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2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}acetamide
1-[2-(dimethylamino)ethyl]-5-[2-({2-methylthieno[3,2-d]pyrimidin-4-yl}amino)ethyl]pyrrolidin-2-one
3-{3-[3-(dimethylamino)pyrrolidin-1-yl]propyl}-8-(pyridine-4-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-cyclopentyl-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-phenylacetamide
1-[3-hydroxy-3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-2-(pyrimidin-2-ylsulfanyl)ethan-1-one
methyl 3-(cyclohex-3-en-1-ylmethyl)-9-[(4-fluorophenyl)methoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(1,3-thiazole-4-carbonyl)piperazin-2-one
2-methyl-4-{3-[2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]phenyl}butan-2-ol
[3-(1H-imidazol-1-yl)propyl][(1-methyl-1H-imidazol-2-yl)methyl](pyridin-4-ylmethyl)amine
ethyl 1-[(3-acetylphenyl)carbamoyl]-4-[(2-chlorophenyl)methyl]piperidine-4-carboxylate
1-(2-methoxyethyl)-N-methyl-N-[2-(oxan-2-yl)ethyl]-7-(pyridine-3-amido)-1H-1,3-benzodiazole-5-carboxamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[3-(1H-pyrazol-1-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
{4-[2-(pyridin-4-yl)pyrimidine-5-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methanol
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(4-methylpent-3-en-1-yl)pyrrolidin-3-yl]-5-methyl-1,2-oxazole-3-carboxamide
1-{7-[(3,4-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3-(pyridin-2-yl)propan-1-one
3-{[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]sulfonyl}-4-methoxybenzoic acid
1-[(6-methylpyridin-2-yl)methyl]-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
(3aR,6aR)-2-[6-(piperidin-1-yl)pyrimidin-4-yl]-5-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{3-[4-(2-chlorophenoxy)piperidin-1-yl]-3-oxopropyl}-1,2-dihydropyridin-2-one
1-[3-(dimethylsulfamoyl)-5-[(furan-3-ylmethyl)amino]benzoyl]piperidine-3-carboxamide
3-[3-(2H-1,3-benzodioxol-5-yl)phenyl]-1-(2-methoxyethyl)-1H-pyrazole
(3S,4R)-4-(2-methoxyphenyl)-1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]pyrrolidine-3-carboxylic acid
N-(2-{7-[(2,4-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)oxolane-2-carboxamide
3-[1-(2-hydroxypyridine-3-carbonyl)piperidin-3-yl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
(3R,5R)-1-[(4-hydroxyphenyl)methyl]-N-(oxolan-2-ylmethyl)-5-(pyrrolidin-1-ylmethyl)piperidine-3-carboxamide
1-[2-(6-methoxypyridin-3-yl)pyrimidin-4-yl]pyrrolidin-3-ol
9-[(4-tert-butylphenyl)methyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
7-[(3-methylphenyl)methyl]-2-(pyridin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
2-(difluoromethoxy)-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]benzamide
N-{7-[4-(2-methoxyethyl)piperazine-1-carbonyl]-1-methyl-2-phenyl-1H-1,3-benzodiazol-5-yl}ethane-1-sulfonamide
methyl 5-[(cyclohexylmethyl)amino]-3-acetamido-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-(4-chloro-2-methoxy-5-methylphenyl)-3-(hydroxymethyl)morpholine-4-carboxamide
1-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
(1S,5R)-3-benzyl-6-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
3-fluoro-N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]benzamide
2-(3,5-dimethylphenyl)-5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]pyridine
ethyl 3-{[1-propyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}propanoate
1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-3-(pyrrolidine-1-carbonyl)piperidine
3-(8-chloroquinoline-2-carbonyl)-3,9-diazaspiro[5.5]undecane
2-cyclopentyl-1-[3-(4-{[methyl(1,3-thiazol-2-ylmethyl)amino]methyl}phenoxymethyl)piperidin-1-yl]ethan-1-one
4-(pyridin-3-yl)-2-[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]pyrimidine
{3-[(4-fluorophenyl)methyl]-1-{[4-(propan-2-yloxy)phenyl]methyl}piperidin-3-yl}methanol
N-(oxan-2-ylmethyl)-3-[(2,2,2-trifluoroethyl)sulfamoyl]benzamide
2,6-dimethyl-3-[3-(4-methylphenoxymethyl)piperidine-1-carbonyl]-1,4-dihydropyridin-4-one
2-({[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)amino)-1-phenylethan-1-ol
2-{[2-amino-6-(5-chloro-2-methoxypyridin-4-yl)pyrimidin-4-yl]amino}ethan-1-ol
N-[2-(1-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)ethyl]acetamide
4-(1-{dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}piperidin-4-yl)thiomorpholine
7-chloro-N-ethyl-N-methyl-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
2-methoxy-N-[1-(3-{4-[3-(trifluoromethyl)phenyl]piperazine-1-carbonyl}phenyl)-1H-pyrazol-4-yl]acetamide