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2-{[5-(3-acetylphenoxymethyl)-1,2-oxazol-3-yl]formamido}-N-(propan-2-yl)acetamide
7-methyl-2-({7-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-2,7-diazaspiro[4.5]decan-6-one
1-(2-aminopyrimidin-4-yl)-N-[2-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
N-[(4-methoxyphenyl)methyl]-1-{4-methyl-6H,7H,8H-cyclopenta[g]quinazolin-2-yl}piperidin-4-amine
(2S)-2-(methoxymethyl)-1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}pyrrolidine
1-{1-[2-(morpholin-4-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}-4-phenylazepane
6-(2-ethoxypyridin-3-yl)-2H-1,3-benzodioxole-5-carboxamide
4-phenyl-3-{1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(2,3-dihydro-1H-inden-2-yl)-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
N-[3-(furan-2-yl)propyl]-4-hydroxy-2-(thiophen-2-yl)pyrimidine-5-carboxamide
N-[(2R,3R)-1'-[(2,3-difluorophenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
5-(1-benzofuran-2-yl)-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-1,2,4-triazin-3-amine
4-(3-hydroxy-3-methylbutyl)-N-methyl-N-(quinoxalin-2-ylmethyl)benzamide
1-[(2,5-dimethoxyphenyl)methyl]-4-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
(2R,6R)-4-[(1-cyclohexyl-1H-imidazol-5-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
(4aR,6R,8aS)-2-(3-chloropyridin-2-yl)-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinoline
3-(1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-2-yl)pyridine
1-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-4-(pyrrolidin-1-ylmethyl)piperidin-4-ol
(3R,4R)-1-(1-benzothiophene-5-carbonyl)-4-ethylpiperidine-3,4-diol
3-[1-(cyclohex-3-en-1-ylmethyl)-1H-pyrazol-5-yl]-1-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]urea
3-(3-hydroxy-3-methylbutyl)-N-(2-methoxyethyl)-N-(1-methylpiperidin-4-yl)benzamide
N-({1-[(2-methyl-1H-imidazol-4-yl)methyl]pyrrolidin-3-yl}methyl)-1H-1,3-benzodiazole-2-carboxamide
2-[1-(3-methylpyridin-4-yl)-1H-pyrazol-4-yl]-4-(pyrrolidine-1-carbonyl)quinoline
N-[2-(1H-imidazol-2-yl)ethyl]-6-methyl-2-(piperidin-1-yl)pyrimidin-4-amine
1-methyl-3-{4-[(methylsulfanyl)methyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
N-[(4-ethylphenyl)methyl]-3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-methylpropanamide
4-{5-[2-(benzyloxy)ethyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1,5-dimethyl-1H-pyrazole
(3S,9aR)-3-[(benzyloxy)methyl]-8-(2,5-difluorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-methoxy-1-[1'-(pyrazin-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
2-{[1-cyclohexyl-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-5-yl]methyl}-6-methyl-2,3-dihydropyridazin-3-one
(3aS,6aS)-5-(3-carbamoylpyridin-2-yl)-2-(cyclopropylmethyl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(3S,4R)-1-{furo[3,2-c]pyridin-4-yl}-4-(hydroxymethyl)piperidin-3-ol
2-methyl-5-[4-(3-methylphenoxy)piperidine-1-carbonyl]-1,4-dihydropyridin-4-one
butyl 2-(dimethylamino)-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carboxylate
N-[3-(3-chlorophenyl)phenyl]-1-[(trimethylpyrazin-2-yl)methyl]piperidine-4-carboxamide
1-{[2-(cycloheptanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-4-methoxypiperidine
6-methoxy-3-({4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}methyl)-1,2-dihydroquinolin-2-one
6-{[methyl(2-methylpropyl)amino]methyl}-N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl](methyl)(3-phenoxypropyl)amine
N-{4-[3-(6-hydroxypyrimidin-4-yl)piperidine-1-carbonyl]phenyl}cyclobutanecarboxamide
5-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]-N,N-dimethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-[5-(5-acetylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]-1-[(1R,3s,6r,8S)-4-azatricyclo[4.3.1.13,8]undecan-4-yl]propan-1-one
5-{[3-(5-fluoro-2-methoxybenzoyl)piperidin-1-yl]methyl}-2-methoxyphenol
1-{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N-ethylpyrrolidine-3-carboxamide
ethyl 1-[3-(dimethylcarbamoyl)propyl]-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylate
2-fluoro-N-[(2S)-1-hydroxy-3-phenylpropan-2-yl]-5-sulfamoylbenzamide
1-{2-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]-2-oxoethyl}piperidine-4-carboxamide
3-(3-hydroxy-3-methylbutyl)-N-[1-(pyridin-4-yl)propan-2-yl]benzamide
3-[1-(2-benzyl-1,3-thiazole-4-carbonyl)pyrrolidin-2-yl]-4-methyl-1,2,5-oxadiazole
methyl 4-(3-{[3-(1H-indol-2-yl)phenyl]carbamoyl}piperidin-1-yl)-4-oxobutanoate