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2-(3-methylbut-2-en-1-yl)-8-[(6-methylpyridin-2-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-[2-(3,4-dimethoxyphenyl)ethyl]-1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-methylpiperidin-3-amine
2-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N,N-dimethylacetamide
N-[1-(cyclohexylmethyl)piperidin-3-yl]-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
6-(2,1,3-benzothiadiazol-5-ylmethyl)-N-[(4-phenyloxan-4-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
1-(methoxymethyl)-N-methyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]cyclobutane-1-carboxamide
(2R,3R,6R)-5-(2,3-dihydro-1-benzofuran-7-carbonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
1-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-(pyridin-4-yl)propan-1-one
3-(1-methyl-1H-pyrrol-2-yl)-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-1H-pyrazole-5-carboxamide
3-[2-(azocan-1-yl)-2-oxoethyl]-3-phenyl-1-(pyridin-3-ylmethyl)pyrrolidine-2,5-dione
1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-3-(4H-1,2,4-triazol-3-yl)piperidine
2-[2-(1H-imidazol-1-yl)ethyl]-1-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]piperidine
1-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]-2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]ethan-1-one
1'-(2-methylbenzoyl)-5-(3-methylbut-2-en-1-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(4aS,8aR)-6-(1H-imidazol-4-ylmethyl)-1-(2-phenylethyl)-decahydro-1,6-naphthyridin-2-one
5-[4-(3-fluorophenoxy)piperidine-1-carbonyl]-1-[2-(pyridin-2-yl)ethyl]piperidin-2-one
5-(2,5-dimethylpyrimidin-4-yl)-N-phenyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
({4-[1-(furan-3-carbonyl)piperidin-2-yl]phenyl}methyl)dimethylamine
3-{[4-(2-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyridine
5-[1-(2-ethoxyacetyl)pyrrolidin-2-yl]-N-[2-(1H-imidazol-4-yl)ethyl]thiophene-2-carboxamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-{1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidin-4-yl}propanamide
1-{[(1R)-1-cyclohexylethyl]carbamoyl}-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
N-{2-[(1-methoxypropan-2-yl)amino]ethyl}pyridin-3-amine
N-[2-(1-methylpiperidin-3-yl)ethyl]isoquinoline-3-carboxamide
N-[4-(furan-2-yl)phenyl]-1-(pyridine-2-carbonyl)piperidine-3-carboxamide
2-(2H-1,3-benzodioxol-5-yl)-N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]acetamide
N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-cyclobutylpyrrolidine-2-carboxamide
N-(1-{2-[(2,6-dimethylphenyl)amino]propanoyl}piperidin-4-yl)methanesulfonamide
N-methyl-N-{3-[(4-methylphenyl)sulfanyl]propyl}-2-[4-(propan-2-yl)morpholin-2-yl]acetamide
N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-2-methyloxane-2-carboxamide
3-{1-[2-(2-fluorophenoxymethyl)-1,3-oxazol-4-yl]-N-methylformamido}-N-methylbutanamide
3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N,N-bis(prop-2-en-1-yl)propanamide
N-[(3-methylpyridin-2-yl)methyl]-2-phenyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
3-[3-(4-phenylpiperazin-1-yl)piperidine-1-carbonyl]-2H-chromen-2-one
7-[(2,3-dimethoxyphenyl)methyl]-2-(4-methylpentanoyl)-2,7-diazaspiro[4.5]decan-6-one
N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
2-{4-[(2-chloro-3,4-dimethoxyphenyl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
5,6-dimethyl-2-(2-{4-[1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl}-2-oxoethyl)-2,3-dihydropyridazin-3-one
6-[(1E)-pent-1-en-1-yl]-2-(pyrrolidin-1-yl)pyrimidin-4-amine
N-(3-{4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-oxopropyl)acetamide
(3R,4R)-4-(azepan-1-yl)-1-[(2,4,5-trimethylphenyl)methyl]piperidin-3-ol
N-[2-(2-phenoxyethoxy)phenyl]-2-(1,2,3,6-tetrahydropyridin-4-yl)acetamide
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
7-[2-(1H-1,2,4-triazol-5-yl)benzoyl]-2,7-diazaspiro[4.5]decane
1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-4-(naphthalen-2-yloxy)piperidine-4-carboxylic acid
2-(pyridin-2-ylsulfanyl)-1-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]propan-1-one
[(1-{1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methyl]urea
2-{1-[(5-methylfuran-2-yl)methyl]-4-[1-(pyridin-2-ylmethyl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
1-(2-ethyl-4-{[1-(1H-imidazol-2-yl)ethyl]amino}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl)-2-methoxyethan-1-one
3-fluoro-N-(1-{1-[(methylcarbamoyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide