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{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)(1,2-oxazol-5-ylmethyl)amine
2-{[(3R,5S)-5-[4-(2-fluorophenyl)piperazine-1-carbonyl]-1-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl]sulfanyl}-4-methylpyrimidine
N-{[7-chloro-2-(4-methoxyphenyl)quinolin-3-yl]methyl}-3-(3-methyl-1H-pyrazol-1-yl)-N-(oxolan-2-ylmethyl)propanamide
7-[2-hydroxy-5-(1H-pyrrol-1-yl)benzoyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
3-{[(5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}furan-2-yl)methyl]sulfanyl}-4H-1,2,4-triazole
2-(2,5-dioxoimidazolidin-1-yl)-N-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]acetamide
N-(2H-1,3-benzodioxol-5-yl)-1-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-amine
3-(2-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl}phenyl)-1H-1,2,4-triazole
N-[(3-chlorophenyl)methyl]-N-[(4-methyl-1H-imidazol-5-yl)methyl]cyclopropanamine
1-methyl-5-[methyl(1,2-oxazol-3-ylmethyl)amino]-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(3S,5R)-N3-butyl-N5-(4-fluorophenyl)-1-(naphthalen-2-ylmethyl)piperidine-3,5-dicarboxamide
N-(1-{7-[(3,4-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)methanesulfonamide
(3S,4R)-4-(3-methylthiophen-2-yl)-1-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-3-ol
5-[(4-fluorophenyl)methyl]-3-(2-methoxyethyl)-5-[1-(4-methylpentanoyl)piperidin-4-yl]imidazolidine-2,4-dione
2-methoxy-N-({8-[(2E)-2-methylbut-2-en-1-yl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)acetamide
N-[(4-methoxyphenyl)methyl]-3-(piperidine-1-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-(2,5-difluorophenyl)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
4-(2H-1,3-benzodioxol-5-yl)-3-(1H-pyrazol-1-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-4-(pyridin-2-ylmethyl)-1,4-diazepane
N-(3-hydroxy-2,2-dimethylpropyl)-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carboxamide
2-({[2-(3,4-dimethoxyphenyl)ethyl]amino}methyl)-4-(6-methoxypyridin-2-yl)phenol
N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-1-{2-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-amine
(2S)-2-acetamido-3-(1H-imidazol-4-yl)-N-(2-methylpropyl)-N-[(2E)-3-phenylprop-2-en-1-yl]propanamide
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-2,3-dimethyl-5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
6-fluoro-N-methyl-2-oxo-N-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-1,2,3,4-tetrahydroquinoline-4-carboxamide
(1R,5S)-6-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-6-azabicyclo[3.2.1]octane
N-{[1-(methoxymethyl)cyclopropyl]methyl}-6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-[3-(2-methyl-1H-imidazol-1-yl)-1-phenylpropyl]-N'-(4-methylphenyl)propanediamide
2-{1-cyclopropyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}-N-methyl-N-(pyridin-2-ylmethyl)acetamide
2-{9-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
3-{[1-(azepane-1-sulfonyl)pyrrolidin-3-yl]methyl}benzoic acid
6-(2,5-dimethylphenyl)-N-[1-(pyridin-3-yl)propan-2-yl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
5-[1-(isoquinolin-5-ylmethyl)pyrrolidin-2-yl]-N-(2-methoxyethyl)thiophene-2-carboxamide
4-methyl-N-[(1S,2R)-2-[(oxan-4-yl)amino]cyclobutyl]-3,4-dihydro-2H-1,4-benzoxazine-7-carboxamide
2-[1-(3-methylbutyl)-4-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-2-yl]ethan-1-ol
1'-(6-methyl-2-propylpyrimidin-4-yl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-[(4-fluorophenyl)methyl]piperazine
3-{1-[(1-butyl-2-cyclobutylmethanesulfonyl-1H-imidazol-5-yl)methyl]pyrrolidin-2-yl}-4-methyl-1,2,5-oxadiazole
1-[(4-methoxyphenyl)methyl]-4-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]acetyl}-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-3-(piperidin-3-yl)benzamide
2-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane-4-carbonyl]pyridin-3-ol
(4aS,8aR)-1-(3-aminopropyl)-6-[3-(pyridin-3-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
1-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
5-benzyl-5-{1-[(3,4-dimethylphenyl)methyl]piperidin-4-yl}-3-[2-(pyridin-2-yl)ethyl]imidazolidine-2,4-dione
(3S,4S)-1-{2-amino-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4-propylpyrrolidine-3-carboxylic acid
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
1-[(3aS,6aS)-1-(pyridin-3-ylmethyl)-octahydropyrrolo[2,3-c]pyrrol-5-yl]-3-(1H-1,3-benzodiazol-1-yl)propan-1-one
4-[(6-methylpyridin-3-yl)oxy]-1-(1H-pyrrole-2-carbonyl)piperidine-4-carboxylic acid
3-(1-{[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-1-ol
methyl 2-{4-[2-(cyclopropylcarbamoyl)ethyl]piperidine-1-carbonyl}benzoate