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(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)(methyl)(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amine
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-1-(4-fluorophenyl)cyclopropane-1-carboxamide
2-(3-{[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-1-yl]methyl}phenoxy)ethan-1-ol
5-[(5-cyclopropyl-4-phenyl-1H-imidazol-1-yl)methyl]-2-(trifluoromethyl)pyridine
4-{1-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]propyl}morpholine
8-[2-(1H-1,3-benzodiazol-2-ylmethoxy)acetyl]-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one
(3S,4R)-1-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
[3-(cyclopropylmethyl)-1-[4-methyl-6-(methylamino)pyrimidin-2-yl]piperidin-3-yl]methanol
6-[(3-methoxyphenyl)methoxy]-4-[(2S)-5-oxopyrrolidine-2-carbonyl]-1-(2-phenylethyl)-1,4-diazepan-2-one
2-[4-hydroxy-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-1-yl]-2-oxo-N-phenylacetamide
N-[(1S)-1-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl]acetamide
1'-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
N-[3-(5-chloro-1H-1,3-benzodiazol-2-yl)propyl]-1-ethyl-3-methylpiperidine-3-carboxamide
(2E)-1-[(4aR,8aS)-6-[2-(thiophen-2-yl)acetyl]-decahydro-1,6-naphthyridin-1-yl]-3-(2,5-difluorophenyl)prop-2-en-1-one
8-fluoro-N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]quinoline-2-carboxamide
1-{2-[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]ethyl}pyrrolidin-2-one
1-[1,3-dioxo-2-(1,3-thiazol-2-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N,N-bis(prop-2-en-1-yl)piperidine-3-carboxamide
N-(1-{4-[(4-cyclopentyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}-1-oxopentan-2-yl)acetamide
{1-[1-(thian-4-yl)piperidin-3-yl]piperidin-4-yl}methanol
2-{1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-4-yl}-1-methyl-1H-1,3-benzodiazole
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N,3,5-trimethyl-1,2-oxazole-4-sulfonamide
N-[1-(4-cyclopentyl-4H-1,2,4-triazol-3-yl)ethyl]-3-ethyl-5-methyl-1,2-oxazole-4-carboxamide
3,7-dimethyl-8-{2-oxa-7-azaspiro[4.5]decan-7-yl}-2,3,6,7-tetrahydro-1H-purine-2,6-dione
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]piperazine
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
7-(2-methoxyethyl)-2-[3-(pyridin-2-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
N-cyclopentyl-1-[(4-methoxyphenyl)methyl]-5-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-(2-methoxyphenyl)-1-[7-(2-methylphenyl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-1-one
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-methanesulfonyl-3-{[2-(6-methyl-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]methyl}piperidine
1-[2-({2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}amino)pyrimidin-4-yl]piperidin-4-ol
3-(5-tert-butyl-1,3,4-thiadiazol-2-yl)-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]urea
N-[2-oxo-4-(quinoxalin-2-yl)-1,2,3,4-tetrahydroquinolin-7-yl]methanesulfonamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-{3-oxo-3-[2-oxo-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-8-yl]propyl}acetamide
2-(4-benzyl-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N-methylacetamide
4-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]butanamide
2-({[(3R,4R)-4-(hydroxymethyl)-1-[(2-methoxy-3,5-dimethylphenyl)methyl]pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-[2-(dimethylamino)ethyl]-N-methyl-3-({1-[3-(1H-pyrazol-1-yl)propanoyl]piperidin-4-yl}oxy)benzamide
6-(benzyloxy)-4-[2-(methylsulfanyl)acetyl]-1-[3-(2-oxopyrrolidin-1-yl)propyl]-1,4-diazepan-2-one
N2-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]pyrimidine-2,4-diamine
N-[(3,4-dimethylphenyl)(pyridin-3-yl)methyl]-2-(3-methyl-1,2-oxazol-5-yl)acetamide
3-(1-butyl-1H-imidazol-2-yl)-1-(3,5-difluorobenzoyl)piperidine
4-(2-methylquinolin-4-yl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N,N-dimethyl-5-{methyl[(4-phenyl-1,3-thiazol-2-yl)methyl]amino}-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-{[3-(4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}benzonitrile
N4-(1H-1,3-benzodiazol-2-ylmethyl)-N4-methyl-6-(morpholin-4-yl)pyrimidine-2,4-diamine
N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1-(5-propylpyrimidin-4-yl)piperidin-4-amine
(3R)-1-[(3-methyl-1-phenyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-ol
(2S,4S)-1-{[4-(diethylamino)phenyl]methyl}-N-methyl-4-{[1-(2-phenylethyl)piperidin-4-yl]amino}pyrrolidine-2-carboxamide