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N-[2-(adamantan-1-yl)propan-2-yl]-1-cyclopentyl-6-oxopiperidine-3-carboxamide
2-[3-oxo-9-(3-phenylbutyl)-2,9-diazaspiro[5.5]undecan-2-yl]acetic acid
2-(3-fluorophenyl)-N-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]-1,3-benzoxazole-5-carboxamide
3-(2,3-dihydro-1H-inden-2-yl)-5-methyl-5-[1-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
3-[4-phenyl-5-(2-phenylethyl)-1H-imidazol-1-yl]propan-1-ol
(3S)-3-({5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)azepan-2-one
1-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]-4-(thiophen-2-yl)butan-1-one
N-[2-(1H-imidazol-4-yl)ethyl]-1-{2-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-amine
4-(3-{[4-(aminomethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-1H-pyrazolo[3,4-d]pyrimidin-6-amine
N-[3-(2-methoxy-2-phenylacetamido)phenyl]-3-methylbenzamide
2-[(4-chlorophenyl)methyl]-N-[2-(methylsulfamoyl)ethyl]benzamide
3-(1,2-oxazinan-2-yl)-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}propanamide
5-methyl-N-{[4-(3-methylpiperidin-1-yl)phenyl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-methyl-5-({4-phenyl-5-[5-(1H-pyrazol-5-yl)furan-2-yl]-1H-imidazol-1-yl}methyl)-1,3,4-oxadiazole
methyl 5-{[(3,4-dimethoxyphenyl)methyl]amino}-3-acetamido-1-(3-methylbutyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-{5-[2-(3-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-[2-(methylsulfanyl)ethyl]propanamide
N-{1-[({1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}(methyl)carbamoyl)methyl]-1H-pyrazol-4-yl}-3-phenoxypropanamide
N-(1H-imidazol-2-ylmethyl)-N-methyl-3-{4-[2-(3-methylphenyl)acetamido]-1H-pyrazol-1-yl}benzamide
(3S,9aR)-3-benzyl-8-{[1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-(2-chlorophenyl)-3-[1-(1,2,3,4-tetrahydronaphthalen-2-yl)piperidin-4-yl]propanamide
3-methyl-8-(3-methylbut-2-en-1-yl)-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(2H-1,3-benzodioxol-5-yl)-1-{[1-(3-methylphenyl)-1H-imidazol-2-yl]methyl}piperidin-3-amine
1-(1-benzylpiperidin-4-yl)-3-(dimethyl-1H-1,2,4-triazol-3-yl)urea
N-[(2S)-1-hydroxy-4-(methylsulfanyl)butan-2-yl]-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
N-{[4-(aminomethyl)phenyl]methyl}-3-(4-methyl-4H-1,2,4-triazol-3-yl)propanamide
2-ethyl-4-(2-fluoro-6-methoxybenzoyl)-1-(propan-2-yl)piperazine
N-{2-[2-(4-methoxynaphthalen-1-yl)-1H-imidazol-1-yl]ethyl}-N-methylmethanesulfonamide
3-fluoro-2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-5-methylimidazo[1,2-a]pyridine
N-[2-(1H-imidazol-4-yl)ethyl]-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
3-(3-hydroxy-3-methylbutyl)-N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}benzamide
7-[(3-hydroxypiperidin-3-yl)methyl]-N,N,2-trimethyl-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
methyl[2-(4-methylphenoxy)ethyl]{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}amine
3-{[4-(dimethylamino)phenyl]methyl}-9-methoxy-N-[(4-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
6-[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]pyrimidin-4-amine
2-{1-[(4-ethoxyphenyl)methyl]-4-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperazin-2-yl}ethan-1-ol
1-{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}-2-(1,3-thiazol-2-yl)piperidine
N-[(5-fluoro-1H-indol-2-yl)methyl]-3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
3-[1-(1,4-dioxan-2-ylmethyl)-1H-imidazol-2-yl]-2-methoxyquinoline
2-[7-(1-benzothiophen-3-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetic acid
4-[3-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-2-(4H-1,2,4-triazol-4-yl)pyridine
N-{1-[2-(3-benzoylpiperidin-1-yl)-2-oxoethyl]-1H-pyrazol-4-yl}-3-phenoxypropanamide
1-{3-[3-(hydroxymethyl)-3-propylpiperidin-1-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(2-fluorophenyl)-4-(5-propyl-1,3,4-oxadiazol-2-yl)piperazine
3,4,5-trimethoxy-N-[1-(pyrimidin-2-yl)piperidin-3-yl]benzamide
1-[3-(2-methylpyrimidin-4-yl)phenyl]-N-(thiophen-2-ylmethyl)piperidin-4-amine
5-(2-fluoro-5-methoxyphenyl)pyrimidin-2-amine
8-[2-(dimethylamino)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]-2-methyl-1,3,8-triazaspiro[4.5]dec-1-en-4-one
1-{2-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-2-oxoethyl}-1,2-dihydropyrimidin-2-one
2-(3-methoxypropanoyl)-N-(1-phenylethyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
1-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-8-(4,4,4-trifluorobutan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione