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3-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-[2-(1H-pyrazol-4-yl)ethyl]benzamide
N-benzyl-N-butyl-1-[(2-chloro-4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
{2-[(4aS,7aR)-4-[(5-methylfuran-2-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-2-oxoethyl}urea
(2S,4S)-4-(benzylamino)-N-ethyl-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
2-[2-(3-phenyl-1H-pyrazol-1-yl)phenyl]acetic acid
1-(3-phenylpropyl)-N-[(1r,4r)-4-hydroxycyclohexyl]-1H-1,2,3-triazole-4-carboxamide
2-[4-(1,3-benzoxazol-2-yl)piperazine-1-carbonyl]-6-methyl-4H-pyran-4-one
2-(4-{3-[(2-methoxyethyl)carbamoyl]piperidin-1-yl}piperidin-1-yl)pyridine-3-carboxylic acid
butyl({[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl})methylamine
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}pyridine-4-carboxamide
1-[4-(2H-1,3-benzodioxol-5-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]-2-phenylethan-1-ol
3-methoxy-1-[2-oxo-2-(3-propoxypiperidin-1-yl)ethyl]-1,2-dihydropyridin-2-one
ethyl 1-[(2,3-dimethylphenyl)carbamoyl]-4-(3-phenylpropyl)piperidine-4-carboxylate
N-(1,3-benzothiazol-2-ylmethyl)-N-methyl-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-(oxolan-3-yl)propanamide
N-[3-(4-methoxyphenyl)propyl]-6-(pyrimidin-5-yl)pyridine-3-carboxamide
6-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-2,5-dimethyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
2-methoxy-N-[(7-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]benzamide
N-[4-(azepan-1-yl)butyl]-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide
4-[4-(2-chlorophenyl)piperidin-4-yl]-2-(2-methoxyethyl)pyrimidine
3-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-1-[3-(2-methylpyrimidin-4-yl)phenyl]urea
methyl 9-(cyclopentyloxy)-3-[(5-ethylfuran-2-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
ethyl 2-(4-{3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanoyl}morpholin-3-yl)acetate
[(2S,4R)-1-methyl-4-({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)pyrrolidin-2-yl]methanol
methyl (2S,4R)-1-(naphthalen-2-ylmethyl)-4-[2-(trifluoromethyl)benzamido]pyrrolidine-2-carboxylate
methyl[(3-methyl-1,2-oxazol-5-yl)methyl]({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)amine
1-benzyl-3-methyl-8-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-{4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]piperidin-1-yl}-N-(1,3-thiazol-2-yl)propanamide
N-[3-(morpholin-4-yl)propyl]-2-(2-phenylethyl)-1,3-benzoxazole-5-carboxamide
1-[(3-hydroxypiperidin-3-yl)methyl]-3-(2-{[(4-methylphenyl)methyl]sulfanyl}phenyl)urea
2-[4-(dimethylamino)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]benzonitrile
3-{1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)propanamide
N-{1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2,5-dimethylfuran-3-carboxamide
(1-{[1-(2-ethyl-1,2,3,4-tetrahydroisoquinoline-3-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methanamine
2-(5-acetylthiophen-3-yl)-1-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
6-methoxy-4-[4-(pyridin-4-yl)piperidine-1-carbonyl]-1,2,3,4-tetrahydroquinolin-2-one
N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}pyrazolo[1,5-a]pyridine-7-carboxamide
N-cyclopropyl-N-[(4-ethoxyphenyl)methyl]-2-(pyridin-2-yl)pyrimidine-5-carboxamide
1-(4-methyl-1,3-thiazole-5-carbonyl)-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine
4-(2,1,3-benzothiadiazol-4-yl)-N-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxamide
N-[3-ethyl-4-(4-fluorophenyl)-1-methyl-1H-pyrazol-5-yl]-3-methoxypiperidine-1-carboxamide
1-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]-4-hydroxypiperidine-4-carboxylic acid
(propan-2-yl)({[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl})[(trimethyl-1H-pyrazol-4-yl)methyl]amine
4-[(4-methoxy-3-methylphenyl)methyl]-3-{2-oxo-2-[4-(propan-2-yl)piperazin-1-yl]ethyl}piperazin-2-one
8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(2-methoxyethyl)-3-(naphthalen-1-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[4-(azepan-1-yl)-4-oxobutanamido]-2-(3,5-dimethyl-1H-pyrazol-4-yl)acetic acid
2-cyclopropyl-8-[2-(propan-2-ylsulfanyl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
N-[1-(3-phenylpropyl)piperidin-3-yl]-3-(thiophen-3-yl)propanamide
2-cyclopropyl-4-hydroxy-N-{2-[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]ethyl}pyrimidine-5-carboxamide
3-[({[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)amino)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one