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N-(4-fluorophenyl)-4-[5-(4-methoxybenzamido)-1H-pyrazol-1-yl]piperidine-1-carboxamide
1-acetyl-N-[3-(1H-imidazol-1-yl)propyl]-N-(pyridin-4-ylmethyl)piperidine-3-carboxamide
3-[1-(furan-2-carbonyl)piperidin-4-yl]-N-(2-methoxyethyl)propanamide
1-{1-[(4R)-3-methyl-1,3-thiazolidine-4-carbonyl]-4-phenylpiperidin-4-yl}ethan-1-one
3-{3-methyl-5-[3-(pyridin-4-yl)-1H-pyrazol-5-yl]-1H-1,2,4-triazol-1-yl}-1λ6-thiolane-1,1-dione
1-[(1R)-1-(4-methoxyphenyl)ethyl]-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
N-[2-(3-{[methyl(thiophen-2-ylmethyl)amino]methyl}phenoxy)propyl]-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
ethyl(methyl){[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}amine
N-[cyclopropyl(3-methylpyridin-2-yl)methyl]-2-(2,3,6-trimethylphenoxy)acetamide
[(2S)-1-[1-(7-methoxy-4-methylquinazolin-2-yl)piperidine-3-carbonyl]pyrrolidin-2-yl]methanol
(2S,4R)-4-[(4-fluorophenyl)sulfanyl]-1-[(4-methoxyphenyl)methyl]-N-methyl-N-(1,2-oxazol-3-ylmethyl)pyrrolidine-2-carboxamide
N-[1-(2,5-difluorophenyl)cyclopropyl]-1-(2-methoxyacetyl)piperidine-3-carboxamide
3-{1-[2-(2,5-difluorophenyl)acetyl]piperidin-3-yl}benzoic acid
(5S,9aS,9bS)-5-[4-(5-methylfuran-2-yl)phenyl]-2-(pyridin-3-ylmethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-[(3S)-1-[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]pyrrolidin-3-yl]acetamide
1-(1-benzothiophene-5-carbonyl)-2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine
N-[4-(4-{[(3,5-dimethylphenyl)formamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]-5-(methoxymethyl)furan-2-carboxamide
N-[(2R,4R,6S)-2-(4-fluoro-3-methoxyphenyl)-6-(2-methylphenyl)oxan-4-yl]acetamide
2-[3-(1H-imidazol-1-yl)propyl]-9-[3-(1H-pyrazol-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
4-(2,4-dioxoimidazolidin-1-yl)-N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}benzamide
4-benzyl-3-ethyl-1-(4-methyl-1,3-thiazole-5-carbonyl)-1,4-diazepan-5-one
N-(3-cyclopentylpropyl)-2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-N,2,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
7-fluoro-1-methyl-2-(2-methyl-4-phenylpyrimidine-5-carbonyl)-1,2,3,4-tetrahydroisoquinoline
3-[2-(azepan-1-yl)-2-oxoethyl]-3-(2-chlorophenyl)-1-[2-(dimethylamino)ethyl]pyrrolidine-2,5-dione
3-[3-(naphthalene-1-carbonyl)piperidin-1-yl]propanamide
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-[(2-methylphenyl)methyl]acetamide
3-{[ethyl(pyridin-4-ylmethyl)amino]methyl}-N,8-dimethyl-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
2-{1-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}-1,2,3,4-tetrahydroisoquinoline
1-[4-({[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)phenyl]imidazolidin-2-one
(3R,4R)-4-cyclobutyl-3-methyl-1-[2-(methylamino)pyridine-4-carbonyl]piperidin-4-ol
2-{[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}benzoic acid
1-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(3-methyl-1H-pyrazol-1-yl)propan-1-one
N-methyl-3-(1-methyl-1H-pyrazol-4-yl)-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}propanamide
[(1-benzylpyrrolidin-3-yl)methyl](methyl)[2-methyl-2-(morpholin-4-yl)propyl]amine
N-cyclopentyl-N-[(2-methylphenyl)methyl]-2-(pyrrolidin-3-yl)acetamide
N-({3-methoxy-4-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]-3-(2-oxopyrrolidin-1-yl)benzamide
3-(3-hydroxy-3-methylbutyl)-N-[1-(pyrimidin-2-yl)piperidin-3-yl]benzamide
(3aS,6aR)-5-[(3-hydroxyphenyl)methyl]-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
1-cyclopropyl-N-methyl-6-oxo-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}piperidine-3-carboxamide
1-[(3-chlorophenyl)methyl]-4-[1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carbonyl]piperazine
6-(2-cyanophenyl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
1-{2-hydroxy-3-[4-methoxy-2-(thiomorpholin-4-ylmethyl)phenoxy]propyl}piperidin-4-ol
N,1-dimethyl-6-(propan-2-yl)-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N,N-dimethyl-1-(2-methylpropyl)-5-{[2-(4-phenylpiperidin-1-yl)ethyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[(4-fluorophenyl)methyl]-4-(3-{2-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-2-yl}propanoyl)piperazin-2-one
1-methyl-5-(piperidin-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
5-ethyl-5-{1-[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propanoyl]piperidin-4-yl}-3-(2-methylprop-2-en-1-yl)imidazolidine-2,4-dione
3-(1H-1,2,3-benzotriazol-1-yl)-1-[(3S,4S)-3-hydroxy-4-[methyl(propyl)amino]pyrrolidin-1-yl]propan-1-one