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3-phenyl-1-[3-(1H-pyrazol-1-yl)propyl]piperidine
N-tert-butyl-2-{[6-(3-fluorophenyl)imidazo[2,1-b][1,3]thiazol-3-yl]formamido}acetamide
3-[(3S,4R)-4-(dimethylamino)-1-(2,2-diphenylethyl)piperidin-3-yl]-1-[4-(4-methoxyphenyl)piperazin-1-yl]propan-1-one
3-(2-methoxyphenoxy)-1-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}azetidine
{2-[2-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]phenyl}methanol
5-cyclohexyl-1-propyl-1H,4H-pyrazolo[3,4-d]imidazole
N-{[7-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-phenylacetamide
5-{1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl}-3-(2,3-dihydro-1H-inden-2-yl)-5-methylimidazolidine-2,4-dione
2-amino-6-(1-ethyl-1H-indol-3-yl)-4-(2-methoxypyrimidin-5-yl)pyridine-3-carbonitrile
3-({5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)benzonitrile
N-[(3S,4R)-4-propyl-1-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}pyrrolidin-3-yl]acetamide
5-acetyl-N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-methylthiophene-3-carboxamide
N-(1-phenylbutyl)thiophene-2-carboxamide
2-amino-7-[2-(dimethylamino)-2-(2-fluorophenyl)acetyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-(dimethylamino)-4-methyl-N-{2-[2-(pyridin-4-yl)-1,3-thiazol-4-yl]ethyl}pyrimidine-5-carboxamide
4-(1,2-oxazolidine-2-carbonyl)-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole
N-[3-(4-fluorophenyl)phenyl]-1-(pyridin-2-ylmethyl)pyrrolidine-2-carboxamide
1-ethyl-3-[2-(2-ethyl-3-oxopiperazin-1-yl)-2-oxoethyl]-3-[3-(trifluoromethyl)phenyl]pyrrolidine-2,5-dione
4-hydroxy-N-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-2-methylpyrimidine-5-carboxamide
{1-[(4-{[4-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methyl]piperidin-2-yl}methanol
(2,1,3-benzothiadiazol-5-ylmethyl)({[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl})methylamine
N-{1-benzyl-2-methyl-7-[2-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1H-1,3-benzodiazol-5-yl}-2-methylpropanamide
N-{3-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidine-1-carbonyl]phenyl}acetamide
N-[(3R,4R)-3-hydroxypiperidin-4-yl]-3-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]propanamide
1-[(2-methyl-1,3-oxazol-4-yl)methyl]-3-(2-methylphenyl)piperidine
1-[4-(thiomorpholin-4-yl)piperidin-1-yl]-2-[2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
3-(4-chlorophenyl)-N-[2-(4-hydroxypiperidin-1-yl)ethyl]-3-phenylpropanamide
1-[3-(dimethylamino)pyrazin-2-yl]-3-[(2-fluorophenyl)methyl]piperidine-3-carboxylic acid
(1R,5R)-6-[(2,6-dimethylphenyl)methyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
[(2-butoxy-3-methoxyphenyl)methyl]({5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl})amine
4-ethyl-3-[1-(5-methyl-1,3-benzoxazol-2-yl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
5-benzamido-1-cyclopentyl-N-[1-(1,3-thiazol-2-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
6-({4-[(benzyloxy)methyl]-1H-1,2,3-triazol-1-yl}methyl)pyrimidin-4-ol
[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
9-methoxy-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-3-[(2E)-3-phenylprop-2-en-1-yl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
(3S,9aR)-8-(3,5-dichlorobenzoyl)-2-methyl-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(3S,4S)-4-cyclopropyl-1-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)pyrrolidine-3-carboxylic acid
2-[3-(1-benzyl-3-cyclopentyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]acetamide
N-(2,6-dimethylphenyl)-3-[(3E)-pent-3-enamido]benzamide
N-{4-[4-(4-hydroxybut-1-yn-1-yl)phenyl]-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl}acetamide
2-[2-(2-methylfuran-3-carbonyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl]pyridine
1-(6-chloroquinolin-2-yl)-3-(hydroxymethyl)piperidin-3-ol
2-fluoro-N-(2-methoxyethyl)-5-sulfamoyl-N-(thiophen-3-ylmethyl)benzamide
1-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}-2-propoxypropan-1-one
2-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-7-(3-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-N-(prop-2-en-1-yl)-1,3-oxazole-4-carboxamide
2-(dimethylamino)-2-(4-fluorophenyl)-1-(4-hydroxy-4-phenylpiperidin-1-yl)ethan-1-one
2-(5-chloro-1H-1,3-benzodiazol-2-yl)-N-{1-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}acetamide
N-cyclopentyl-N-(3-phenylprop-2-yn-1-yl)-3-(1H-1,2,4-triazol-1-yl)propanamide
N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-1,9-dioxaspiro[5.5]undecan-4-amine