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1-[9-methoxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(thiophen-3-yl)ethan-1-one
1-tert-butyl-4-({[4-(4-hydroxypiperidin-1-yl)pyrimidin-2-yl](methyl)amino}methyl)pyrrolidin-2-one
5-[(4-fluorophenyl)methyl]-5-{3-[4-(2-methoxybenzoyl)piperazin-1-yl]-3-oxopropyl}pyrrolidin-2-one
3-(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)-1-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)urea
(2S,4R)-1-[(4-hydroxy-3-methoxyphenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-[2-(2,4-difluorophenyl)-1-[1-(2,6-dimethoxybenzoyl)piperidin-4-yl]ethyl]-N-methylcyclopropanecarboxamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
3-(1-{[(2-chloro-5-ethoxy-4-propoxyphenyl)methyl]amino}ethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(3-methylbutyl)-3-(pyridin-3-ylmethyl)-8-{[3-(trifluoromethyl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{1-[4-(2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)phenyl]-1H-pyrazol-4-yl}oxane-4-carboxamide
2,7,8-trimethyl-4-[3-(pyridin-2-yl)azetidine-1-carbonyl]quinoline
2-[(quinolin-6-yloxy)methyl]-N-[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]-1,3-oxazole-4-carboxamide
2-methoxy-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)pyridine-3-carboxamide
2-[6-(5-fluoroquinolin-8-yl)pyridin-3-yl]acetic acid
N-[(3R,4S)-4-cyclopropyl-1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]pyrrolidin-3-yl]-2-hydroxyacetamide
N-(4-chloro-2-fluorophenyl)-2-{[(1-cyclopentyl-5-oxopyrrolidin-3-yl)methyl](methyl)amino}acetamide
3-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-6-ethyl-3,4-dihydroquinazolin-4-one
1-(4-methoxyphenyl)-4-{1-[(3-methylphenyl)methyl]piperidin-3-yl}piperazine
N-[2-hydroxy-2-(pyridin-3-yl)ethyl]-4-(3-hydroxy-3-methylbutyl)benzamide
2,2-diphenyl-1-[4-(1,3-thiazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]ethan-1-ol
3-(3,4-dimethoxyphenyl)-N-{[5-fluoro-7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
3-(2-fluorophenyl)-1-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]propan-1-one
(2S,4S)-4-amino-1-(2,3-dihydro-1H-indene-5-carbonyl)-N-ethylpyrrolidine-2-carboxamide
2-{1-[(2-chloro-4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(methylsulfanyl)ethyl]acetamide
1-[4-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
4-[5-(4-methoxyphenyl)furan-2-carbonyl]-1λ6-thiomorpholine-1,1-dione
methyl[(4-{[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl][2-(pyridin-2-yl)ethyl]amine
1-{3-[4-(thiophen-2-ylmethyl)-1,4-diazepane-1-carbonyl]phenyl}ethan-1-one
4-[1-(2-hydroxyethyl)-3-[(2-methoxyphenyl)methyl]-1H-1,2,4-triazol-5-yl]-3,5-dimethyl-1H-pyrrole-2-carboxylic acid
9-(oxan-2-ylmethyl)-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[3-(1H-indol-2-yl)phenyl]-1-(3-methoxypropanoyl)piperidine-3-carboxamide
N-(cyclopropylmethyl)-3-{2-[(3,4-dimethoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
3-methyl-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
2-({[(3R,4R)-1-[3-(dimethylamino)benzoyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
ethyl 3-(2-phenylethyl)-1-[3-(1H-1,2,4-triazol-1-yl)propanoyl]piperidine-3-carboxylate
2-(1H-pyrazol-1-yl)-N-{2-[2-(pyridin-4-yl)-1,3-thiazol-4-yl]ethyl}butanamide
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-2-(morpholin-2-yl)acetamide
N-(2-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}-2-oxoethyl)methanesulfonamide
5-methoxy-1-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-5-yl)-1H-indole-2-carboxamide
1-benzyl-5-(cyclopentylamino)-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-cyclohexyl-N-[(4-methanesulfonylmorpholin-2-yl)methyl]-1H-pyrazole-4-carboxamide
N-[2-methyl-1-(piperidin-1-yl)propan-2-yl]-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
3-[3-(4-phenoxybenzoyl)piperidin-1-yl]propanamide
1-(4-butyl-3-oxopiperazine-1-carbonyl)cyclopropane-1-carbonitrile
2-(3-methoxyphenyl)-1-[3-(thiophen-2-yl)-1H-pyrazole-4-carbonyl]piperidine
N-(2,3-dihydro-1H-inden-1-yl)-1-[(4-fluorophenyl)methyl]-5-(2-methoxyacetamido)-1H-1,3-benzodiazole-7-carboxamide
1-({3-[(quinolin-7-yl)carbamoyl]phenyl}methyl)piperidine-4-carboxamide
(3S,4S)-1-[4-(hydroxymethyl)-1,3-thiazol-2-yl]-4-methylpiperidine-3,4-diol
2-[2-(2-cyclohexylpyrimidin-5-yl)-1H-imidazol-1-yl]-1-phenylethan-1-ol
3-(3-fluoro-4-methoxybenzoyl)-1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidine