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(1-{[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)methanol
8-[(1,5-dimethyl-1H-indol-2-yl)methyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
3-methyl-1-propyl-N-{[5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H-pyrazole-4-carboxamide
2-{4-cyclobutyl-1-[(4-methoxy-3-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
4-(piperidin-3-yl)-N-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]benzamide
5-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-3-(thiophen-3-ylmethyl)-1,2,4-oxadiazole
2-[4-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazin-1-yl]acetamide
2-[(4aR,7aS)-6,6-dioxo-4-[3-(pyridin-3-yl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
N-[(4-fluorophenyl)methyl]-N-methyl-4-oxo-3,4-dihydroquinazoline-2-carboxamide
2-amino-4-(isoquinolin-5-yl)-6-(trimethyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)piperidine-1-carboxamide
1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}-N-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-2-carboxamide
1-[4-(4-methoxyphenoxy)piperidin-1-yl]-3-[methyl(1-methylpyrrolidin-3-yl)amino]propan-1-one
1-[(3R,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-2-(1-methyl-1H-indol-3-yl)ethan-1-one
6-chloro-N-[(3R,4S)-4-cyclopropyl-1-propanoylpyrrolidin-3-yl]-2H-chromene-3-carboxamide
1-(azocan-1-yl)-3-(2-hydroxyphenyl)-3-(3-hydroxyphenyl)propan-1-one
3-ethoxy-1-[3-(3-phenylpropanoyl)piperidin-1-yl]propan-1-one
2-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyrimidin-4-yl]pyridine-4-carboxylic acid
1-(2-ethoxyethyl)-4-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}piperazine
4-{[4-(3-methoxyphenyl)-3-oxopiperazin-1-yl]methyl}benzoic acid
ethyl 4-benzyl-1-[(3-hydroxy-4-methoxyphenyl)methyl]piperidine-4-carboxylate
2-[1-cyclopropyl-2,5-dioxo-3-(4-phenylphenyl)pyrrolidin-3-yl]-N-methyl-N-(propan-2-yl)acetamide
N-[(2-chlorophenyl)methyl]-5-(morpholin-4-ylmethyl)furan-3-carboxamide
N-{1-[1-(oxolan-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2H-1,3-benzodioxole-5-carboxamide
1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
N-(1-{7-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)methanesulfonamide
3-(2-chlorophenyl)-1-(2-methoxyethyl)-3-(2-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}-2-oxoethyl)pyrrolidine-2,5-dione
1-(2-methylpropyl)-5-oxo-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}pyrrolidine-3-carboxamide
N-({1-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]piperidin-3-yl}methyl)furan-2-carboxamide
4-(3-amino-1H-1,2,4-triazole-5-carbonyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-(oxolan-3-yl)-5-(1-phenylcyclohexyl)-1,2,4-oxadiazole
3-[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]-1-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}urea
3-(1-{[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-2-yl)pyridine
7-(5-ethoxyfuran-2-carbonyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
1-methyl-3-(2-methylpropyl)-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1H-pyrazole-5-carboxamide
ethyl 4-(4-cyclohexyl-3-oxopiperazin-1-yl)piperidine-1-carboxylate
N-[2-hydroxy-3-(pyrrolidin-1-yl)propyl]-3,4,7-trimethyl-1H-indole-2-carboxamide
2-(2,3-dihydro-1-benzofuran-5-yl)-4-[1-(1,2,3-thiadiazole-4-carbonyl)pyrrolidin-3-yl]pyridine
N-[2-(3,4-dimethoxyphenyl)ethyl]-1-(1,4-dithiepan-6-yl)-N-methylpiperidin-3-amine
2-[3-(3-methoxyphenoxymethyl)-5-[(1R,2R)-2-phenylcyclopropyl]-1H-1,2,4-triazol-1-yl]ethan-1-ol
N-{[7-chloro-5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(thiophen-3-yl)acetamide
2-(2,3-dihydro-1H-inden-1-yl)-N-[1-(morpholin-4-ylmethyl)cyclopentyl]acetamide
1-methyl-8-[(3-methylthiophen-2-yl)methyl]-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[3-(2-methoxyphenyl)-1-(3-methoxypropyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-(thiophen-3-ylmethyl)acetamide
5-chloro-2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-[(4-methyl-1,3-thiazol-2-yl)methyl]benzamide
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-hydroxyacetamide
3-ethyl-1-methyl-N-({3-methyl-7-[2-(3-methylphenyl)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-1H-pyrazole-5-carboxamide
2-(4-chlorophenyl)-5-{1-[(2S)-oxolan-2-ylmethyl]-1H-imidazol-2-yl}pyrimidine
1-cyclopentyl-4-[5-(3-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]piperazin-2-one
3-(2-chlorophenyl)-1-cyclopentyl-3-{2-[4-(furan-2-carbonyl)piperazin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione