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2-[4-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperazin-1-yl]pyridine-3-carboxamide
8-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-2-oxo-2,3-dihydro-1H-imidazole-4-carboxamide
2-[2-(1H-indol-1-yl)acetyl]-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[3-(pyrrolidin-1-yl)propyl]benzamide
methyl 5-oxo-5-(2-{[3-(trifluoromethyl)phenyl]methyl}morpholin-4-yl)pentanoate
2-methyl-4-{[4-(5-methyl-1,3-benzoxazol-2-yl)piperazin-1-yl]methyl}phenol
1-[(3,4-dimethylphenyl)methyl]-4-[3-(ethylsulfanyl)propanoyl]piperazin-2-one
8-(5-ethyl-1,2-oxazole-3-carbonyl)-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
(1S,5R)-6-(cyclopropylmethyl)-3-[(2-methoxynaphthalen-1-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(1-{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)piperidin-3-ol
2-[4-(4-cyclobutaneamidobenzoyl)morpholin-3-yl]acetic acid
butyl 3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carboxylate
7-(3-chlorophenyl)-4-[1-(propan-2-yl)piperidin-4-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(4-hydroxybutyl)-9-[3-(methylsulfanyl)butyl]-2,9-diazaspiro[5.5]undecan-3-one
3-[(4aR,7aS)-4-[(2-methoxy-4-methylphenyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-2-(1-methyl-1H-indol-3-yl)acetamide
methyl 1-[(3R,5S)-5-{[3-(methylsulfanyl)phenyl]carbamoyl}-1-{[4-(propan-2-yl)phenyl]methyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
2-methyl-7-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}-2,7-diazaspiro[4.4]nonane
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
2-(1H-indazol-1-yl)-N-({5-methyl-2-[4-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)acetamide
N-ethyl-3-(1,2-oxazinan-2-yl)-N-[2-(pyridin-2-yl)ethyl]propanamide
3-[(3S)-1-benzylpyrrolidin-3-yl]-1-[3-(2-oxo-1,3-oxazolidin-3-yl)phenyl]urea
(4aS,8aR)-1-(2-phenylethyl)-6-(1H-pyrazole-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
N-{2-[1-(furan-2-ylmethyl)piperidin-3-yl]ethyl}-3-methylbut-2-enamide
2-ethyl-5-{1-[2-(3-methoxyphenyl)ethyl]-1H-imidazol-2-yl}pyrimidine
N-cyclopropyl-3-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}propanamide
6-fluoro-2-({[(1S)-1-(3-methylpyridin-2-yl)ethyl]amino}methyl)quinolin-4-ol
1-cyclohexyl-4-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
methyl({[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl})[1-(pyrimidin-4-yl)ethyl]amine
N-[2-(5-cyano-2-methyl-1H-indol-3-yl)ethyl]-2-cyclopropyl-6-oxo-1,6-dihydropyrimidine-5-carboxamide
{3-[(3-chlorophenyl)methyl]-1-[3-(thiophen-3-yl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}methanol
4-chloro-5-{[3-(3-chlorobenzoyl)piperidin-1-yl]methyl}-N,N-dimethyl-1,3-thiazol-2-amine
3-[(2,3-dimethoxyphenyl)methyl]-5-{1-[2-(3,5-dimethyl-1H-pyrazol-1-yl)acetyl]piperidin-4-yl}-5-methylimidazolidine-2,4-dione
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-(furan-3-carbonyl)piperidin-3-yl]piperazine
2-(2-fluorophenyl)-N-[2-(5-methylpyrazine-2-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]acetamide
N-({5-[(2-fluoro-4-methylphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
4-{[3-(4-tert-butylbenzoyl)piperidin-1-yl]methyl}-2,6-dimethoxyphenol
4-[2-(aminomethyl)-5-fluoro-2,3-dihydro-1-benzofuran-7-yl]-N,N,6-trimethylpyrimidin-2-amine
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-(oxan-4-yl)piperazine
3-[3-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]-6-phenyl-1,2-dihydropyridin-2-one
2-methyl-N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}pyrimidin-4-amine
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
7-fluoro-N,3-dimethyl-N-(quinoxalin-2-ylmethyl)-1-benzofuran-2-carboxamide
methyl 6-(cyclohex-3-ene-1-carbonyl)-2-[(2-methylphenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-(2-methylphenyl)-1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}pyrrolidin-3-ol
N,2-dimethyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-(oxan-4-yl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
3-{[5-(1H-pyrazol-5-yl)furan-2-yl]methyl}-3,9-diazaspiro[5.6]dodecan-10-one
9-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one