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ethyl 3-[(3-methoxyphenyl)methyl]-1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidine-3-carboxylate
1-methyl-4-[2-(thiophen-3-yl)acetyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
4-[(2-chloro-4-fluorophenyl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
(3S,4R)-1-[2-(2-hydroxyethoxy)ethyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
5-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}-2-methoxypyrimidine
6-(benzyloxy)-4-(1-ethylpiperidin-4-yl)-1-(2-methylpropyl)-1,4-diazepan-2-one
3-(furan-2-yl)-4-[(4-methoxyphenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
(1S,6R)-N-(4-methoxy-2-methylphenyl)-3,9-diazabicyclo[4.2.1]nonane-9-carboxamide
2-methyl-6-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}-2,3-dihydropyridazin-3-one
N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
2-{2-[4-hydroxy-4-(pyridin-3-yl)piperidin-1-yl]pyrimidin-4-yl}pyridine-4-carboxylic acid
N-ethyl-3,5,7-trimethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-1H-indole-2-carboxamide
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1H-imidazol-4-ylmethyl)piperidine
N-[(5-fluoro-2-methylphenyl)methyl]-1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
(3S,4S)-1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
5-(2,5-dimethylphenoxymethyl)-N-methyl-N-(1-methylpyrrolidin-3-yl)-1,2-oxazole-3-carboxamide
2-[1-(2,2-dimethylpropyl)-4-(quinolin-2-ylmethyl)piperazin-2-yl]ethan-1-ol
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-benzyl-N-[(3-methylpyridin-2-yl)methyl]acetamide
N-methyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}pyrimidin-2-amine
1-methyl-N-(2-phenylethyl)-5-(piperidin-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-methyl-N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(3-methoxyphenoxy)ethan-1-one
1-[(3-methylpyridin-2-yl)methyl]-4-(5-phenyl-1,2,4-oxadiazol-3-yl)piperazine
dimethyl[2-(2-{1-[3-(pyrrolidin-1-yl)pyrazin-2-yl]piperidin-3-yl}-1H-imidazol-1-yl)ethyl]amine
5-[1-(2-chloro-6-fluorobenzoyl)piperidin-4-yl]-3-(furan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
1-ethyl-4-(2-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)piperazine
2-[(4-hydroxyazepan-1-yl)methyl]-6-methylquinolin-4-ol
[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl](methyl){[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}amine
N-(2,2-dimethyloxan-4-yl)-N-ethyl-2-[(2-methylprop-2-en-1-yl)oxy]benzamide
N-[(3,4-difluorophenyl)methyl]-3-(1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidin-3-yl)propanamide
1-(azocan-1-yl)-3-[5-(4-phenylphenyl)-1,3,4-oxadiazol-2-yl]propan-1-one
2-[2,5-dioxo-3-phenyl-1-(thiophen-2-ylmethyl)pyrrolidin-3-yl]-N-(2-methoxyethyl)-N-(propan-2-yl)acetamide
N-{[7-chloro-2-(3-methylphenyl)quinolin-3-yl]methyl}-2-oxo-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
3-[(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)amino]pyrazine-2-carbonitrile
4-[3-(morpholin-4-yl)azetidin-1-yl]-5,6,7,8-tetrahydroquinazolin-2-amine
1-[(3-fluoro-4-methylphenyl)methyl]-5-{2-[(prop-2-en-1-yl)amino]ethyl}pyrrolidin-2-one
8-{[2-methoxy-5-(propan-2-yl)phenyl]methyl}-2,8-diazaspiro[4.5]decan-3-one
1-(azocan-1-yl)-3-[2-methoxy-5-({[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)phenoxy]propan-2-ol
1-[7-(2-cyclohexylethyl)-2,7-diazaspiro[4.5]decan-2-yl]-3-(4-methylpiperazin-1-yl)propan-1-one
2-ethyl-N-[3-(pyridin-2-yl)propyl]pyrimidine-5-carboxamide
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzamide
6-tert-butyl-2-(2-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}phenyl)-3,4-dihydropyrimidin-4-one
methyl 3-[(3S,4R)-1-[(2,6-difluorophenyl)methyl]-4-(dimethylamino)piperidin-3-yl]propanoate
1-{1-[1-(2-methoxy-5-methylbenzoyl)piperidin-4-yl]ethyl}-4-methylpiperazine
(2R,3R,6R)-5-(2-methoxypyridine-4-carbonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
{3-benzyl-1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperidin-3-yl}methanol
5-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]-3-[3-(dimethylamino)propyl]-5-[(4-fluorophenyl)methyl]imidazolidine-2,4-dione
methyl (2S)-1-{3-[2-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-2-yl]propanoyl}pyrrolidine-2-carboxylate
1-(1-{[1-(2-hydroxyethyl)-3-phenyl-1H-1,2,4-triazol-5-yl]methyl}-3,5-dimethyl-1H-pyrazol-4-yl)ethan-1-one