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2-amino-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-6-(3-methyl-1-propyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
1-(4-{[4-(hydroxymethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-2-(1H-indazol-1-yl)ethan-1-one
{[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl}(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
4-{3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}-6-(propan-2-yl)pyrimidin-2-amine
2-[(1,4-dioxan-2-ylmethyl)(methyl)amino]-6-(2-methoxyphenyl)-N-{[1-(morpholin-4-yl)cycloheptyl]methyl}pyridine-3-carboxamide
1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-2-{[6-(pyrrolidin-1-yl)pyridazin-3-yl]oxy}ethan-1-one
6-amino-2-[2-({1,9-dioxaspiro[5.5]undecan-4-yl}amino)ethyl]pyrimidin-4-ol
4-[(2,6-difluorophenyl)methyl]-9-methoxy-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-{methyl[1-(pyrimidin-4-yl)ethyl]sulfamoyl}-N-(2-methylpropyl)benzamide
N-(1,1-dioxo-1λ6-thiolan-3-yl)-1-methyl-3-(2-methylpropyl)-N-(prop-2-en-1-yl)-1H-pyrazole-5-carboxamide
4-(2-amino-5,6,7,8-tetrahydroquinazoline-4-carbonyl)-1-(3-chlorophenyl)piperazin-2-one
N-(furan-2-ylmethyl)-N-(3-methylbutan-2-yl)pyrazolo[1,5-a]pyridine-3-carboxamide
2-(2-methoxyethyl)-8-(1H-pyrrole-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
3-({[5-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-3-yl]methyl}amino)-N-(1,3-thiazol-2-yl)propanamide
3-(furan-2-yl)-6-(trifluoromethyl)-[1,2,4]triazolo[4,3-a]pyridine
6-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]pyridine-3-carboxylic acid
4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]butanamide
1-(pyridin-4-ylmethyl)-4-{1H-pyrrolo[2,3-b]pyridin-6-yl}-1,4-diazepane
(1-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}-3-(3-phenylpropyl)piperidin-3-yl)methanol
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-(1-ethyl-1H-pyrazole-3-carbonyl)pyrrolidine-3-carboxylic acid
N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
1-{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}-4-(pyrrolidine-1-carbonyl)piperidine
1-[1-(3-methylbut-2-en-1-yl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
7-[5-(4-methoxyphenyl)furan-2-carbonyl]-2-oxa-7-azaspiro[4.5]decane
1-(2-methoxyphenyl)-5-oxo-N-[2-(pyridin-4-yl)ethyl]pyrrolidine-3-carboxamide
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[3-(3-methoxyphenoxymethyl)piperidin-1-yl]ethan-1-one
N-{[3-(propan-2-yl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}thiophene-2-sulfonamide
5-(4-cyclopentyl-1,4-diazepane-1-carbonyl)-1-[(3-methoxyphenyl)methyl]piperidin-2-one
N-{[5-methyl-2-(2-phenylmethanesulfonamidophenyl)-1,3-oxazol-4-yl]methyl}-3-(1H-pyrazol-1-yl)propanamide
1-(1H-imidazol-4-ylmethyl)-4-(1H-pyrrole-2-carbonyl)-1,4-diazepane-6-carboxylic acid
2-oxo-2-[4-oxo-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-N-phenylacetamide
3-(2-methoxyethyl)-5-[(4-methyl-1H-pyrazol-1-yl)methyl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
4-[1-(4-fluorophenyl)cyclopropanecarbonyl]-1-(4-methylphenyl)piperazin-2-one
(1-{[4-(cyclopentyloxy)phenyl]methyl}-3-(2-methoxyethyl)piperidin-3-yl)methanol
N-(3-{4-[(2-cyclohexylacetamido)methyl]-5-methyl-1,3-oxazol-2-yl}phenyl)-2-methoxyacetamide
3-{5-benzyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1-(morpholin-4-yl)propan-1-one
(1R,2R)-1-(2-methyl-1,3-benzoxazol-5-yl)-2,3-dihydro-1H-inden-2-ol
1-(2-aminoethyl)-N-methyl-N-[3-(pyrrolidin-1-yl)butyl]-1H-1,2,3-triazole-4-carboxamide
1-(7-chloro-3,5-dimethyl-1-benzofuran-2-carbonyl)-4-(furan-2-carbonyl)piperazine
methyl 2-hydroxy-5-[1-(3-hydroxypropyl)-4-phenyl-1H-imidazol-5-yl]benzoate
(3S,4R)-1-(1-tert-butyl-1H-pyrrole-3-carbonyl)-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[(3,4-dimethoxyphenyl)methyl]-N-methylpropanamide
(5S,9aS,9bS)-5-(2,1,3-benzoxadiazol-4-yl)-2-[(3-chlorophenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-({8-[(3,5-dimethylphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-2-methoxyacetamide
4-methyl-N-(3-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)-1H-imidazole-5-carboxamide
1-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-3-(furan-2-yl)propan-1-one
5-{4-[(3,5-difluorophenyl)methyl]piperazin-1-yl}-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
(2S,4S)-N-ethyl-4-(2-methoxyacetamido)-1-[(3-methylthiophen-2-yl)methyl]pyrrolidine-2-carboxamide