl]piperidine-4-carboxamide
N-{[7-(3,6-dimethylpyrazin-2-yl)-4-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-(4-methoxyphenyl)cyclopentane-1-carboxamide
1-(4-methylphenyl)-4-[6-(4H-1,2,4-triazol-4-yl)pyridine-3-carbonyl]piperazin-2-one
8-{[4-hydroxy-3-methoxy-5-(prop-2-en-1-yl)phenyl]methyl}-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
6-{1-cyclohexyl-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl}-2-methyl-2,3-dihydropyridazin-3-one
3-{[(4-chlorophenyl)methyl]amino}-5-(dimethylsulfamoyl)-N-[(1R)-1-(4-methoxyphenyl)ethyl]benzamide
1-[2-({methyl[2-(oxan-4-yl)ethyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
(3R,4R)-4-(2-methoxyethyl)-1-{[2-(2-methoxyphenyl)pyrimidin-5-yl]methyl}-3-methylpiperidin-4-ol
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(oxan-4-ylmethyl)acetamide
6-[(2E)-3-(3,4-difluorophenyl)prop-2-enoyl]-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
2-(dimethyl-1,3-thiazol-5-yl)-N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]acetamide
1-[2-(dimethylamino)ethyl]-5-(4-phenylpiperidine-1-carbonyl)piperidin-2-one
2-{1-[(4-ethoxyphenyl)methyl]-4-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
2-{[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-3,5-dimethyl-1,4-dihydropyridin-4-one
N-butyl-4-(cyclopropylamino)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
1-(2-methoxyphenyl)-5-(1H-1,2,3-triazol-1-ylmethyl)-1H-1,2,4-triazole
2-{[3-(2-hydroxyethyl)-4-(2-methylpropyl)piperazin-1-yl]methyl}-4-methoxyphenol
1-cyclopentanecarbonyl-N-[(1R,2S)-1-hydroxy-1-phenylpropan-2-yl]piperidine-4-carboxamide
2-(1,2-benzoxazol-3-yl)-N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}acetamide
4-[1-(1-{6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidin-4-yl)ethyl]morpholine
3-[cyclopropyl(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-1-[2-fluoro-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
5-benzenesulfonamido-1-ethyl-2-methyl-N-[1-(pyridin-2-yl)propan-2-yl]-1H-1,3-benzodiazole-7-carboxamide
(4aR,7aS)-1-acetyl-4-(pyrazine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
{3-[2-(6-fluoro-1H-1,3-benzodiazol-2-yl)-6-methoxyphenoxy]propyl}dimethylamine
4-hydroxy-N-methyl-2-(4-methylphenyl)-N-[1-(pyridin-2-yl)ethyl]pyrimidine-5-carboxamide
2-phenyl-N-[2-(1H-pyrazol-4-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-hydroxy-1-[1-(4-phenoxyphenyl)-1H-1,2,3,4-tetrazol-5-yl]piperidine-4-carboxylic acid
2-(3-hydroxypropyl)-9-[3-(2-methylphenyl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(1,3-thiazol-2-yl)piperidine
N-{[5-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-methylpiperidine-2-carboxamide
4-fluoro-N-{[5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
3-[2-(2-fluorophenyl)acetyl]-9-methoxy-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
5-[1-(4-ethenylbenzoyl)piperidin-4-yl]-5-[(3-fluorophenyl)methyl]-3-(2-methoxyethyl)imidazolidine-2,4-dione
N-[5-(morpholin-4-yl)pentyl]-1-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
N-(5-chloro-2-methoxyphenyl)-3-{1-[(5-cyano-1H-pyrrol-3-yl)methyl]piperidin-3-yl}propanamide