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methyl 4-{6-amino-5-cyano-4-[5-(hydroxymethyl)furan-2-yl]pyridin-2-yl}-5-methylfuran-2-carboxylate
1-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-(pyrrolidine-1-carbonyl)piperidine
6-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)-1H-imidazol-1-yl]-3,4-dihydro-2H-1,4-benzoxazin-3-one
5-(2-{4-[1-(dimethylamino)ethyl]piperidin-1-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-{1-[(4-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-(2-methoxyethyl)-N-methylacetamide
N-[(3,4-dimethoxyphenyl)methyl]-4-(3-fluorophenyl)-N-(pyridin-2-ylmethyl)benzamide
4-(2,1,3-benzothiadiazol-4-yl)-7-hydroxy-6-methyl-1,2,3,4-tetrahydroquinolin-2-one
6,7-dimethoxy-2-{1-[1-(propan-2-yl)piperidin-4-yl]piperidin-3-yl}-1,2,3,4-tetrahydroisoquinoline
N-[2-(2-ethoxyphenoxy)ethyl]-N,4-dimethylpyridine-3-carboxamide
methyl({2-[(4-methylpyridin-2-yl)oxy]hex-5-en-1-yl})(pyridin-3-ylmethyl)amine
N-[1-(4-{[(4-chlorophenyl)(pyridin-4-yl)methyl]carbamoyl}phenyl)-1H-pyrazol-4-yl]furan-3-carboxamide
1-{2-[2-(2-methoxyethyl)piperidin-1-yl]-2-oxoethyl}-5,5-dimethylimidazolidine-2,4-dione
N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)-3-(2-oxopiperidin-1-yl)propanamide
2-(4-{[3-(2-hydroxyethyl)-4-[(4-methylphenyl)methyl]piperazin-1-yl]methyl}phenoxy)ethan-1-ol
N-ethyl-1,5-bis[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
6-{[3-(furan-2-yl)phenyl]methyl}-N-[3-(pyridin-4-yl)propyl]-6-azaspiro[2.5]octane-1-carboxamide
3-chloro-N-[2-(dimethylamino)ethyl]-4-({1-[1-(methylsulfanyl)propan-2-yl]piperidin-4-yl}oxy)benzamide
3-{[(1-{1-[(4-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-4-yl)oxy]methyl}pyridine
1-{2-[(cycloheptylamino)methyl]-4-methoxyphenoxy}-3-(dimethylamino)propan-2-ol
2-{[1-(4-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1,3-thiazole
2-(4-chlorophenoxy)-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]acetamide
(3S,4S)-1-({[(5-carboxyfuran-2-yl)methyl]carbamoyl}methyl)-4-propylpyrrolidine-3-carboxylic acid
N-[2-(4-fluorophenyl)ethyl]-N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}thiophene-2-carboxamide
2-(4-chloro-2-methylphenoxy)-1-[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]ethan-1-one
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-methoxypyridine-4-carboxamide
(3S)-4-[(5-chloro-2,4-dimethoxyphenyl)methyl]-3-ethylmorpholine
5-[1-(2-chlorobenzoyl)piperidin-4-yl]-3-[(2,3-dimethoxyphenyl)methyl]-5-methylimidazolidine-2,4-dione
(3S,4R)-1-(4-carboxybutyl)-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
[(1-ethyl-1H-imidazol-2-yl)methyl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
N-[1-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-amine
6-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carbonyl}-4-methyl-1,3-benzothiazol-2-amine
2-(1-butyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N,N-dimethylacetamide
2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-(2-methylpropyl)-N-[(2E)-3-phenylprop-2-en-1-yl]acetamide
(2H-1,3-benzodioxol-4-ylmethyl)(methyl){[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}amine
1-[(2-hydroxy-5-methoxyphenyl)methyl]-N-[2-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
1-(3,3-dimethyl-4-phenylpyrrolidin-1-yl)-2-(morpholin-4-yl)ethan-1-one
3-(2-carbamoylethyl)-1-[(1-ethylpyrrolidin-2-yl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
N-(2-fluoro-5-methylphenyl)-2-{[1-(4-methylbenzoyl)piperidin-4-yl]amino}acetamide
4-chloro-2-fluoro-N-[1-(2-phenylethyl)piperidin-3-yl]benzamide
methyl[(3-methylpyridin-4-yl)methyl]{[3-(propan-2-yl)-1H-pyrazol-5-yl]methyl}amine
4-(4-{1,2-dihydrospiro[indole-3,4'-piperidine]-1'-ylmethyl}phenyl)-2-methylbutan-2-ol
4-{[5-(1-methyl-1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]methyl}benzoic acid
3-(4-methylphenyl)-3-[4-(quinolin-4-yl)-1H-1,2,3-triazol-1-yl]propan-1-ol
7-methyl-2-(5-phenyl-1H-pyrrole-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-5-oxo-1-phenyl-2,5-dihydro-1H-pyrazole-3-carboxamide
(1R,3S)-N3-ethyl-1,2,2-trimethyl-N1-[2-(piperidin-1-yl)ethyl]cyclopentane-1,3-dicarboxamide
1-[(5-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}-2-methoxyphenyl)methyl]-1H-1,2,4-triazole
N-{[7-(2,4-difluorobenzoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(pyrrolidin-1-yl)acetamide
8-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
1-[(3-methoxyphenyl)methyl]-4-[2-(methylsulfanyl)pyridine-3-carbonyl]piperazin-2-one