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N-{4-[4-(cyclopentylamino)piperidin-1-yl]phenyl}-2,4-dimethylbenzamide
4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]piperidine
4-[(2-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-yl}-1H-imidazol-1-yl)methyl]pyrimidine
2-{2-[(dimethylamino)methyl]-4-phenylphenoxy}-N-(oxolan-2-ylmethyl)acetamide
[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl](methyl)({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)amine
4-(4-chlorophenyl)-N-methyl-N-(1,2-oxazol-5-ylmethyl)butanamide
1-methyl-N-[3-(2-methyl-1H-imidazol-1-yl)-1-phenylpropyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
4-phenyl-3-(1-{1H-pyrazolo[1,5-a]imidazole-7-carbonyl}piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(2-methoxyphenyl)-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-1H-pyrazole-4-carboxamide
methyl(naphthalen-1-ylmethyl)[(4-{[1-(3,4,5-trimethoxybenzoyl)piperidin-3-yl]methoxy}phenyl)methyl]amine
(2S,4R)-N-ethyl-4-(3-methyloxetane-3-amido)-1-[(3-methylthiophen-2-yl)methyl]pyrrolidine-2-carboxamide
N-{1-[1-(4-aminopyrimidin-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methylbenzamide
N5-(1,4-dioxan-2-ylmethyl)-N5-methyl-N6-(thiophen-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
3-fluoro-N-(3-{2-methoxy-4-[(3-methylpiperidin-1-yl)methyl]phenoxy}propyl)benzamide
N-(4-{[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]carbamoyl}-2-methylphenyl)furan-2-carboxamide
8-fluoro-2-({[3-(methylsulfanyl)propyl]amino}methyl)quinolin-4-ol
1-cyclopentyl-5-[4-(2-hydroxyphenyl)piperazine-1-carbonyl]-N-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
2-(4-fluorophenyl)-1-[4-(2-methoxyphenoxy)piperidin-1-yl]ethan-1-one
6-methyl-N-[1-(thiophen-3-yl)propan-2-yl]imidazo[1,2-a]pyridine-2-carboxamide
1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-3-(pyridin-4-yl)propan-1-one
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carboxamide
2-[1-(2-methoxyphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]pyrazine
N,N-dimethyl-5-{5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-ylmethyl}pyrimidin-2-amine
ethyl 4-{1-[2-(dimethylamino)ethyl]-3-(ethoxycarbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}piperidine-1-carboxylate
1-[2-(dimethylamino)-6-[(1-methyl-1H-imidazol-2-yl)methyl]-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-4-yl]piperidin-4-ol
8-(2-cyclohexylacetyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
1-ethyl-4-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,2-dihydropyridin-2-one
N-(furan-2-ylmethyl)-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-(oxolan-3-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
{[2-(4-cyclohexylpiperazine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}(methyl)(pyridin-3-ylmethyl)amine
6-{[(4-hydroxy-1-methylpiperidin-4-yl)methyl]amino}-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
N-{1-[(2-methylphenyl)methyl]cyclopropyl}-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
N-({2-[2-(2,5-dimethylfuran-3-amido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-5-propyl-1,2-oxazole-3-carboxamide
1-[(2,3-difluorophenyl)methyl]-3-hydroxy-3-{[(2-methylprop-2-en-1-yl)amino]methyl}piperidin-2-one
(3R,5R)-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
3-(2,3-dihydro-1H-inden-2-yl)-5-methyl-5-[1-(2-methylfuran-3-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
4-{3-[(E)-2-phenylethenyl]phenyl}-4H-1,2,4-triazole
{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)(quinolin-4-ylmethyl)amine
7-(2-methylphenyl)-4-[(2R)-oxolane-2-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-(3-hydroxy-3-methylbutyl)-N-[1-(1H-imidazol-2-yl)ethyl]benzamide
3-hydroxy-1-(2-methoxyethyl)-3-{[methyl(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)amino]methyl}piperidin-2-one
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]propan-1-one
N-[(2R,4R,6S)-2-cyclohexyl-6-[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]oxan-4-yl]acetamide
3-(2-methyl-1H-1,3-benzodiazol-1-yl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]propanamide
3-{[1-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)pyrrolidin-3-yl]methyl}benzamide
1-[(2-fluorophenyl)methyl]-4-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}-1,4-diazepane
3-(1H-imidazol-2-yl)-1-[2-(piperidin-1-yl)-1,3-thiazole-4-carbonyl]piperidine
1-ethyl-4-{[3-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl}-1H-indole
1-(3-{2-[1-(piperidin-4-yl)-1H-1,2,3-triazol-4-yl]-1H-imidazol-1-yl}propyl)-2,3-dihydro-1H-indole
2-{[ethyl(2-methylprop-2-en-1-yl)amino]methyl}-4-phenylphenol