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(3R,4R)-3-cyclopropyl-4-methyl-1-[2-(methylamino)pyridine-3-carbonyl]pyrrolidin-3-ol
methyl[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl](4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)amine
[(2,3-dimethyl-1H-indol-5-yl)methyl][1-(methylsulfanyl)propan-2-yl]amine
N-butyl-2-{1-[6-(4-fluorophenyl)imidazo[2,1-b][1,3]thiazol-3-yl]-N-methylformamido}acetamide
N-[(2R,3R)-1'-[2-(2,6-difluorophenyl)acetyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-4-carboxamide
(3R,4S)-1-{4-[(butylsulfanyl)methyl]-5-methylfuran-2-carbonyl}-4-cyclopropylpyrrolidin-3-amine
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-[2-(pyridin-2-yl)ethyl]piperidin-4-amine
4-benzyl-3-ethyl-1-[5-(hydroxymethyl)furan-2-carbonyl]-1,4-diazepan-5-one
(4aR,7aS)-N,N-dimethyl-6,6-dioxo-4-[(5-propylfuran-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
6-chloro-2-(2-cyclopropylpyrimidin-5-yl)-4-(pyrrolidine-1-carbonyl)quinoline
3-{2-[4-(3-chlorophenyl)piperazin-1-yl]-2-oxoethyl}-3-(2-methoxyphenyl)-1-methylpyrrolidine-2,5-dione
[(1-{[2-(cyclopentyloxy)phenyl]methyl}piperidin-3-yl)methyl](methyl)amine
6-[2-(2,3-dihydro-1H-inden-1-yl)acetyl]-2,3-dimethyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
ethyl 4-[1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)piperidin-3-yl]piperazine-1-carboxylate
N'-[4-(2,2-dimethylpropanamido)-3-methoxyphenyl]-N-(2-methylpropyl)ethanediamide
[1-(dimethyl-1,3-thiazol-4-yl)ethyl][(4-methanesulfonylphenyl)methyl]methylamine
(2S,4R)-N-ethyl-1-methyl-4-(4-oxo-4-phenylbutanamido)pyrrolidine-2-carboxamide
methyl 3-(2-phenylacetamido)-5-[(4,5,6,7-tetrahydro-2H-indazol-3-ylformamido)methyl]benzoate
4-[2-(benzyloxy)acetyl]-1-[(2-fluorophenyl)methyl]piperazin-2-one
4-(2-methoxyethoxy)-1-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}piperidine
methyl({[3-(1H-pyrazol-1-yl)phenyl]methyl})({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)amine
2-{4-[2-(furan-2-yl)azepane-1-carbonyl]-1H-1,2,3-triazol-1-yl}ethan-1-amine
5-(2-{2-[(5-acetylpyridin-2-yl)amino]ethyl}morpholin-4-yl)-2-methyl-2,3-dihydropyridazin-3-one
N,1,3-trimethyl-N-[2-(morpholin-4-yl)propyl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-ethyl-5-[1-(3-fluorobenzoyl)piperidin-4-yl]-3-(2-methylprop-2-en-1-yl)imidazolidine-2,4-dione
(2R)-2,5-diamino-1-{4-[4-(propan-2-yl)-6-(trifluoromethyl)pyrimidin-2-yl]piperazin-1-yl}pentan-1-one
N-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-fluoro-4-methylbenzamide
(2R)-2-amino-N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)propanamide
5-{2-[4-(cyclopropylmethyl)-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl]ethyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
ethyl 3-[(2,4-difluorophenyl)methyl]-1-(pyridin-4-ylmethyl)piperidine-3-carboxylate
9-methoxy-3-[2-(3-methylphenyl)acetyl]-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-{2-[7-(cyclohexylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-4-fluorobenzamide
{[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}({[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl})amine
(2H-1,3-benzodioxol-5-ylmethyl)[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]amine
N-{[4-(aminomethyl)phenyl]methyl}-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
2-{5-[4-(3-chloropyridin-2-yl)piperazine-1-carbonyl]-1H-pyrazol-3-yl}phenol
methyl 3-(2,5-dimethylfuran-3-carbonyl)-7-oxo-9-(3-phenylpropoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-methyl-7-(2-propyl-1,3-thiazole-4-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
3-(3-hydroxy-3-methylbutyl)-N-methyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]benzamide
3-[2-(3,4-difluorophenyl)ethyl]piperidine
1-(furan-2-ylmethyl)-3-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-1-carbonyl}piperidine
N-cyclopentyl-2-({2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl}amino)propanamide
ethyl 5-[(2,1,3-benzoxadiazol-5-ylmethyl)(methyl)carbamoyl]-1H-imidazole-4-carboxylate
(3R,4R)-1-(3-chloropyridin-2-yl)-4-(hydroxymethyl)piperidin-3-ol
2-methoxy-N-[2-(pyrrolidine-1-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]benzamide
1-[2-methyl-6-(piperidin-3-yl)pyrimidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
5-{1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-5-[(3-methoxyphenyl)methyl]-3-methylimidazolidine-2,4-dione
N-[(3S,7S,8aS)-3-(4-aminobutyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-phenyl-5-(trifluoromethyl)-1H-pyrazole-4-carboxamide
7-(cyclobutylmethyl)-2-[2-(4H-1,2,4-triazol-4-yl)ethyl]-2,7-diazaspiro[4.5]decan-6-one