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3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methyl-1-(4-methyl-1,3-thiazole-5-carbonyl)piperidine
N3-benzyl-N5-cyclooctyl-N3-ethyl-4-oxo-1-(oxolan-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
4-[(2-methoxypyrimidin-5-yl)methyl]-2-(naphthalen-1-ylmethyl)morpholine
2-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]acetamide
2-{5-[5-(1,5-dimethyl-1H-pyrazol-4-yl)-1,2-oxazol-3-yl]-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl}-6-methylpyridine
(2S,4R)-N-{imidazo[1,2-a]pyridin-2-ylmethyl}-4-[(4-methoxyphenyl)sulfanyl]-1-{[4-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxamide
5-(2H-1,3-benzodioxol-4-ylmethyl)-N-(2-hydroxyethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
dimethyl({4-[1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperidin-2-yl]phenyl}methyl)amine
(2S,4S)-4-amino-N,N-diethyl-1-{[1-(propan-2-yl)-1H-1,3-benzodiazol-2-yl]methyl}pyrrolidine-2-carboxamide
2-(dimethylamino)-N-{[1-(methoxymethyl)cyclopentyl]methyl}-2-(4-methylphenyl)acetamide
N-[(4-fluoro-3-methylphenyl)methyl]-2-(pyrrolidin-3-yl)benzamide
4-{4-[({[1-(hydroxymethyl)cyclopropyl]methyl}(methyl)amino)methyl]phenyl}-2-methylbutan-2-ol
N-({3-[(2-chloroprop-2-en-1-yl)oxy]-4-methoxyphenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]-3-(2-oxoimidazolidin-1-yl)benzamide
1-{4-[4-(2-chlorophenyl)piperidin-4-yl]pyrimidin-2-yl}piperidin-3-ol
N-[(3R,4S)-4-cyclopropyl-1-(2,3-dihydro-1H-inden-2-yl)pyrrolidin-3-yl]oxane-4-carboxamide
2-{4-[(4-fluoro-3-methoxyphenyl)methyl]-1-[(2-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-[(2R,3R)-2-ethoxy-1'-[(2E)-3-(thiophen-2-yl)prop-2-enoyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-3-carboxamide
N-[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-8-(1-propylpiperidin-4-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl (2S,4R)-4-hydroxy-1-[3-(1H-indol-3-yl)propanoyl]pyrrolidine-2-carboxylate
N-({7-[(4-methoxy-2,5-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-5-(methoxymethyl)furan-2-carboxamide
methyl N-{1-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}carbamate
(2R)-2-amino-1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-3-(1H-indol-3-yl)propan-1-one
1-[1'-(1H-pyrrole-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
1-(furan-3-carbonyl)-4-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-1,4-diazepane
2-(3-chloro-4-fluorobenzoyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
2-fluoro-N-{3-oxo-3-[3-(piperidine-1-carbonyl)piperidin-1-yl]propyl}benzamide
N-{[1-(3,5-difluoropyridine-2-carbonyl)piperidin-4-yl]methyl}acetamide
(1R,7S)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-3-[(3-methylphenyl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
ethyl 4-({4-[5-(3-hydroxy-3-methylbut-1-yn-1-yl)furan-2-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperazine-1-carboxylate
methyl 8-[(6-methyl-4-oxo-4H-chromen-3-yl)methyl]-2-oxo-1-propoxy-1,8-diazaspiro[4.5]decane-4-carboxylate
5-cyclopropyl-1-[4-(5-methylfuran-2-yl)pyrimidin-2-yl]-N-[3-(morpholin-4-yl)propyl]-1H-pyrazole-4-carboxamide
2-(1H-indazol-1-yl)-1-[7-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-2-yl]ethan-1-one
ethyl 5-{2,7-diazaspiro[4.5]decan-2-ylmethyl}-2-oxo-2,3-dihydro-1H-imidazole-4-carboxylate
3-(6-aminopyridin-3-yl)-5-[2-(piperidin-2-yl)ethyl]phenol
5-[(1-oxo-1,2-dihydrophthalazin-2-yl)methyl]-1,2,4-oxadiazole-3-carboxamide
1-{6-hydroxy-4-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]-1,4-diazepan-1-yl}ethan-1-one
(3aS,6aR)-3-[3-(4-fluorophenyl)propyl]-5-[(trimethylpyrazin-2-yl)methyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
3-[({4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]phenyl}formamido)methyl]benzoic acid
N-[(2R,3R)-1'-(cyclopropylmethyl)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]thiophene-2-carboxamide
1-methyl-6-[3-(1H-pyrazol-1-yl)propyl]-3-(quinolin-6-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
2-amino-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)acetamide
2-[2-(dimethylamino)ethyl]-9-(3,5-dimethylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
(4aS,8aR)-6-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-decahydro-1,6-naphthyridine-4a-carboxylic acid
1-(2-cyclohexylethyl)-N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-1H-1,2,3-triazole-4-carboxamide
1-(4,6-dimethylquinazolin-2-yl)-N-(5-hydroxyadamantan-2-yl)piperidine-4-carboxamide
N-(cyclopropylmethyl)-3-(2-hydroxyphenyl)-N-(2-methoxyethyl)-1H-pyrazole-5-carboxamide
N-(3,4-dimethylphenyl)-1-(1H-indazole-3-carbonyl)piperidin-3-amine
[(3R,4R)-4-[(dimethylamino)methyl]-1-[4-(2-fluorophenyl)benzoyl]pyrrolidin-3-yl]methanol
4-amino-2-(3-chloro-4-methoxyphenyl)pyrimidine-5-carbonitrile