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{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}[2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl]amine
1-[(2-chloro-3,4-dimethoxyphenyl)methyl]-3-propylpiperidine-3-carboxylic acid
1-(4-methyl-3-phenylpiperazin-1-yl)-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butan-1-one
methyl({[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})(oxan-2-ylmethyl)amine
3,5-dimethyl-4-{1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl}-1,2-oxazole
3-[(1-methanesulfonylpyrrolidin-3-yl)methyl]benzoic acid
ethyl 1-[(6-methoxy-2H-chromen-3-yl)methyl]-4-[(3-methoxyphenyl)methyl]piperidine-4-carboxylate
N-(4-{2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidine-1-carbonyl}phenyl)cyclobutanecarboxamide
N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-2,3-dihydro-1H-indene-5-carboxamide
N-[3-(1H-pyrazol-1-yl)phenyl]quinoxaline-6-carboxamide
1-[cyclohexyl(methyl)amino]-3-(2-methoxy-4-{[methyl(pyrazin-2-ylmethyl)amino]methyl}phenoxy)propan-2-ol
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
4-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidine
N,5,6-trimethyl-N-{[2-(2-methylpropoxy)phenyl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
2-[(4-fluorophenyl)methyl]-4-[2-(methylsulfanyl)pyridine-3-carbonyl]morpholine
N,2-dimethyl-N-(2-phenyl-1-{1-[3-(prop-2-en-1-yloxy)benzoyl]piperidin-4-yl}ethyl)furan-3-carboxamide
1-(pyrimidin-2-yl)-N-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-4-amine
N-{1-[2-(2-benzyl-3-oxopiperazin-1-yl)-2-oxoethyl]-1H-pyrazol-4-yl}-2-(phenylsulfanyl)acetamide
[1-(adamantane-1-carbonyl)-3-[(4-fluorophenyl)methyl]piperidin-3-yl]methanol
N-(2-phenylethyl)-N-(pyridin-3-ylmethyl)-2-(1H-1,2,4-triazol-3-yl)benzamide
5-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-({1-[(2-fluoro-5-methoxyphenyl)methyl]piperidin-3-yl}methyl)thiophene-2-carboxamide
4-methyl-3-(2-oxoimidazolidin-1-yl)-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]benzamide
3-(4-fluorophenyl)-3-[2-(2,4,7-trimethyl-1H-indol-3-yl)acetamido]propanoic acid
2-({2-oxo-3-oxatricyclo[7.3.1.05,13]trideca-1(12),5(13),6,8,10-pentaen-8-yl}methyl)-5-(piperidin-1-yl)-2,3-dihydropyridazin-3-one
(3S,4R)-1-[1-(benzenesulfonyl)cyclopropanecarbonyl]-3-ethyl-4-methylpiperidin-4-ol
1-(pyridin-3-ylmethyl)-N-[4-(pyridin-3-yloxy)phenyl]piperidine-4-carboxamide
1-[1-methyl-3-(pyridin-3-yl)-1H-pyrazol-5-yl]-3-[2-(N-methylmethanesulfonamido)ethyl]urea
N-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-4-(1H-pyrazol-3-yl)benzamide
N-{2-[methyl(phenyl)amino]ethyl}-2-(pyridin-3-yl)pyrimidine-5-carboxamide
4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]-1-(thiolan-3-yl)piperidine
N-[2-(2,3-dimethoxyphenyl)ethyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(1R,5S,6S)-6-[4-(2-methylphenyl)-1,4-diazepane-1-carbonyl]-3-azabicyclo[3.1.0]hexane
2-{[4-(adamantan-2-yl)piperazin-1-yl]methyl}-4-(pyridin-2-yl)phenol
2-(3-methylbutyl)-8-[2-(methylsulfanyl)pyridine-3-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
5-[1-(5-methylthiophene-2-carbonyl)piperidin-4-yl]-3-(oxolan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
N-[1-(1-{[4-(cyclopentyloxy)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]pyridine-3-carboxamide
3-{2-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-5-oxo-1-(prop-2-en-1-yl)pyrrolidine-3-carboxamide
2-(furan-2-yl)-1-{1,3,6-trimethyl-1H-pyrazolo[3,4-b]pyridine-4-carbonyl}pyrrolidine
2-(5-methyl-1,2-oxazol-3-yl)-1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)piperidine
2-acetyl-7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-6-one
N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}oxane-4-carboxamide
1-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-propyl-1H-1,2,4-triazole
N-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-amine
(4aR,8aR)-2-methanesulfonyl-7-[(5-propylfuran-2-yl)methyl]-decahydro-2,7-naphthyridin-4a-ol
6-{3-oxo-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-9-yl}pyridine-2-carbonitrile
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-1-(2-hydroxyethyl)piperidine-4-carboxamide
N-[2-(azepane-1-carbonyl)phenyl]-2-(1H-1,2,3,4-tetrazol-1-yl)acetamide
ethyl 1-(2-amino-6-methylpyrimidine-4-carbonyl)-4-(3-phenylpropyl)piperidine-4-carboxylate