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N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-1-[(2-fluorophenyl)methyl]-6-oxopiperidine-3-carboxamide
4-(3-hydroxy-3-methylbutyl)-N-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]benzamide
N-butyl-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
5-oxo-1-[4-(propan-2-yl)phenyl]-N-[2-(1H-pyrrol-1-yl)ethyl]pyrrolidine-3-carboxamide
6-methyl-3-({2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}methyl)-1,2-dihydroquinolin-2-one
methyl 3-[(2,4-dimethylphenyl)methyl]-7-oxo-9-[2-(2-oxopyrrolidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-chloro-N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
2,6-dimethyl-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)pyrimidine-4-carboxamide
3-(azepane-1-carbonyl)-5-[4-(2,3-dimethylphenyl)piperazine-1-carbonyl]-1-(2-methylpropyl)-1,4-dihydropyridin-4-one
N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-3-oxo-3,4-dihydro-2H-1,4-benzoxazine-7-carboxamide
5-benzamido-1-cyclopentyl-N-[3-(1H-pyrazol-1-yl)propyl]-1H-1,3-benzodiazole-7-carboxamide
3-[(2R,3R,6R)-5-(4-methyl-1H-imidazole-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
2-[(adamantan-1-ylmethyl)({[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]ethan-1-ol
1-methyl-4-(5-{3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)piperazin-2-one
N-(2-chloro-6-methylphenyl)-3-(4-phenylpiperazin-1-yl)piperidine-1-carboxamide
1-[2-(4-methoxyphenyl)ethyl]-N-methyl-6-oxo-N-(2-phenoxyethyl)piperidine-3-carboxamide
4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-(3-methylbutyl)benzamide
5-{[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]methyl}-2-(furan-2-yl)pyrimidine
2-{4-[(4-fluoro-3-methoxyphenyl)methyl]-1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-2-yl}ethan-1-ol
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-methyl-N-[(5-methylfuran-2-yl)methyl]-1H-pyrazole-3-carboxamide
(3R,5S)-N-cyclopentyl-5-(3-fluorophenoxymethyl)-1-(naphthalen-2-ylmethyl)piperidine-3-carboxamide
N-[2-(2,5-dimethylphenyl)ethyl]-6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
5-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]-1-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[3-(pentan-3-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-1-one
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}acetamide
ethyl 5-(3-methoxy-3-oxopropyl)-1-[2-(4-methoxyphenyl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-[3-({3-[2-(hydroxymethyl)-2,5-dihydro-1H-pyrrole-1-carbonyl]-1H-pyrazol-5-yl}methoxy)phenyl]ethan-1-one
N-(1-{7-[(2E)-3-(4-hydroxy-3-methoxyphenyl)prop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)pyridine-2-carboxamide
1-[3-(naphthalene-2-carbonyl)piperidin-1-yl]but-3-en-1-one
1-{1-[(2-methylfuran-3-yl)methyl]piperidin-4-yl}piperidin-3-ol
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-2-(2-methyl-1,3-thiazol-4-yl)acetamide
7-{[4-(propan-2-yl)phenyl]methyl}-2-(thiophene-2-carbonyl)-2,7-diazaspiro[4.5]decane
1-(4-{[(2-methylpropyl)(pyridin-2-ylmethyl)amino]methyl}phenyl)ethan-1-one
4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-[3-(methylsulfanyl)propyl]piperidine
5-[(2-fluorophenyl)methyl]-5-{1-[2-(3-methylphenyl)acetyl]piperidin-4-yl}imidazolidine-2,4-dione
(1R,2S,4R)-N-[2-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]bicyclo[2.2.1]hept-5-ene-2-carboxamide
2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[4-(2-methoxybenzoyl)piperazin-1-yl]ethan-1-one
2-(3-methoxypropyl)-8-(4-methylpyridine-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
methyl (2S)-2-({1-[4-(2,4-dimethylbenzamido)phenyl]piperidin-4-yl}amino)-3-phenylpropanoate
3-butyl-4-[3-(difluoromethoxy)benzoyl]-1-methylpiperazin-2-one
2-(4-{4-[(propan-2-yl)amino]pyrimidin-2-yl}-1-(thiophen-2-ylmethyl)piperazin-2-yl)ethan-1-ol
4-{[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}morpholine
1-(4-{[(2,3-dimethyl-1H-indol-5-yl)methyl]amino}piperidin-1-yl)ethan-1-one
5-[4-(3,4-dichlorophenyl)piperazine-1-carbonyl]-N-methylpyrimidin-2-amine
N-[cyclopropyl(6-methylpyridin-2-yl)methyl]-3-(2-oxopiperidin-1-yl)propanamide
9-[3-(1H-imidazol-1-yl)propyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-[(4-{2-[4-(methylsulfanyl)phenyl]-1H-imidazol-1-yl}piperidin-1-yl)methyl]pyridine
N-(1-{1-[(5-cyclopentylthiophen-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-phenylacetamide
8-fluoro-2-({4-[2-(2-hydroxyethoxy)ethyl]piperazin-1-yl}methyl)quinolin-4-ol
(2S,4S)-1-[(3-chlorophenyl)methyl]-4-{[(2,6-difluorophenyl)methyl]amino}-N-[2-(2-fluorophenyl)ethyl]pyrrolidine-2-carboxamide