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4-ethyl-3-({1-[(5-propylfuran-2-yl)methyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[4-(1H-1,2,4-triazol-1-yl)butanoyl]piperidin-3-yl}propanamide
(1S,6R)-3-{[5-(1H-1,2,4-triazol-5-ylsulfanyl)furan-2-yl]methyl}-3,9-diazabicyclo[4.2.1]nonane
2-{1-[5-(propan-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl]piperidin-2-yl}pyridine
3-(2,3-difluorophenyl)-5-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
1-[7-(5-chloropyridin-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methoxybutan-1-one
1-methyl-5-[(3-methylbutyl)amino]-N-[2-(morpholin-4-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-benzyl-8-(pyrimidin-4-yl)-2,8-diazaspiro[5.5]undecane
N-{[5-(5-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}oxane-4-carboxamide
1-[(1S,3R)-1-(2-aminoethoxy)-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-2-(5-ethyl-1-benzofuran-3-yl)ethan-1-one
1-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(3-fluorophenoxy)ethan-1-one
N-[(5-methyl-2-{3-[3-(pyridin-3-yl)propanamido]phenyl}-1,3-oxazol-4-yl)methyl]-4-(2-methylpropyl)benzamide
3-methoxy-1-{2-oxo-2-[(2S)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]ethyl}-1,2-dihydropyridin-2-one
2-amino-2-methyl-1-{3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}propan-1-one
N'-(3-chloro-2-methylphenyl)-N-ethyl-N-(4-hydroxybutyl)propanediamide
[(3S,5R)-1-[(5-methylthiophen-2-yl)methyl]-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol
2-(2,4-dichlorophenoxy)-N-(2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)acetamide
N-{3-[(4aS,8aR)-1-(3-hydroxypropyl)-2-oxo-decahydro-1,6-naphthyridin-6-yl]-3-oxopropyl}acetamide
1-[4-({3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}methyl)thiophen-2-yl]ethan-1-one
3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methoxyethyl)-8-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)benzamide
2-[5-(1-methanesulfonylpyrrolidin-2-yl)-3-phenyl-1H-1,2,4-triazol-1-yl]-3-methylpyridine
N-{7-[3-(dimethylamino)pyrrolidine-1-carbonyl]-1-(2-methoxyethyl)-2-(pyridin-2-yl)-1H-1,3-benzodiazol-5-yl}acetamide
14-[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
N-methyl-N-(2-phenyl-1-{1-[3-(1H-1,2,4-triazol-1-yl)propanoyl]piperidin-4-yl}ethyl)thiophene-2-carboxamide
3-{2-[4-(1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}-4-[(5-methylfuran-2-yl)methyl]piperazin-2-one
1-(3-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}phenyl)imidazolidin-2-one
(2S)-2-[2-(2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamido]-3-phenylpropanamide
3-{[3-(2-chlorophenoxy)azetidin-1-yl]methyl}pyridine
N-ethyl-N-methyl-6-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]pyridine-3-carboxamide
5-(2H-1,3-benzodioxol-5-ylmethyl)-3-(3-methoxyphenyl)-1,2,4-oxadiazole
(1r,4r)-4-({[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}amino)cyclohexan-1-ol
N-methyl-N-[(3-methylpyridin-4-yl)methyl]-6-(thiomorpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
5-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-3-propyl-1H-pyrazole
N-{1-[1-(2-methoxybenzoyl)piperidin-4-yl]-2-phenylethyl}-N,1-dimethyl-1H-pyrazole-3-carboxamide
3-(1-{[2-(difluoromethoxy)phenyl]methyl}piperidin-3-yl)-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
N-tert-butyl-2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]acetamide
2-(2-{2-[1-(propan-2-yl)piperidin-4-yl]acetyl}-1,2,3,4-tetrahydroisoquinolin-1-yl)acetic acid
1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}-N-[2-(pyridin-4-yl)ethyl]piperidine-4-carboxamide
2-ethyl-N-({2-[3-(4-methoxybenzenesulfonamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)butanamide
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-5-(5-methylfuran-2-yl)-1,2,4-triazin-3-amine
methyl (1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxylate
N-(3-hydroxy-2,2-dimethylpropyl)-3-[5-(3-phenylpropyl)-1,3,4-oxadiazol-2-yl]propanamide
N-[2-(propan-2-yl)phenyl]-5-(1H-pyrazol-3-yl)furan-2-carboxamide
3-(5-{2-methylimidazo[1,2-a]pyridin-3-yl}-1,2,4-oxadiazol-3-yl)pyridine
3-{[(2-chlorophenyl)formamido]methyl}-N-(2,3-dimethylphenyl)piperidine-1-carboxamide
N-methyl-2-(pyridin-3-yl)-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]acetamide
(3S)-3-[5-(4-fluoro-2-methoxyphenyl)-4-phenyl-1H-imidazol-1-yl]azepan-2-one
N-cyclohexyl-7-(hydroxymethyl)-3,9-diazaspiro[5.5]undecane-3-carboxamide
1-[3-(morpholin-4-yl)propyl]-6-oxo-N-(2-phenylethyl)piperidine-3-carboxamide