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3-[N-(propan-2-yl)-1-[2-(pyridin-3-yl)pyrimidin-5-yl]formamido]propanamide
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-1-(furan-2-ylmethyl)piperidine-3-carboxamide
(3aS,6aS)-2-(dimethylcarbamoyl)-5-[2-(1H-indol-3-yl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-cyclohexyl-5-(2,6-dimethoxyphenyl)furan-2-carboxamide
1-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]piperidine
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methyl-1-phenyl-1H-pyrazole-4-carboxamide
1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-3-(naphthalene-2-carbonyl)piperidine
1-methyl-5-[4-(2-propoxyethyl)piperazine-1-carbonyl]-1,2-dihydropyridin-2-one
3-(1-{2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxybenzoyl}piperidin-2-yl)propan-1-ol
3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(4,6-dimethylpyrimidin-2-yl)methyl]benzamide
N-[(6-methylpyridin-2-yl)methyl]-3-(1-phenylethyl)-1,2-oxazole-5-carboxamide
2-(3-methyl-4-{[3-(1-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}-1H-pyrazol-1-yl)ethan-1-ol
6-(cyclopropylmethoxy)-1-[(3-methoxyphenyl)methyl]-4-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]-1,4-diazepan-2-one
3-(2-methoxybenzoyl)-1-[3-(prop-2-en-1-yloxy)benzoyl]piperidine
3-[5-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
5-({3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}methyl)-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
3-[2-(4-cyclohexylpiperazin-1-yl)-2-oxoethyl]-3-phenyl-1-(pyridin-4-ylmethyl)pyrrolidine-2,5-dione
1-cyclopentyl-4-[({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)methyl]pyrrolidin-2-one
1-(4-methoxyphenyl)-4-[3-(2-methoxyphenyl)propanoyl]-6,6-dimethylpiperazin-2-one
N-({8-[(4-phenylphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)furan-2-carboxamide
1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-3-methyl-2-phenylbutan-1-one
1-(4-ethylpiperazin-1-yl)-3-(2-methoxy-4-{[methyl(oxan-4-yl)amino]methyl}phenoxy)propan-2-ol
5-cyclobutanecarbonyl-1'-[(2S)-1-methylpyrrolidine-2-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-(1-methyl-3-oxopiperazin-2-yl)-N-[(3,4,5-trimethoxyphenyl)methyl]acetamide
2-[4-(5-propyl-1,2-oxazole-3-carbonyl)piperazin-1-yl]-1-(pyrrolidin-1-yl)ethan-1-one
3-[(5-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-3H,4H-pyrido[2,3-d]pyrimidin-4-one
(2S,4S)-4-[(4,6-dimethylpyrimidin-2-yl)sulfanyl]-1-(9H-fluoren-2-ylmethyl)-N-[2-(3-fluorophenyl)ethyl]pyrrolidine-2-carboxamide
3-[2-(4-benzylpiperidin-1-yl)-2-oxoethyl]-3-(2-chlorophenyl)-1-(2-methoxyethyl)pyrrolidine-2,5-dione
4-[7-(5-ethyl-1,3-oxazole-4-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]morpholine
1-methyl-8-[3-(1-methyl-1H-pyrazol-5-yl)propanoyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-({7-[(3-ethoxy-4-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)pyridine-4-carboxamide
N-[(2S,4R,6S)-2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-6-(2-phenylethyl)oxan-4-yl]acetamide
4-[(2S,6S)-6-(hydroxymethyl)-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-4-yl]-2-methoxypyridine-3-carbonitrile
1-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-3-(2,3-dimethylquinoxalin-6-yl)urea
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(2-propoxyethyl)amine
N-{[5-fluoro-7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(4-fluorophenyl)acetamide
(2-{2-[1-(5-chlorothiophene-2-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
3-(2H-1,3-benzodioxol-5-ylmethyl)-1-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)-3-methylpiperidine
6-[1-(oxan-4-yl)piperidine-3-carbonyl]-5,6,7,8-tetrahydro-1,6-naphthyridine
N-{[5-methyl-7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
1-ethyl-4-{[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl}piperazine-2,3-dione
1-{3-[(1-methylpiperidin-4-yl)methyl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl}-3-(methylsulfanyl)propan-1-ol
N-{[4-(2,3-dihydro-1H-inden-2-yloxy)-3-methoxyphenyl]methyl}-3,4-difluoro-N-(oxolan-2-ylmethyl)benzene-1-sulfonamide
N-[(3R,4S)-4-cyclopropyl-1-(2-methoxyethyl)pyrrolidin-3-yl]-2-(trifluoromethyl)benzamide
N,6-dimethyl-N-{[2-(trifluoromethyl)phenyl]methyl}pyridine-2-carboxamide
N-{5H,6H,7H,8H,9H,10H,11H-cycloocta[b]indol-2-ylmethyl}-1H-pyrazole-3-carboxamide
3-(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)-1-(2-hydroxyethyl)-1-(thiophen-2-ylmethyl)urea
2-(2-ethylpyrimidin-5-yl)-7,8-dimethyl-N-(propan-2-yl)quinoline-4-carboxamide
2-[3-(hydroxymethyl)-3-(2-phenoxyethyl)piperidin-1-yl]pyridine-4-carbonitrile
N-[6-methyl-4-(trifluoromethyl)-1H,6H-[1,2]diazolo[3,4-c]pyrazol-3-yl]-5-(pyrrolidin-1-yl)pyridazin-3-amine