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1-(2-ethoxyethyl)-5-(4-ethyl-3,3-dimethylpiperazine-1-carbonyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
5-benzyl-5-{1-[(5-methylthiophen-2-yl)methyl]piperidin-4-yl}-3-[2-(pyridin-2-yl)ethyl]imidazolidine-2,4-dione
5-[(4-chlorophenyl)methyl]-5-{3-[2-(2-methoxyphenyl)pyrrolidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
methyl 1-[(3R,5S)-1-[(2,5-dimethylphenyl)methyl]-5-[4-(4-fluorophenyl)piperazine-1-carbonyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
2-ethyl-N-[(1-hydroxycyclohexyl)methyl]pyrimidine-5-carboxamide
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-1-phenyl-1H-pyrazole-4-carboxamide
2-amino-2-methyl-1-{3-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
5-{2-[2-(2,3-dimethoxyphenyl)-1H-imidazol-1-yl]ethyl}-4-methyl-1,3-thiazole
methyl 5-[(1-benzofuran-2-ylmethyl)amino]-1-ethyl-3-(oxolane-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-(pyridin-3-ylmethyl)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-{[7-(furan-2-ylmethyl)-3-(oxan-4-yl)-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazin-5-yl]methyl}-1H-imidazole
N-cyclopentyl-3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-(prop-2-en-1-yl)propanamide
(2S)-1-[6-(3-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]pyrrolidine-2-carboxamide
N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)-2-(1H-1,2,3,4-tetrazol-1-yl)acetamide
N-[2-(3-{[methyl(thiophen-3-ylmethyl)amino]methyl}phenoxy)propyl]-2-(piperidin-1-yl)acetamide
2-(2H-1,3-benzodioxol-5-yl)-1-[7-(5-chloro-2-methoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-(3-hydroxyadamantan-1-yl)propanamide
2-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decane
(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(3-methoxyphenyl)methyl]-9-oxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
N-[(1R,2S)-2-(methoxymethyl)cyclopentyl]-4-(4-methylphenyl)-5-(pyrimidin-5-yl)pyrimidin-2-amine
methyl 5-(cycloheptylamino)-3-acetamido-1-[2-(4-methoxyphenyl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-(2-methoxyethyl)-1-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)piperidine
2-[4-(4-chlorophenyl)butanamido]-2-(3,5-dimethyl-1H-pyrazol-4-yl)acetic acid
2-(4-methoxy-3-methylphenyl)-5-[(6-methylpyridin-2-yl)methyl]-2,3,4,5-tetrahydro-1,5-benzothiazepine
[(2S,6S)-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
5-[(2-chlorophenyl)methyl]-5-{1-[4-(morpholin-4-yl)benzoyl]piperidin-4-yl}imidazolidine-2,4-dione
N-[(1-ethylpiperidin-3-yl)methyl]-N-methyl-5-propyl-1,3,4-oxadiazol-2-amine
2-chloro-6-methoxy-4-{[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]methyl}phenol
3-(3,4-dimethyl-1H-pyrazol-5-yl)-1-[7-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-2-yl]propan-1-one
4-(3-propyl-1H-pyrazole-5-carbonyl)-1,4-oxazepane
3-(dimethyl-1H-1,2,4-triazol-1-yl)-N,2-dimethyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]propanamide
N-(1,2-oxazol-3-ylmethyl)-5-[1-(piperidin-1-yl)ethyl]furan-2-carboxamide
3-({[2-(dimethylamino)ethyl](ethyl)carbamoyl}methyl)-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
2-ethoxy-3-[3-(2-ethylphenoxy)azetidine-1-carbonyl]pyridine
methyl({[5-(oxan-2-yl)furan-2-yl]methyl}){[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}amine
4-({3-[2-(3-methoxyphenyl)ethyl]piperidin-1-yl}methyl)pyridine
2-(5-{3-[1-(dimethylamino)ethyl]phenyl}-4-phenyl-1H-imidazol-1-yl)acetamide
5-acetyl-N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]thiophene-3-carboxamide
(4aR,7aS)-1-methyl-4-(1-methyl-2-oxo-1,2-dihydroquinoline-4-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[5-(2-fluorophenyl)-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-1-yl]butan-2-ol
1-benzyl-N,N-dimethyl-5-{[3-(propan-2-yloxy)propyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-{[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]sulfonyl}azepane
4-[(2-methylphenyl)methyl]-1-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1,4-diazepan-5-one
5-{[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]methyl}-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
({5-[1-(1-benzofuran-2-ylmethyl)piperidin-4-yl]-4-cyclopropyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
(1R,5R)-3-(dimethylsulfamoyl)-N-methyl-N-phenyl-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
7-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one