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N-[cyclopropyl(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-3-(1H-pyrazol-1-yl)benzamide
2-amino-6-(2,6-difluorophenyl)-4-[1-(2-hydroxyethyl)-3,5-dimethyl-1H-pyrazol-4-yl]pyridine-3-carbonitrile
1-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carbonyl}spiro[azepane-4,2'-chromene]
N-{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}-N-(prop-2-yn-1-yl)cyclohexanamine
1-(9H-purin-6-yl)-N-[1-(pyrazin-2-yl)propan-2-yl]piperidin-4-amine
(3S)-3-({[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}amino)azepan-2-one
3-[1-(carbamoylmethyl)-4-phenyl-1H-imidazol-5-yl]-5-methyl-1H-indole-2-carboxylic acid
4-(2,2-dimethyloxane-4-carbonyl)-9-methoxy-7-(8-methoxy-4-methylquinolin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-{[(2-ethoxypropyl)(methyl)amino]methyl}-6-methylquinolin-4-ol
5-[1-(3,4-dimethylbenzoyl)piperidin-4-yl]-5-[(3-fluorophenyl)methyl]-3-(2-methoxyethyl)imidazolidine-2,4-dione
6-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}-2-(2-hydroxyethyl)-1H,2H,3H,4H,5H,6H,7H-pyrazolo[3,4-c]pyridin-3-one
2-(4-{[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]methyl}phenoxy)acetic acid
5-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-1,2-dihydropyridin-2-one
[(3-{2-[4-(2-methoxybenzoyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)(naphthalen-1-ylmethyl)amine
1-[2-(benzenesulfonyl)ethyl]-4-methyl-1,4-diazepan-6-ol
5-methyl-2-{4-[(1-methylpiperidin-3-yl)methyl]piperazin-1-yl}pyrimidine
(3aR,6aS)-5-(2-cyclopropylpyrimidine-5-carbonyl)-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
[(1R,3S,3aS,6aR)-1-ethyl-3-(3-fluoro-4-methylphenyl)-5-phenyl-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
3-[2-oxo-2-(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)ethyl]-4-(2-phenylethyl)piperazin-2-one
6-tert-butyl-3-[1-(pyrazin-2-yl)propan-2-yl]-3H,4H-thieno[3,2-d]pyrimidin-4-one
N-(4-methoxyphenyl)-1-(thiophene-2-carbonyl)piperidin-3-amine
4-(6-chloro-2H-1,3-benzodioxol-5-yl)-1-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]-1H-1,2,3-triazole
1-{1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carbonyl}-2-(2-methylphenyl)pyrrolidine
{1-ethyl-5-[(8-methoxyquinolin-2-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}methanol
3-methoxy-5-methyl-N-[2-(1-methylpyrrolidin-2-yl)ethyl]thiophene-2-carboxamide
8-[3-(propan-2-yl)-5-[6-(4H-1,2,4-triazol-4-yl)pyridin-2-yl]-1H-1,2,4-triazol-1-yl]quinoline
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-1-ethylpiperidine-4-carboxamide
3-[N-benzyl-1-(6-methoxy-3-methyl-1-benzofuran-2-yl)formamido]propanamide
N-{4-[({[2-(piperidin-1-yl)-2,3-dihydro-1H-inden-2-yl]methyl}amino)methyl]phenyl}acetamide
N-[2-hydroxy-2-(3-methoxyphenyl)ethyl]-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
N-{[7-(cyclohex-3-ene-1-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-5-ethyl-1,2-oxazole-3-carboxamide
8-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-1-oxa-8-azaspiro[4.6]undecan-9-one
2-[1-(1-methylpiperidin-4-yl)-4-{[4-(trifluoromethyl)phenyl]methyl}piperazin-2-yl]ethan-1-ol
{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amine
N-({4-hydroxy-1-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]azepan-4-yl}methyl)piperidine-1-carboxamide
2-(4-methylpentyl)-4-[(6-methylpyridin-2-yl)methyl]morpholine
1-{4-[4-(2-methylphenoxy)piperidine-1-carbonyl]phenyl}pyrrolidin-2-one
{2-[2-(propan-2-yloxy)phenyl]-1,3-thiazol-4-yl}methanol
N-(furan-2-ylmethyl)-1-(4-methyl-3-phenyl-1H-pyrazole-5-carbonyl)piperidine-4-carboxamide
{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}(1-methoxybutan-2-yl)amine
(5-{1-[2-(phenylamino)ethyl]-1H-1,2,3-triazol-4-yl}furan-2-yl)methanol
2-[3-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]pyrimidine
2-methyl-6-(2-{[1-(3-methylphenyl)propan-2-yl]amino}ethyl)-3,4-dihydropyrimidin-4-one
2-{2-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-2-oxoethyl}-5,6-dimethyl-2,3-dihydropyridazin-3-one
N-{2-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}pyridine-2-carboxamide
(3R,5S)-N3-(4-fluorophenyl)-1-(2-methylpropyl)-N5-(naphthalen-1-ylmethyl)piperidine-3,5-dicarboxamide
(4aS,8aR)-6-[(2E)-hex-2-en-1-yl]-1-(4-hydroxybutyl)-decahydro-1,6-naphthyridin-2-one
(2S,4S)-4-amino-N,N-diethyl-1-(6-oxo-1,6-dihydropyridine-3-carbonyl)pyrrolidine-2-carboxamide
{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}({2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl})amine
N-[(2-chloropyridin-3-yl)methyl]-N-methyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide