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(3aS,6aR)-5-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-[2-(6-methoxynaphthalen-2-yl)ethyl]-1H-imidazole
[(2-ethylpyrimidin-4-yl)methyl](methyl)[1-(pyrimidin-4-yl)ethyl]amine
1-{[3-(methylsulfanyl)phenyl]methyl}-N-phenylpiperidin-3-amine
2-methyl-3-[2-methyl-4-(2-methylphenyl)piperazine-1-carbonyl]-4,5,6,7-tetrahydro-1H-indol-4-one
1-methanesulfonyl-N-[(4-methoxyphenyl)(pyridin-4-yl)methyl]piperidin-4-amine
7-(oxan-4-yl)-2-(1H-pyrazole-4-sulfonyl)-2,7-diazaspiro[4.5]decan-6-one
(2S)-2-[(7-chloro-3,5-dimethyl-1-benzofuran-2-yl)formamido]-4-methylpentanamide
methyl 7-oxo-3-[(1-phenyl-1H-pyrazol-4-yl)methyl]-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-(4-chloro-1H-pyrazol-1-yl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]ethan-1-one
7,8-dimethyl-2-(1-methyl-1H-pyrazol-4-yl)-4-(2-methylpiperidine-1-carbonyl)quinoline
2-ethoxy-5-{2-[4-(methylamino)piperidin-1-yl]pyrimidin-4-yl}benzoic acid
N-methyl-N-(1,2-oxazol-3-ylmethyl)-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanamide
5-chloro-2-fluoro-N-[2-(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]benzamide
1-methyl-9-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1,4,9-triazaspiro[5.5]undecan-5-one
N-(1-{1-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2H-1,3-benzodioxole-5-carboxamide
3-methyl-3-[2-(morpholin-4-yl)propyl]-1-{4-[2-(pyridin-2-yl)ethyl]phenyl}urea
[(3R,4R)-4-(morpholin-4-ylmethyl)-1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}pyrrolidin-3-yl]methanol
1-[1-(1-aminocyclopentanecarbonyl)piperidin-4-yl]-N,N-diethyl-1H-1,2,3-triazole-4-carboxamide
4-(2H-1,3-benzodioxol-4-ylmethyl)-1-[(1-methyl-1H-pyrazol-4-yl)methyl]-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
1-{4H,5H,6H,7H,8H-cyclohepta[b]thiophene-2-carbonyl}-3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
1-(1-aminocyclopropanecarbonyl)-4-(2,3-dihydro-1H-inden-5-yloxy)piperidine-4-carboxylic acid
1-(benzenesulfonyl)-4-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperazine
6-[(diethylamino)methyl]-N-[3-(hydroxymethyl)phenyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-{[7-chloro-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(furan-2-ylmethyl)propanamide
2-{5-[4-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)phenyl]-3-methyl-1H-1,2,4-triazol-1-yl}pyridine
1-{2-hydroxy-3-[3-({[3-(1H-pyrazol-1-yl)propyl]amino}methyl)phenoxy]propyl}piperidin-4-ol
4,6-dimethyl-1-(2-{[1-(morpholin-4-yl)propan-2-yl]amino}ethyl)-1,2-dihydropyrimidin-2-one
4-oxo-N-[(1S,2R)-2-[(propan-2-yl)amino]cyclobutyl]-2,3,4,5-tetrahydro-1,5-benzothiazepine-7-sulfonamide
7-(6-methylpyridazin-3-yl)-2,7-diazaspiro[4.4]nonane-1,3-dione
2-{[4-(2-methoxybenzoyl)piperazin-1-yl]methyl}-6-methyl-4-(thiomorpholin-4-yl)quinazoline
1-{1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-phenylpiperidin-4-ol
N-{1-[1-(3-methoxybenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-phenylbutanamide
6-[4-(furan-3-ylmethyl)-3-(2-hydroxyethyl)piperazine-1-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
(1R,3S)-3-methoxy-7-{[3-(trifluoromethoxy)phenyl]methyl}-7-azaspiro[3.5]nonan-1-ol
3-[(4-fluorophenyl)methyl]-5-(pyridin-3-yl)-5-{1-[2-(thiophen-3-yl)acetyl]piperidin-4-yl}imidazolidine-2,4-dione
5-(4-methylphenyl)-4-[1-(2,4,5-trifluorobenzoyl)piperidin-3-yl]pyrimidine
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1,3-oxazole-4-carboxamide
3-{[1-(2-methyl-1,3-benzothiazol-6-yl)-1H-1,2,4-triazol-5-yl]methyl}-1,3-oxazolidin-2-one
N-[1-({[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]carbamoyl}methyl)-1H-pyrazol-4-yl]-2-(phenylsulfanyl)acetamide
(4aS,8aR)-6-(2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetyl)-decahydro-1,6-naphthyridine-4a-carboxylic acid
(3S,4S)-4-(1H-imidazol-2-yl)-1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]pyrrolidine-3-carboxylic acid
1-{[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl}-3-(methoxymethyl)piperidine
ethyl 1-{1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carbonyl}piperidine-4-carboxylate
5-[(3-methoxyphenyl)methyl]-3-methyl-5-[1-(2-phenylpropyl)piperidin-4-yl]imidazolidine-2,4-dione
5-[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-4-yl]-3-(cyclopropylmethyl)-5-[(4-fluorophenyl)methyl]imidazolidine-2,4-dione
6-[2-(3-methoxypropyl)-3-oxo-2,8-diazaspiro[4.5]decan-8-yl]pyridine-3-carboxylic acid
2,3-dimethoxy-N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)benzamide
5-(5-chlorothiophen-2-yl)-1-(propan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazole