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N-{1-oxaspiro[4.4]nonan-3-yl}-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-3-(4,5-dimethyl-1H-pyrazol-3-yl)propan-1-one
(2S,4R)-4-amino-N-ethyl-1-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)pyrrolidine-2-carboxamide
2-(3-hydroxypropyl)-9-(2-phenylbutanoyl)-2,9-diazaspiro[5.5]undecan-3-one
3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methylpropanamide
5-[1-(2,1,3-benzothiadiazol-5-ylmethyl)-4-hydroxypiperidin-4-yl]-N-(2-methylpropyl)-1-benzofuran-2-carboxamide
(3S,5R)-N3-(2H-1,3-benzodioxol-5-ylmethyl)-N5-(2,3-dihydro-1H-inden-5-yl)-1-[(4-hydroxyphenyl)methyl]piperidine-3,5-dicarboxamide
1-[(3R,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-2-(methylsulfanyl)ethan-1-one
3-(5-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)phenol
2-(3-fluorophenyl)-N-({7-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)acetamide
(2S,4R)-4-amino-N-methyl-1-(2-methyl-4-phenylpyridine-3-carbonyl)pyrrolidine-2-carboxamide
1-(2-phenylethyl)-N-[3-(pyridin-3-yloxy)propyl]-1H-1,2,3-triazole-4-carboxamide
4-[(2-methylpyridin-3-yl)oxy]-1-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]piperidine-4-carboxylic acid
5-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-(pyrazin-2-ylmethyl)pyridin-2-amine
2-(2-methyl-3-{[({2-[(2-oxopyrrolidin-1-yl)methyl]phenyl}methyl)amino]methyl}-1H-indol-1-yl)acetamide
N-[2-(methylsulfanyl)ethyl]-3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N,N-dimethyl-3-({3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}sulfonyl)benzamide
(2R,6R)-4-{[2-(propylamino)pyrimidin-5-yl]methyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-4-methyl-2-oxopentanamide
2-(ethylamino)-4-methyl-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-1,3-thiazole-5-carboxamide
N-(2-methoxyethyl)-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}-N-(propan-2-yl)benzamide
[(1R)-1-(4-methoxyphenyl)ethyl]({[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]pyridine-2-carboxamide
N-cyclobutyl-2-(phenoxymethyl)-1,3-oxazole-4-carboxamide
2-({4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)benzonitrile
1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-4-(pyridin-3-ylmethyl)piperazine
N-[(3S,4R)-1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
2-(3-methyl-4-{2-[(2-methylprop-2-en-1-yl)oxy]benzoyl}-2-oxopiperazin-1-yl)acetic acid
2-(2,2-dimethylpropanamido)-5-methyl-N-[2-(2-oxoimidazolidin-1-yl)ethyl]thiophene-3-carboxamide
ethyl 2-[1-(3-{2-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-2-yl}propanoyl)piperidin-2-yl]acetate
methyl (2S,4R)-4-(5-chloro-3-phenyl-1H-indole-2-amido)-1-[(3-ethoxy-4-hydroxyphenyl)methyl]pyrrolidine-2-carboxylate
N-[2-(4-fluorophenyl)ethyl]-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
2-methoxy-4-{1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-3-carbonitrile
2-(azetidine-3-carbonyl)-8-methyl-2,8-diazaspiro[4.5]decane
3-({1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl}oxy)pyridine
4-[1-(2-chlorophenyl)-1H-pyrazol-4-yl]-N-[(2S)-oxolan-2-ylmethyl]pyrimidin-2-amine
3-[4-(2-amino-5-ethyl-6-methylpyrimidin-4-yl)piperazin-1-yl]propan-1-ol
N-(1-{1-[(5-cyclohexylthiophen-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)oxolane-3-carboxamide
3,5-dimethoxy-N-({1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-3-yl}methyl)benzamide
N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-1,7-dimethyl-1H-indole-2-carboxamide
2-methyl-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)propanamide
N-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-{[1-(pyridine-3-carbonyl)piperidin-4-yl]oxy}benzamide
1-(2-methanesulfonylethyl)-4-(4-methyl-3-phenyl-1H-pyrazole-5-carbonyl)piperazine
N-[2-(cyclohex-1-en-1-yl)ethyl]-2-(3-methyl-1H-pyrazol-1-yl)-N-{[6-(morpholin-4-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}acetamide
methyl[1-(pyrimidin-4-yl)ethyl]{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
(2R)-2-{[3-(1H-pyrazol-1-ylmethyl)phenyl]formamido}pentanediamide
4-(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)-N-(naphthalen-1-yl)piperidine-1-carboxamide
(1R,7S)-3-(2-ethylbutyl)-6-(3-oxopiperazine-1-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
2-(4-fluorophenyl)-N-{[4-methoxy-3-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)acetamide
3-(3,4-difluorophenyl)-5-(2,2-dimethyloxane-4-carbonyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine