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3-(1-{[1-(cyclohexylmethyl)-2-cyclopropylmethanesulfonyl-1H-imidazol-5-yl]methyl}piperidin-3-yl)propan-1-ol
2-methoxy-N-{5-[(2-phenylazetidin-1-yl)methyl]-1,3-thiazol-2-yl}pyridin-3-amine
2-cyclopropyl-N-{[7-(5-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}[(2-fluorophenyl)methyl](2-methoxyethyl)amine
dimethyl({4-[1-(thiophene-3-carbonyl)piperidin-2-yl]phenyl}methyl)amine
1-[(3-fluorophenyl)methyl]-4-{[(3-methylphenyl)methyl]amino}pyrrolidin-2-one
1-[3-(5-benzyl-2-methylpyrimidin-4-yl)piperidin-1-yl]-2-(2-chlorophenoxy)ethan-1-one
(1R,2R)-2-{5-[(3-methoxyphenyl)methyl]-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl}cyclohexan-1-ol
2-{1-cyclopropyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}-N-methyl-N-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)acetamide
N-[2-(4-chlorophenyl)ethyl]-1-(2-methylpropyl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[3-(oxolan-3-yl)propyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
4-(2-methoxyethyl)-1-[8-(trifluoromethyl)quinolin-4-yl]piperidine-4-carboxylic acid
1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4-(2-fluorophenoxy)piperidine-4-carboxylic acid
2-cyclopropanecarbonyl-8-[(3-fluoro-4-methylphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-phenoxy-N-{1-[7-(quinolin-8-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}acetamide
N-(4-methoxy-2-methylphenyl)-3-[1-(pyridazine-4-carbonyl)piperidin-3-yl]propanamide
(3aR,5R,6S,7aS)-2-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]-octahydro-1H-isoindole-5,6-diol
3-({4-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}methyl)pyridine
6-[(2-fluorophenyl)methoxy]-1-(2-methylpropyl)-4-{4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carbonyl}-1,4-diazepan-2-one
N-methyl-2-[(propan-2-yl)amino]-N-{[4-(trifluoromethyl)phenyl]methyl}pyrimidine-5-carboxamide
3-[2-(2-fluorophenyl)acetyl]-9-methoxy-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
[(2S,4R)-1-{[5-(2-chlorophenyl)furan-2-yl]methyl}-4-(dimethylamino)pyrrolidin-2-yl]methanol
N-[(2R,3R)-2-ethoxy-1'-{[3-(trifluoromethyl)phenyl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-4-yl)-N-[1-(3-fluoro-4-methoxyphenyl)ethyl]acetamide
7-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}-2-oxa-7-azaspiro[4.5]decane
2-({[1-(2-methoxyphenyl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]methyl}sulfanyl)pyrimidine
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-(pyridin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
6-(morpholin-4-yl)-N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
5-[4-(4-chlorophenoxy)piperidine-1-carbonyl]-1H-1,2,3-benzotriazole
3-[2-(4-ethylpiperazin-1-yl)ethyl]-8-[(2E)-3-phenylprop-2-en-1-yl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(2R,3R,6R)-5-(3,5-dimethylbenzoyl)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(4-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-6-hydroxy-1,4-diazepan-1-yl)ethan-1-one
4-(2-fluoro-5-methylphenoxy)-1-[(5-hydroxy-2-methoxyphenyl)methyl]piperidine-4-carboxylic acid
1-[2-(1-methylpyrrolidin-2-yl)acetyl]-4-phenylpiperidine-4-carbonitrile
N-({7-[(4-methoxynaphthalen-1-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-3-(pyridin-3-yl)propanamide
(2E)-N-[2-(3,4,5-trimethoxyphenyl)phenyl]but-2-enamide
1-[2-(3,5-dimethyl-1H-pyrazol-4-yl)acetyl]-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
2-[(3R,4R)-3-[(4-ethylpiperazin-1-yl)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-N-methylpyridine-3-carboxamide
3-methyl-4-oxo-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)-3,4-dihydroquinazoline-7-carboxamide
[3-(2-phenoxyethyl)-1-(quinolin-5-ylmethyl)piperidin-3-yl]methanol
1-(2,3-dihydro-1H-inden-2-yl)-4-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-1,4-diazepane
2-hydroxy-N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}pyridine-3-carboxamide
3-(2-chlorophenyl)-3-{2-[2-(2-methoxyphenyl)pyrrolidin-1-yl]-2-oxoethyl}-1-methylpyrrolidine-2,5-dione
N-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine-1-carboxamide
2-{1-[(2E)-hex-2-en-1-yl]piperidin-4-yl}-N-methylacetamide
3-[(2,6-dimethylquinolin-3-yl)formamido]-N-(2-methoxyphenyl)propanamide
3-fluoro-5-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidine-1-carbonyl]benzonitrile
4-[5-(pyridin-3-yl)-1H-imidazol-2-yl]-1-(pyridin-3-ylmethyl)pyrrolidin-2-one
2-ethyl-N-[(5-methylpyrazin-2-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
3-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2,4-dichlorophenyl)urea