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6-({methyl[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]amino}methyl)-2-oxo-N-{[3-(trifluoromethyl)phenyl]methyl}-1,2-dihydropyridine-3-carboxamide
5-fluoro-3-methyl-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-1H-indole-2-carboxamide
1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]cyclopropane-1-carboxamide
4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-7-(2-methylphenyl)-9-(oxolan-3-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(dicyclopropylmethyl)-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidine-4-carboxamide
N-(4-{3-[1-(dimethylamino)ethyl]phenyl}-2-ethylphenyl)acetamide
(1R,5R)-3-cyclobutanecarbonyl-6-[(2-ethylpyrimidin-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
3-{3-[4-(hydroxymethyl)piperidin-1-yl]piperidine-1-carbonyl}-1,4,6-trimethyl-1,2-dihydropyridin-2-one
N-(furan-2-ylmethyl)-N,1-dimethyl-5-{[(3,4,5-trimethoxyphenyl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-cyclopropyl-2-(3-acetamidophenyl)pyridine-3-carboxamide
2-[4-(3-hydroxypropyl)phenyl]-2-[4-(6-methylpyridin-2-yl)piperazin-1-yl]acetic acid
3-{1-[(6-chloroquinolin-2-yl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)propanamide
3-{2-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-1-yl]-2-oxoethyl}-4-[(2-methylphenyl)methyl]piperazin-2-one
3-[4-(3-chlorophenyl)-2-methyl-5-oxopiperazin-1-yl]propanoic acid
1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-3-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine
(2S,4S)-1-(2,2-diphenylethyl)-N-methyl-4-[(naphthalen-2-ylmethyl)amino]pyrrolidine-2-carboxamide
1-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(3-chloro-4-hydroxyphenyl)ethan-1-one
1-{3-[benzyl(methyl)amino]piperidin-1-yl}-2-(pyridin-2-ylsulfanyl)ethan-1-one
8-[(2,4-dimethoxyphenyl)methyl]-1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{4-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperazin-1-yl}-1,3-benzoxazole
5-(4-methanesulfonylphenyl)-2-methylpyridine
methyl 3-benzamido-1-(furan-2-ylmethyl)-5-[(oxan-4-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1,4-dimethyl 2-{[1-(4-benzenesulfonamidophenyl)piperidin-4-yl]amino}butanedioate
1-[(2-chlorophenyl)methyl]-N-methyl-N-(pyrazin-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-1,2,3,4-tetrahydroquinolin-2-one
1-(3-fluoro-4-methoxybenzoyl)-N-[4-(propan-2-yl)phenyl]piperidin-3-amine
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1-methyl-2-oxo-1,2-dihydropyridine-4-carboxamide
3-(1-methylpiperidin-2-yl)-N-{[2-(1H-1,2,4-triazol-1-yl)pyridin-3-yl]methyl}propanamide
1-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-3-[3-(propan-2-yloxy)benzoyl]piperidine
2-{2-[3-(2-methylpropyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]phenyl}-1H-imidazole
3-(azocan-1-yl)-N-[3-(2-oxopyrrolidin-1-yl)propyl]propanamide
N-[3-(2-fluoro-3-methoxyphenyl)phenyl]-2-methoxyacetamide
[(1-cyclopentylpiperidin-4-yl)methyl][(5-methoxy-3-methyl-1H-indol-2-yl)methyl](pyridin-3-ylmethyl)amine
N-[(4-fluorophenyl)(pyridin-4-yl)methyl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
5-(2-{5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-oxoethyl)imidazolidine-2,4-dione
(3S,4S)-4-(morpholin-4-yl)-1-[2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]pyrrolidin-3-ol
1-(4,6-dimethylquinazolin-2-yl)-N-[(4-fluorophenyl)methyl]piperidin-4-amine
5-(2-chloro-4-methoxyphenoxymethyl)-N-(oxan-4-ylmethyl)-1,2-oxazole-3-carboxamide
3-methyl-N-(1-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)butanamide
1-(naphthalen-1-ylmethyl)-N,N-bis(prop-2-en-1-yl)-1H-1,2,3-triazole-4-carboxamide
1-[1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-3-(piperidin-1-ylmethyl)piperidine
1-(4-fluorophenyl)-2-(oxane-4-carbonyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
6-[3-(4-chlorobenzoyl)piperidine-1-carbonyl]-2,3-dimethylquinoxaline
1-{3-[methyl(2-phenylethyl)amino]piperidin-1-yl}-2-(quinazolin-4-yloxy)ethan-1-one
[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]({[4-(1H-pyrazol-1-yl)phenyl]methyl})amine
[(3-ethoxy-4-methoxyphenyl)methyl]({2-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl})amine
2-[(1-{4-[(2-methylprop-2-en-1-yl)oxy]benzoyl}piperidin-4-yl)oxy]pyrimidine
5-{1-[(2,3-difluorophenyl)methyl]piperidin-4-yl}-5-methyl-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
N-[2-(2-fluorophenyl)-1-{1-[(2-hydroxy-5-methoxyphenyl)methyl]piperidin-4-yl}ethyl]-N-methylthiophene-2-carboxamide
5-tert-butyl-4-({[1-(dimethyl-1,3-thiazol-4-yl)ethyl](methyl)amino}methyl)furan-2-carboxamide