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1-(2-{4-azaspiro[2.5]octan-4-ylmethyl}-5-methoxyphenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
1-(5-chloro-3-methyl-1H-indole-2-carbonyl)-N-(1-methoxypropan-2-yl)piperidine-4-carboxamide
N-cyclopropyl-3-{1-[3-(prop-2-en-1-yloxy)benzoyl]piperidin-4-yl}propanamide
1-(azocan-1-yl)-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propan-1-one
[5-(1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}-1H-imidazol-2-yl)furan-2-yl]methanol
7-[(2,3-dimethoxyphenyl)methyl]-2-[2-(dimethylamino)acetyl]-2,7-diazaspiro[4.5]decan-6-one
4-hydroxy-N-[(1R,2S)-2-phenylcyclopropyl]-2-[(phenylsulfanyl)methyl]pyrimidine-5-carboxamide
2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[3-(1H-pyrazol-1-yl)propyl]acetamide
methyl (2S,4R)-1-methyl-4-{5-[(4-methylpiperidin-1-yl)methyl]furan-2-amido}pyrrolidine-2-carboxylate
6-(pyrrolidin-1-yl)-N-[1-(1,3-thiazol-2-yl)ethyl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
(1R,3S)-7-(1H-imidazol-2-ylmethyl)-7-azaspiro[3.5]nonane-1,3-diol
N-[(1S,2S)-2-[(4-fluorophenyl)methyl]cyclopentyl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
3-ethyl-5-{[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1H-pyrazole
3-(1-methyl-1H-pyrazol-4-yl)-1-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
2-(2,5-dioxoimidazolidin-4-yl)-N-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]acetamide
(2R,3R)-1'-(6-chloropyridazin-3-yl)-3-(1H-imidazol-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
4-{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}thiomorpholine
1-(morpholin-4-yl)-3-{1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-yl}propan-1-one
5-(methoxymethyl)-N-{[4-(2-methylpropoxy)phenyl]methyl}-N-(pyridin-4-ylmethyl)furan-2-carboxamide
3-(5-methylfuran-2-yl)-N-[2-(5-methylthiophen-2-yl)ethyl]-1H-pyrazole-5-carboxamide
6-(aminomethyl)-2-(3-phenylpropyl)-3,4-dihydropyrimidin-4-one
N-ethyl-2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}benzamide
2-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]quinoline
3-[5-(benzylsulfanyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-[(3-methoxyphenyl)methyl]piperidine
2-cyclopropyl-4-phenyl-9-(1H-pyrrole-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-2-[1-(3-methoxypropyl)-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]acetamide
2-[2-(3-fluorobenzoyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl]-6-methylpyridine
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N-methyl-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-amine
2-methyl-N-[(2-methylphenyl)methyl]-4-oxo-N-(prop-2-en-1-yl)pentanamide
1-methyl-3-(2-methylpropyl)-8-(1,3-thiazol-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
[(3R,4R)-1-(2-chlorobenzoyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
5-{2-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]-2-oxoethyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-7-fluoro-1,2-dihydroquinolin-2-one
(1R,2R,3R,4S)-N-cyclopropyl-3-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]bicyclo[2.2.1]hept-5-ene-2-carboxamide
5-(4-fluorophenyl)-7-{octahydropyrrolo[1,2-a]piperazin-2-yl}pyrazolo[1,5-a]pyrimidine
3-methoxy-1-(2-oxo-2-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethyl)-1,2-dihydropyridin-2-one
N-(2-methanesulfonylethyl)-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
N-benzyl-3-{[1-(thian-4-yl)piperidin-4-yl]oxy}benzamide
2-(3-fluoro-4-hydroxyphenyl)-1-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
2-cyclooctyl-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decane
5-({methyl[(3-{2-[4-(2-methylpropanoyl)piperazin-1-yl]ethoxy}phenyl)methyl]amino}methyl)pyrrolidin-2-one
N-[(2-aminopyrimidin-5-yl)methyl]-N-methyl-2-[(quinolin-6-yloxy)methyl]-1,3-oxazole-4-carboxamide
6-{[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-methyl-5-phenyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1,2,4-oxadiazol-3-amine
2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]-N-[3-(1H-pyrazol-1-yl)propyl]acetamide
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
1-(cyclopropylmethyl)-5-{4H-thieno[3,2-b]pyrrole-5-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
3-({7-[(1-ethyl-1H-pyrazol-4-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)pyridine
1-[({[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}amino)methyl]-N,N-dimethylcyclohexan-1-amine
6-chloro-N-ethyl-N-(pyridin-4-ylmethyl)-2-(pyrimidin-5-yl)quinoline-4-carboxamide