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3-methoxy-N-{3-methyl-1-[7-(2,3,6-trifluorobenzoyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]butyl}propanamide
2-[(4-benzylpiperazin-1-yl)methyl]-N-ethyl-N-(2-hydroxyethyl)-1,3-oxazole-4-carboxamide
N-[2-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-4-(4-methylpiperazin-1-yl)benzamide
N-[1-(propan-2-yl)-1H-pyrazol-5-yl]-1-(pyridin-3-ylmethyl)piperidin-4-amine
1-(2-chlorophenyl)-3-{1-[1-(2-hydroxyacetyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
2-ethyl-9-(2-methylpyrimidine-5-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecane
8-(2-hydroxybenzoyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
4-methyl-2-oxo-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)pentanamide
N,2-dimethyl-3-[4-(2,3,5-trifluorophenyl)-1H-1,2,3-triazol-1-yl]propanamide
(1S,5R)-6-propyl-3-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
3-(4-methoxyphenyl)-1-(3-methylbutyl)-3-[2-oxo-2-(3-propanoylpiperidin-1-yl)ethyl]pyrrolidine-2,5-dione
2,4,5-trifluoro-N-{[7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
3-[(3R,4S)-1-(2-methyl-1,3-thiazole-4-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
2-cyano-N-({1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]pyrrolidin-3-yl}methyl)benzamide
1-[(2,6-difluorophenyl)methyl]-N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-methyl-3-(2-methylpropyl)-N-{1-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-pyrazole-5-carboxamide
3-({4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}methyl)pyrrolidin-3-ol
(2S,4R)-4-amino-N-ethyl-1-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]pyrrolidine-2-carboxamide
2-({[(3R,4R)-4-(hydroxymethyl)-1-{thieno[2,3-d]pyrimidin-4-yl}pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-methylpyrazine-2-carboxamide
2-(2-{[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}ethyl)-1,2-dihydrophthalazin-1-one
3-(2-{7-ethyl-2,7-diazaspiro[4.4]nonan-2-yl}-2-oxoethyl)-3-phenyl-1-(thiophen-2-ylmethyl)pyrrolidine-2,5-dione
N-[2-(2-chlorophenyl)ethyl]-3-fluoroimidazo[1,2-a]pyridine-2-carboxamide
2-ethoxy-6-({[(1-methylpiperidin-3-yl)methyl](2-phenylethyl)amino}methyl)phenol
methyl 9-(oxan-2-ylmethoxy)-7-oxo-3-[2-(1,3-thiazol-4-yl)acetyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-(4-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl)ethan-1-ol
methyl 1-[5-(2-chloro-4-fluorophenoxymethyl)-1,2-oxazole-3-carbonyl]piperidine-4-carboxylate
2-{1-[(4-methoxy-3-methylphenyl)methyl]-4-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl}ethan-1-ol
9-[(2R)-2-hydroxy-3-methylbutanoyl]-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}pyrimidin-2-amine
1-[4-(3-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-(2-methyl-1H-imidazol-1-yl)propan-1-one
N-[(3S,4R)-4-(propan-2-yl)-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}pyrrolidin-3-yl]methanesulfonamide
N-methyl-N-(2-phenylethyl)-1-(thiophene-3-sulfonyl)piperidin-3-amine
4-[(1,4-dithiepan-6-yl)amino]-1-[2-(4-methoxyphenyl)ethyl]pyrrolidin-2-one
N-[2-(4-chlorobenzenesulfonamido)ethyl]-5-ethoxyfuran-2-carboxamide
N-methyl-3-(1-methyl-1H-pyrrol-2-yl)-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazole-5-carboxamide
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-(morpholin-3-yl)acetamide
5-(2,6-difluorophenoxymethyl)-N-methyl-N-[2-(oxan-4-yl)ethyl]-1,2-oxazole-3-carboxamide
5-(3-phenylpropyl)-5-[1-(5-propyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
N-[2-(4-fluorophenyl)ethyl]-1,4-dioxane-2-carboxamide
3-cyano-N-{[(3S,4S)-3-hydroxy-1-[2-(2-hydroxyphenyl)acetyl]piperidin-4-yl]methyl}benzamide
4-chloro-N,N-diethyl-3-(hept-6-ynamido)benzamide
2-amino-4-(furan-3-yl)-8-hydroxy-5H-indeno[1,2-b]pyridine-3-carbonitrile
4-[(2R,6S)-2,6-dimethylpiperidine-1-carbonyl]-2-(1-ethyl-1H-pyrazol-4-yl)-8-methylquinoline
2-methyl-6-[1-(2-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-2,3-dihydropyridazin-3-one
3-(1H-1,2,3-benzotriazol-1-yl)-N-methyl-N-(quinolin-5-ylmethyl)propanamide
N-cyclopentyl-2-(2,6-dioxo-1,3-diazinan-1-yl)-N-[(2-methylphenyl)methyl]acetamide
1-[4-(quinazolin-4-yl)piperazin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
2-amino-4-benzyl-6-(4-methanesulfonylphenyl)pyridine-3-carbonitrile
1-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine