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1-[2-(4-{1H-pyrazolo[3,4-b]pyridin-1-yl}phenoxy)ethyl]pyrrolidine
1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-4-(4-methyl-5-{[2-(piperidin-1-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)piperidine
N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-2-(2-phenyl-1H-imidazol-1-yl)acetamide
3-({[3-(1H-imidazol-1-yl)propyl](pyridin-4-ylmethyl)amino}methyl)-4H-chromen-4-one
4-chloro-2-hydroxy-N-[(4-methyloxan-4-yl)methyl]benzamide
1-[(4-methoxyphenyl)methyl]-3-{[(pyridin-3-ylmethyl)amino]methyl}-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-2-one
1-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3,5-dimethyl-1H-1,2,4-triazole
4-(1-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}azetidin-3-yl)pyridine
1-methyl-8-(naphthalene-1-carbonyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-N-(1H-indol-4-ylmethyl)propanamide
2-(1,2-benzoxazol-3-yl)-1-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}ethan-1-one
1-[(3,4-dimethoxypyridin-2-yl)methyl]-3-methoxy-1,2-dihydropyridin-2-one
4-ethyl-6-[3-(1H-imidazol-2-yl)piperidin-1-yl]-2-(piperidin-1-yl)pyrimidine
(1S,5R)-N-ethyl-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
N-(4-{4-[(quinolin-6-ylmethyl)amino]piperidin-1-yl}phenyl)cyclopentanecarboxamide
N-[3-(methylamino)propyl]-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
2-methyl-N-({3-methyl-7-[2-(4-methylphenoxy)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)furan-3-carboxamide
9-methoxy-7-(2-methoxyphenyl)-4-(1,3-thiazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
[(2-methoxypyridin-3-yl)methyl](methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
4-methyl-6-[4-({2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}amino)piperidin-1-yl]pyrimidin-2-amine
[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
N,3,4,7-tetramethyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-1H-indole-2-carboxamide
6-{2-[(4,6-dimethylpyrimidin-2-yl)amino]ethyl}-2-methylpyrimidin-4-ol
4-[(dimethylamino)methyl]-1-(5-fluoro-1H-indole-2-carbonyl)azepan-4-ol
2-fluoro-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-5-sulfamoylbenzamide
(5-{[methyl({[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl})amino]methyl}furan-2-yl)methanol
4-(1-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}azetidin-3-yl)pyridine
4-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}-6-(pyrrolidin-1-yl)pyrimidine
N-butyl-2-[3-(2-chlorophenyl)-1-(2-methoxyethyl)-2,5-dioxopyrrolidin-3-yl]-N-methylacetamide
N-{2-[5-(3-methyl-1H-indol-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}acetamide
N-[(2-ethyl-5-fluoro-3-methyl-1H-indol-7-yl)methyl]-3-(N-methylmethanesulfonamido)propanamide
4-(5-chlorothiophene-2-carbonyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one
1-(6-cyanopyridin-2-yl)-4-(2-fluoro-5-methylphenoxy)piperidine-4-carboxylic acid
(2,4,6-trimethyl-3-{[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidin-1-yl]methyl}phenyl)methanol
5-chloro-4-({4-[(2-ethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)-2-methoxyphenol
3-(1,3-benzoxazol-2-ylmethyl)-8-fluoro-3,4-dihydroquinazolin-4-one
2-(4-fluoro-2-methoxyphenyl)-5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridine
N-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]-1,9-dioxaspiro[5.5]undecan-4-amine
6-(3-fluoro-4-phenylphenyl)-9H-purin-2-amine
2-(4-fluorophenoxymethyl)-N-[1-(pyrazin-2-yl)propan-2-yl]-1,3-oxazole-4-carboxamide
3-{[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl](benzyl)amino}propanamide
3-[5-(3-methoxypropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
1-[9-methoxy-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
4-[(4-fluorophenyl)methyl]-1-methanesulfonyl-3-(propan-2-yl)-1,4-diazepan-5-one
(1S,5R)-3-(2,3-difluoro-4-methoxybenzoyl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[3-(furan-2-yl)propanoyl]-4-(2-methylphenoxy)piperidine-4-carboxylic acid
6-ethyl-N2,N2-dimethyl-N4-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyrimidine-2,4-diamine
2-(2-fluoro-6-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
7-(cyclopropylmethyl)-2-[5-(methoxymethyl)thiophene-2-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
1-(6-{4-[3-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}pyridin-3-yl)ethan-1-one