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2-methyl-4-(4-{[3-(2-methylpiperidin-1-yl)azetidin-1-yl]methyl}phenyl)butan-2-ol
2-[(1-hydroxycyclohexyl)methyl]-4-(4-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)-2,3-dihydro-1H-isoindole-1,3-dione
2-methoxy-5-{1-[(4-phenyl-1,3-thiazol-5-yl)methyl]-1H-imidazol-2-yl}phenol
ethyl 2-{1-[5-(3-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]piperidin-2-yl}acetate
N-{2-[(1-cyclopentyl-6-oxopiperidin-3-yl)formamido]ethyl}pyridine-3-carboxamide
(2R)-2-{[6-(aminomethyl)pyrimidin-4-yl]amino}-3-methylbutan-1-ol
3-[5-(2-methylpropyl)-4H-1,2,4-triazol-3-yl]-1-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]urea
N-[(2,6-difluorophenyl)methyl]-1-methyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-methyl-N-(oxolan-3-yl)benzamide
N-[2-(dimethylamino)ethyl]-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)-5-methyl-1,2-oxazole-3-carboxamide
6-[4-(benzenesulfonyl)piperazine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-(1H-1,2,3-benzotriazol-1-yl)-1-[2-(morpholine-4-carbonyl)piperazin-1-yl]propan-1-one
3-(piperidine-1-carbonyl)-N-(pyridin-4-ylmethyl)pyrazine-2-carboxamide
3-(methylsulfamoyl)-N-[3-(methylsulfanyl)phenyl]-5-[(quinolin-8-ylmethyl)amino]benzamide
N-{3-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}-2-(pyridin-3-yloxy)acetamide
1-(4-{4-cyclopropyl-5-[(dimethylamino)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-phenylethan-1-one
N-(3-methanesulfonamido-4-methoxyphenyl)-4-methyl-1,2,3,6-tetrahydropyridine-1-carboxamide
3-{[1-(benzenesulfonyl)pyrrolidin-3-yl]methyl}benzoic acid
1-benzyl-N3-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-N5-ethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
methyl 2-({1,8-dioxa-4,11-diazaspiro[5.6]dodecane-4-carbonyl}amino)benzoate
3-cyclohexyl-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1H-pyrazole-4-carboxamide
2-(1-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-1H-1,2,3-triazol-4-yl)-1H-1,3-benzodiazole
1-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-4-ethylpiperazine-2,3-dione
1-{2-[5-(5-ethylfuran-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}imidazolidin-2-one
1,5-dimethyl-4-{[3-(3-methylthiophene-2-carbonyl)piperidin-1-yl]methyl}-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
(2-{1-[2-chloro-4-(1H-pyrazol-1-yl)benzoyl]piperidin-2-yl}ethyl)dimethylamine
3-(1H-imidazol-4-yl)-2-[2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamido]propanoic acid
2-amino-4-[6-(dimethylamino)pyridin-3-yl]-6-methyl-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
[(4-methyl-1H-imidazol-5-yl)methyl](prop-2-en-1-yl)(pyridin-3-ylmethyl)amine
3-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-1-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]urea
(3R,4R)-3-cyclobutyl-4-methyl-1-[2-(morpholin-4-yl)benzoyl]pyrrolidin-3-ol
{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
3-(3-chloro-1,2-oxazol-5-yl)-1-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]propan-1-one
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(1-methyl-1H-pyrrol-2-yl)-2-oxoacetamide
N-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-4-(3-hydroxy-3-methylbutyl)benzamide
5-tert-butyl-4-[(2-butyl-4-methyl-3-oxopiperazin-1-yl)methyl]furan-2-carboxamide
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-(1-methylpiperidin-4-yl)piperidine
[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl](methyl)[2-(pyridin-2-yl)ethyl]amine
3-(2-methyl-1H-indol-1-yl)-N-[1-(pyridin-3-yl)propyl]propanamide
5-[2-(aminomethyl)-2,3-dihydro-1-benzofuran-7-yl]-N-methylthiophene-2-carboxamide
methyl(pyridin-3-ylmethyl)[2-(quinolin-4-yloxy)hex-5-en-1-yl]amine
4-[2-(3,4-dichlorophenyl)morpholin-4-yl]-N,N-dimethyl-4-oxobutanamide
4-ethyl-2-(piperidin-1-yl)-6-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
1-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}isoquinoline
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-(4-fluoro-3-methylbenzoyl)pyrrolidin-3-yl]methanol
3-[2-(dimethylamino)ethyl]-1-[2-(4-methoxyphenyl)ethyl]-8-(thiolan-3-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]pyrazine-2-carboxamide
1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-3-(3-methyl-1H-pyrazol-1-yl)propan-1-one
3-[3-(hydroxymethyl)phenyl]-5-(pyrrolidine-1-sulfonyl)benzoic acid
5-{[1-(2H-1,3-benzodioxol-5-yl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]methyl}-1,3,4-thiadiazol-2-amine