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(1S,5R)-3-(pyridin-3-ylmethyl)-6-[(2,3,4-trifluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
4-[(3-methylquinoxalin-2-yl)methyl]-7-(pyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{[7-(4,6-dimethylpyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinan-4-yl]acetamide
2-[3-(pyridin-4-yl)-5-[2-(1H-1,2,3,4-tetrazol-1-yl)ethyl]-1H-1,2,4-triazol-1-yl]ethan-1-ol
methyl (2S)-1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidine-2-carboxylate
2-{3-methyl-5-[3-(pyridin-4-yl)-1H-pyrazol-5-yl]-1H-1,2,4-triazol-1-yl}acetic acid
3-methyl-5-[1-(propan-2-yl)-1H-pyrazol-4-yl]-1H-1,2,4-triazole
N-[(3R,4R)-1-[(1-ethyl-1H-indol-4-yl)methyl]-3-hydroxypiperidin-4-yl]pyridine-4-carboxamide
5-(2,6-difluorophenoxymethyl)-N-[2-(pyridin-3-yloxy)propyl]-1,2-oxazole-3-carboxamide
3-[2-(dimethylamino)-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-N-(3-methylphenyl)-3-oxopropanamide
3-[2-amino-6-(morpholin-4-yl)pyrimidin-4-yl]benzonitrile
N-[1-(2-{4-[hydroxy(thiophen-2-yl)methyl]piperidin-1-yl}-2-oxoethyl)-1H-pyrazol-4-yl]-3-(2-methoxyphenyl)propanamide
(3aR,6aR)-2-(2-methoxyacetyl)-N-methyl-N-(3-methylbutyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
(2S,4S)-1-{[4-(diethylamino)phenyl]methyl}-4-({[4-(dimethylamino)phenyl]methyl}amino)-N-methylpyrrolidine-2-carboxamide
N-(4-{[1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-8-yl]methyl}phenyl)acetamide
1-{2-[4-(4-fluorophenyl)-1,4-diazepane-1-carbonyl]phenyl}ethan-1-one
4-[(2S,4S)-4-amino-1-methylpyrrolidine-2-amido]-N-cyclohexylpiperidine-1-carboxamide
1-methyl-4-[3-(methylsulfanyl)propyl]-2-phenylpiperazine
(3aS,6aS)-2-[6-(2-methylpropyl)-2-oxo-1,2-dihydropyrimidine-4-carbonyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[2-(1,4-dioxo-1,2,3,4-tetrahydrophthalazin-2-yl)ethyl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
4-(4-methoxy-2-methylphenyl)-3-(pyridin-3-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
5-(3-{4-[(4-methoxyphenyl)methyl]-3-oxopiperazin-1-yl}-3-oxopropyl)imidazolidine-2,4-dione
({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)(methyl){[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}amine
3-{2-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-{spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl}propanamide
4-(3,4-dimethoxyphenyl)-3-(1H-imidazol-1-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(4-methyl-1,4-diazepan-1-yl)-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}acetamide
1-[2,2-dimethyl-3-(pyrrolidin-1-yl)propyl]-4-(4-methoxybenzoyl)piperazine
N-ethyl-3-fluoro-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}pyridine-4-carboxamide
(2S,4S,5R)-5-(2-fluorophenyl)-1-methyl-4-(morpholine-4-carbonyl)pyrrolidine-2-carboxylic acid
N-(2-methoxyethyl)-1-(4,6,7-trimethylquinazolin-2-yl)piperidine-4-carboxamide
N-[2-(dimethylamino)ethyl]-3-{[1-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]sulfamoyl}benzamide
7-(1,3-benzothiazol-2-yl)-4-[(2-methyl-1H-imidazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-benzyl-3-[(4-hydroxypiperidin-1-yl)methyl]-N-methylimidazo[1,2-a]pyridine-2-carboxamide
3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-1-(pyridin-2-ylmethyl)urea
N-cyclopropyl-N-{[3-(2-methylpropoxy)phenyl]methyl}-2-(4-oxo-3,4-dihydrophthalazin-1-yl)propanamide
2-[(4-phenylbutyl)amino]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-(1,4-dimethyl-1H-pyrazol-5-yl)-3-{[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}benzamide
5-(3,4-dimethoxyphenyl)-1-(4-methoxyphenyl)-3-methyl-1H,4H-pyrazolo[3,4-d]imidazole
7-(5-chloropyridin-2-yl)-4-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
{1-[(2,4-dimethoxyphenyl)methyl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl}methanol
2-[3-(hydroxymethyl)-3-(2-phenylethyl)piperidin-1-yl]pyridine-4-carbonitrile
methyl (2S,4R)-1-[(3-methylphenyl)methyl]-4-(quinoline-2-amido)pyrrolidine-2-carboxylate
N-(cyclobutylmethyl)-5-[(isoquinolin-5-yloxy)methyl]-N-(oxolan-2-ylmethyl)-1,2-oxazole-3-carboxamide
4-(3-fluorobenzoyl)-7-(2-methylphenyl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(pyridin-3-ylmethyl)-8-(2,2,3-trimethylbut-3-enoyl)-2,8-diazaspiro[5.5]undecan-3-one
5-{[(5-chloropyridin-3-yl)oxy]methyl}-N-cyclopropyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,2-oxazole-3-carboxamide
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-ethyl-5-methoxy-N-(oxolan-2-ylmethyl)benzamide
4-(2-methoxy-2-phenylacetyl)-1-[(4-methoxyphenyl)methyl]piperazin-2-one
1-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}-4-(thiophen-2-yl)butan-1-one
4-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}thiomorpholine