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N-ethyl-2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-(oxolan-2-ylmethyl)benzamide
1-(4-{2-[7-(3,4-dimethoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxoethyl}phenyl)imidazolidin-2-one
N-(1-cyanocyclohexyl)-3-(1H-pyrazol-1-ylmethyl)benzamide
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-2-hydroxybutanamide
N-(adamantan-2-yl)-2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}benzamide
N-[2-(3,4-dimethoxyphenyl)ethyl]-1-(7-methoxy-4-methylquinazolin-2-yl)piperidine-3-carboxamide
1-[2-(1-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-2-yl)ethyl]pyrrolidin-2-one
1-(oxan-4-ylmethyl)-4-pentyl-1H-1,2,3-triazole
{[2-cyclohexylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)[(3-methylthiophen-2-yl)methyl]amine
1-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}-2-(pyridin-3-yl)ethan-1-one
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-(pyridine-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
methyl 3-{[(1,4-dioxan-2-ylmethyl)carbamoyl]amino}-4-methylbenzoate
2-cyclopentyl-9-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
3-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-ethyl-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]butanamide
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-5-(4-fluorophenyl)-1,2,4-triazin-3-amine
(3aS,6aR)-3-(pyridin-2-ylmethyl)-5-(1,3-thiazol-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-(1-methyl-4-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperazin-2-yl)ethan-1-ol
4-(3,4-difluorobenzoyl)-1-{dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}piperidine
1-[(3,4-difluorophenyl)methyl]-3-[5-(2-methylbutan-2-yl)-1,3,4-thiadiazol-2-yl]urea
methyl 4-oxo-4-{9-oxo-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}butanoate
(2R,3R,6R)-3-(3,5-difluorophenyl)-N-(propan-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxamide
(3S,4R)-1-{4-[(2-fluorophenyl)methoxy]benzoyl}-4-methylpiperidine-3,4-diol
N-(butan-2-yl)-3-oxo-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecane-9-carboxamide
N-ethyl-4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-N-methylpiperidine-1-sulfonamide
5-oxo-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
4-[5-(2,5-dimethylfuran-3-yl)-3-(oxan-4-yl)-1H-1,2,4-triazol-1-yl]pyridine
5-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-N-phenylpyrimidin-2-amine
5-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-3,4-dihydropyrimidin-4-one
1-(2-phenylpropyl)-4-(4H-1,2,4-triazol-3-yl)piperidine
2-{2,5-dioxo-3-phenyl-1-[3-(pyridin-3-yloxy)propyl]pyrrolidin-3-yl}-N-(2-methoxyethyl)-N-(propan-2-yl)acetamide
N-{[2-(4-acetylpiperazin-1-yl)-7-methoxyquinolin-3-yl]methyl}-N-(2-methoxyethyl)-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
(2R)-N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N-methyloxolane-2-carboxamide
1'-[1-(propan-2-yl)-1H-pyrrole-2-carbonyl]-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[(3-methylpyridin-2-yl)methyl]-4-[2-(pyrrolidin-3-yl)benzoyl]piperazine
N-(4-{2-oxo-2-[2-(1H-pyrazol-1-ylmethyl)pyrrolidin-1-yl]ethoxy}phenyl)propanamide
2-[3-(2-chlorophenyl)-1-cyclopentyl-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-(oxan-2-ylmethyl)acetamide
2-amino-3-ethyl-N-methyl-N-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
4'-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-1-(1-methylcyclopropanecarbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-(3,4-dimethoxyphenyl)-3-methyl-3-[3-(oxolan-2-yl)propyl]urea
1-methyl-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carboxamide
2-{8-[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl}acetamide
(2R,6S)-2,6-dimethyl-4-{6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carbonyl}morpholine
1-[(2,6-difluorophenyl)methyl]-N-methyl-N-(1,3-thiazol-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-methoxyethyl 4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxylate
propan-2-yl 2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carboxylate
{[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)[1-(pyrimidin-4-yl)ethyl]amine
3-(2,6-dimethoxyphenyl)pyrazine-2-carbonitrile
3-hexyl-8-(5-methyl-1,3-oxazole-4-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
ethyl 4-({3-[2-hydroxy-3-(piperidin-1-yl)propoxy]-4-methoxyphenyl}methyl)piperazine-1-carboxylate
1-ethyl-N-{1-[(3-hydroxyphenyl)methyl]piperidin-4-yl}-3-(propan-2-yl)-1H-pyrazole-5-carboxamide