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(2S,4S)-4-[5-(1,5-dimethyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]-1-methylpyrrolidine-2-carboxylic acid
3-[(diethylamino)methyl]-6-methoxy-1,2-dihydroquinolin-2-one
5-{[4-(1,5-dimethyl-1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-2-ethoxypyridine
9-(2-methoxypyridine-4-carbonyl)-1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane
3-hydroxy-3-(1,4-oxazepan-4-ylmethyl)-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
(1S,4S)-2-(2-fluorophenyl)-5-[1-(2-phenylethyl)piperidin-4-yl]-2,5-diazabicyclo[2.2.1]heptan-3-one
(3S,4R)-N,N-dimethyl-4-propyl-1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-amine
2-[(3,5-difluorophenyl)methyl]-8-[(dimethyl-1,2-oxazol-4-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
[(3R,4R)-4-[(4-ethylpiperazin-1-yl)methyl]-1-(3-fluoropyridin-2-yl)pyrrolidin-3-yl]methanol
methyl(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl){[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}amine
ethyl 2,4-dimethyl-5-[methyl({[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl})carbamoyl]-1H-pyrrole-3-carboxylate
7-[(2-fluorophenyl)methyl]-2-(5-methyl-1H-pyrazole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxo-N-phenylacetamide
3-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]-1,2,3,4-tetrahydroisoquinolin-1-one
N-[(1-cyclohexylpiperidin-3-yl)methyl]-3-(1,2-oxazolidin-2-yl)-N-(pyridin-3-ylmethyl)propanamide
4-[1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)piperidin-3-yl]-2-methyl-5-(3-methylphenyl)pyrimidine
4-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)butan-1-ol
3-[(1-ethyl-2-oxo-1,2-dihydropyridin-4-yl)formamido]-N-phenylpropanamide
3-{[2-(2-chlorophenyl)-2-hydroxyethyl]amino}-N-(thiophen-2-ylmethyl)propanamide
1-(cyclohexylmethyl)-N-[1-(6-methoxynaphthalen-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-(3-phenylpropyl)-1-(pyrimidin-2-yl)piperidine-3-carboxylic acid
N-(1,4-dioxan-2-ylmethyl)-2-[7-methyl-2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetamide
7,7-dimethyl-2-[2-(pyrrolidin-1-yl)ethyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-methyl-6-{1-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]piperidin-3-yl}-3,4-dihydropyrimidin-4-one
N-[3-hydroxy-2-(thiophen-3-ylmethyl)propyl]-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
6-[3-hydroxy-2-(thiophen-3-ylmethyl)propyl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
4-[(6-chloro-2-fluoro-3-methylphenyl)methyl]-1-methyl-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
2-{4-[3-(azepan-1-ylmethyl)benzoyl]morpholin-3-yl}acetic acid
N-[2-(dimethylamino)ethyl]-4-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
N-{1-[(4-methylphenyl)methyl]cyclopropyl}-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-2-[1-cyclopentyl-3-(3-fluorophenyl)-2,5-dioxopyrrolidin-3-yl]-N-methylacetamide
N-[(3R,4S)-1-[(2-aminopyridin-3-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]-3-hydroxypropanamide
(3-cyclopentylpropyl)({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)methylamine
2-ethoxy-4-{[3-(2-hydroxyethyl)-4-(thiophen-2-ylmethyl)piperazin-1-yl]methyl}phenol
1-(6-aminopyrimidin-4-yl)-4-(1H-1,3-benzodiazol-1-yl)piperidine-4-carboxylic acid
5-(3-{2-amino-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-5-yl}-3-oxopropyl)imidazolidine-2,4-dione
2-[1-(morpholine-4-sulfonyl)pyrrolidin-3-yl]benzoic acid
N-[2-(2-phenoxyethoxy)phenyl]-1,4-dioxane-2-carboxamide
1-[(3-chlorophenyl)methyl]-3-(2-methoxyethyl)-5-[2-(5-methyl-1H-pyrazol-1-yl)ethyl]-1H-1,2,4-triazole
2-[(3-fluorophenyl)methyl]-4-(pyridin-3-ylmethyl)morpholine
N-{[(3S,4S)-1-(2,1,3-benzoxadiazol-4-ylmethyl)-3-hydroxypiperidin-4-yl]methyl}furan-2-carboxamide
4-[6-(2,5-dimethylphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]morpholine
N-[(3R,4R)-3-hydroxy-1-[(4-methoxy-2-methylphenyl)methyl]piperidin-4-yl]pyridine-4-carboxamide
3-(azepane-1-sulfonyl)-N-(pyrimidin-4-ylmethyl)benzamide
N-methyl-N-(quinolin-2-ylmethyl)-6-[(thiophen-2-ylmethyl)amino]pyridine-3-carboxamide
2-[3-(2,5-difluorobenzoyl)piperidin-1-yl]-5-ethylpyrimidine
3-(4-chloro-2-methylbenzoyl)-1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidine
4-methyl-N-{[8-(3-methylbutanoyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}benzamide
6-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-4-amine
3-[2-(4-ethylpiperazin-1-yl)ethyl]-8-(piperidin-3-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one