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3-{[(4aS,7aR)-4-(carboxymethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]methyl}benzoic acid
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(piperidin-1-yl)butanamide
methyl 2-[2,4-dioxo-1-(2-phenylethyl)-8-(thiophen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
1-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-(phenylsulfanyl)ethan-1-one
(2S)-N-[(3-chloro-2-methylphenyl)methyl]-1-(piperidin-4-yl)pyrrolidine-2-carboxamide
1-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2,2-dimethylpropan-1-one
N-[1-(4-methanesulfonylphenyl)propyl]-5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[1-methyl-5-({2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}methyl)-1H-pyrrol-3-yl]ethan-1-one
1-[3-(pyridin-3-yl)propyl]-3-(2,4,6-trimethylphenyl)urea
2-ethoxy-3-{2-methyl-1H-imidazo[4,5-b]pyridin-6-yl}pyridine
3-{2-[2-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}-3-phenyl-1-(thiophen-2-ylmethyl)pyrrolidine-2,5-dione
2-[(4-methoxypiperidin-1-yl)sulfonyl]-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
3-(4-chloro-1H-pyrazol-1-yl)-1-[3-(pyridin-3-yl)azetidin-1-yl]propan-1-one
5-methanesulfonyl-2-methyl-4-{3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}pyrimidine
2-chloro-5-acetamido-N-{[1-(hydroxymethyl)cyclobutyl]methyl}-N-methylbenzamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}benzamide
5-{1-[2-(3-fluorophenyl)acetyl]piperidin-4-yl}-5-methyl-3-[2-(morpholin-4-yl)ethyl]imidazolidine-2,4-dione
N-[2-(4-amino-6-hydroxypyrimidin-2-yl)ethyl]-2-(2,5-dimethylphenoxy)propanamide
N-{[7-(6-methoxypyridazin-3-yl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-methyl-3-phenyl-1,2-oxazole-4-carboxamide
(1R,5R)-6-[(5-methoxy-4-oxo-4H-pyran-2-yl)methyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-(2-hydroxyethyl)-N-methyl-1-{1-[(3-phenoxyphenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
N-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]-3-(2-oxoazepan-1-yl)propanamide
N-(1-hydroxy-2-methylpropan-2-yl)-1-(4-methylquinazolin-2-yl)pyrrolidine-2-carboxamide
3-[(4aS,8aR)-4a-(hydroxymethyl)-decahydro-1,6-naphthyridine-6-carbonyl]-6-(trifluoromethyl)pyridin-2-ol
4-[(1-acetylpiperidin-4-yl)oxy]-N-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-3-methoxybenzamide
3-[2-(ethylsulfanyl)-1,3-benzoxazol-6-yl]-1-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}urea
5-[4-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-3-chloro-1,2-dihydropyridin-2-one
1-[2-(1H-imidazol-1-yl)ethyl]-4-(2,3,5,6-tetramethylbenzoyl)piperazine
({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)[2-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)propyl]amine
N-{2-[4-(4-fluorophenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]ethyl}-2-(pyridin-2-ylsulfanyl)acetamide
6-[3-oxo-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-9-yl]pyridine-3-carboxylic acid
N-methyl-N-(1,2-oxazol-3-ylmethyl)-1-propyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-[(2-fluorophenyl)methyl]-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
1-[1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-1H,2H,3H,4H,6H,10bH-pyrimido[2,1-a]isoindol-6-one
N-[2-(2,4-difluorophenyl)-1-{1-[2-(phenylsulfanyl)acetyl]piperidin-4-yl}ethyl]-N-methylpropanamide
1-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
1-[5,6,7-trimethoxy-3-({[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)quinolin-2-yl]piperidin-3-ol
3-{[3-(pyrimidin-4-yl)piperidin-1-yl]methyl}phenol
6-[(diethylamino)methyl]-N-(3-hydroxyphenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
3-[cycloheptyl(pyridin-3-ylmethyl)amino]propane-1,2-diol
N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
5-methyl-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]-1H-pyrazole-3-carboxamide
ethyl 3-(2-phenylethyl)-1-(pyridin-2-ylmethyl)piperidine-3-carboxylate
N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
1-[2-methoxy-4-({[2-(propan-2-yloxy)ethyl]amino}methyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
N2,N2,N4,5,6-pentamethyl-N4-[2-(pyridin-4-yl)ethyl]pyrimidine-2,4-diamine
N-benzyl[(5-methyl-2,1,3-benzothiadiazol-4-yl)amino]sulfonamide
2-[3-(2-fluorophenyl)-1-(2-methoxyethyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}acetamide