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N-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-2,7,8-trimethylquinoline-4-carboxamide
3-{1-[(3-hydroxy-4-methoxyphenyl)methyl]piperidin-3-yl}-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
1-[(2,6-difluoro-3-methoxyphenyl)methyl]-4-(1H-pyrrole-2-carbonyl)piperazine
(1-{3-[(cycloheptylamino)methyl]-7-fluoroquinolin-2-yl}piperidin-3-yl)methanol
5-(2-phenylethyl)-5-[1-(3-phenylpropyl)piperidin-4-yl]imidazolidine-2,4-dione
6-(2-methoxyphenyl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
1-[4-({4-[3-(furan-2-yl)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperazin-1-yl]ethan-1-one
N-[(4-fluorophenyl)methyl]-N-methyl-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
2-ethyl-N-[(2-fluorophenyl)methyl]-N-(2-methoxyethyl)pyrimidine-5-carboxamide
N-cyclopropyl-3-phenyl-N-(1,3-thiazol-2-ylmethyl)-1H-pyrazole-4-carboxamide
3-(dimethylamino)-N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
1-[(1-methyl-1H-imidazol-2-yl)methyl]-3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
9-(2,6-dimethylpyrimidine-4-carbonyl)-3-methyl-3,9-diazaspiro[5.6]dodecane
(3S,4R)-1-{[4-(4-chlorophenoxy)phenyl]methyl}-4-(hydroxymethyl)piperidin-3-ol
1-(2-fluoro-4-methylbenzoyl)-2-(4-fluorophenyl)piperidine
2-(pyridin-3-yl)-N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}acetamide
3-(2-methyl-6-propylpyrimidin-4-yl)-3,9-diazaspiro[5.6]dodecan-10-one
N-methyl-N-[(3-methylthiophen-2-yl)methyl]thiophene-2-carboxamide
{[2-cyclohexylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
6-(2-chlorophenyl)-N-[(5-methylpyrazin-2-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-(4-fluorophenyl)-N-[(1r,4r)-4-hydroxycyclohexyl]imidazo[1,2-a]pyridine-6-carboxamide
N-(4-methylphenyl)-3-{[4-(4H-1,2,4-triazol-4-yl)phenyl]formamido}propanamide
5-methoxy-2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenol
1-(2-{1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]piperidin-2-yl}ethyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
2-methyl-5-phenyl-N-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
6-[2-(trifluoromethoxy)phenyl]pyridine-2-carboxamide
2-(3-methoxypropyl)-1-[(1-propyl-1H-imidazol-2-yl)methyl]piperidine
1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine
2-cyclopropyl-N-[(3R,4R)-4-(morpholin-4-yl)oxolan-3-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-(4-methoxyphenyl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]cyclopentane-1-carboxamide
2-[(2-chlorophenyl)methyl]-4-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
1-cyclobutanecarbonyl-N-(3-hydroxypropyl)-N-(pyridin-4-ylmethyl)piperidine-4-carboxamide
2-{[2-({[1-(phenoxymethyl)cyclopropyl]methyl}carbamoyl)phenyl]amino}acetic acid
(3-{[1-(2,3-dimethyl-1H-indole-5-carbonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
2-(4-oxo-3,4-dihydrophthalazin-1-yl)-N-[3-(1H-1,2,3-triazol-1-yl)propyl]propanamide
8-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-{1-benzyl-4-[(1-ethyl-1H-indol-3-yl)methyl]piperazin-2-yl}ethan-1-ol
8-[4-(2,3-dihydro-1H-isoindol-2-yl)butanoyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-{[(4aS,8aS)-4a-hydroxy-decahydroisoquinolin-2-yl]methyl}-2-methoxybenzoic acid
N-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-2-(6-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-4-yl)acetamide
(1R,5R)-N,N-dimethyl-6-(2-methyl-1,3-benzothiazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
3-(azetidine-1-carbonyl)-N-[(1R,2R)-2-hydroxycyclohexyl]-N-propylbenzene-1-sulfonamide
1-{3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-4-[(4-methoxyphenyl)methyl]-1,4-diazepan-5-one
2,3,6-trimethyl-4-[2-(5-methyl-1,2-oxazol-3-yl)piperidine-1-carbonyl]quinoline
N,N,4-trimethyl-3-{[(1H-1,2,4-triazol-3-ylmethyl)carbamoyl]methyl}-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
{3-[(3-chlorophenyl)methyl]-1-(2,3-dimethyl-1H-indole-7-carbonyl)piperidin-3-yl}methanol
2,8-dimethyl-N-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethyl)quinoline-4-carboxamide
1-{7-[(2,6-dimethylphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-methylpropan-1-one
1-{2-phenyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidine-4-carboxamide
1-methyl-3-(2-methylpropyl)-N-[1-(6-methylpyridin-2-yl)propyl]-1H-pyrazole-5-carboxamide