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7-chloro-4-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(piperidin-1-yl)-3-[2-({[2-(pyridin-3-yloxy)ethyl]amino}methyl)phenoxy]propan-2-ol
2,8-dimethyl-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}quinoline-4-carboxamide
2-[4-(1H-pyrazol-5-yl)phenyl]-3-(pyrrolidine-1-carbonyl)pyridine
N-(diphenylmethyl)-2-[(5-ethoxyfuran-2-yl)formamido]acetamide
2-(dimethyl-1,2-oxazol-4-yl)-2-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}acetic acid
2-cyclopropyl-N-ethyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecane-9-carboxamide
{1-[5,6-dimethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-3-(2-methoxyethyl)piperidin-3-yl}methanol
4-phenyl-N-{1-[1-(1,2,5-thiadiazole-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}butanamide
4-(5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-1H-pyrazol-3-yl)phenol
N-({3-methyl-7-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(phenylsulfanyl)acetamide
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-({[2-(2-oxoimidazolidin-1-yl)ethyl]amino}methyl)piperidin-2-one
6-methyl-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]imidazo[1,2-a]pyridine-2-carboxamide
N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-6-(quinolin-8-yl)pyridine-3-carboxamide
9-[(2R)-2-hydroxy-2-phenylethyl]-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
4-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-6-methyl-1,2-dihydroquinolin-2-one
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(propan-2-yl)benzamide
4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-(1-methylcyclopropyl)benzamide
(3S,5S)-1-[(3-hydroxyphenyl)methyl]-5-(4-methylpiperazine-1-carbonyl)piperidine-3-carboxylic acid
4-chloro-N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1H-pyrazole-3-carboxamide
(1S,4S)-2-{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}-2-azabicyclo[2.2.1]heptane
2-(2-{[1-(3-methylphenyl)-1H-imidazol-2-yl]methyl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl)pyridine
[3-({1-[(2,3-dimethoxyphenyl)methyl]pyrrolidin-3-yl}methyl)phenyl]methanol
1-{[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
N-{[1-(2,1,3-benzoxadiazol-4-ylmethyl)piperidin-3-yl]methyl}-1H-pyrrole-2-carboxamide
(1R,5R)-6-[(5-methylthiophen-2-yl)methyl]-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(2S,4R)-4-amino-1-(5-chloro-7-methoxy-1-benzofuran-2-carbonyl)-N-ethylpyrrolidine-2-carboxamide
5-[({[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(propan-2-yl)amino)methyl]pyrrolidin-2-one
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
N5-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-N6-(3-methoxypropyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
2-(4-{[2-(dimethylamino)pyrimidin-5-yl]methyl}piperazin-1-yl)-1-(pyrrolidin-1-yl)ethan-1-one
1,3,5-trimethyl-N-[1-(2-methylpropyl)azepan-3-yl]-1H-pyrazole-4-sulfonamide
1-methyl-4-(thiophene-2-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
4,6-dimethyl-1-{[1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}-1,2-dihydropyrimidin-2-one
2-cyclobutyl-1-methyl-N-{[1-(2-methylpropyl)piperidin-4-yl]methyl}-7-(oxolane-2-amido)-1H-1,3-benzodiazole-5-carboxamide
7-[(1S,4S)-3,3-dimethyl-2-methylidenebicyclo[2.2.1]heptane-1-carbonyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-1-ethyl-3,5-dimethyl-1H-pyrazole-4-carboxamide
2-(cyclohex-1-ene-1-carbonyl)-1-(4-ethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
(3S,4S)-1-{[5-(3-chlorophenyl)furan-2-yl]methyl}-4-(morpholin-4-yl)pyrrolidin-3-ol
N-butyl-3-methyl-3-phenylpiperidine-1-carboxamide
1-[2-(3-fluorophenyl)piperidin-1-yl]-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
4-benzyl-3-ethyl-1-(5-hydroxypyridine-2-carbonyl)-1,4-diazepan-5-one
{[3-(1H-indol-4-yl)-1,2,4-oxadiazol-5-yl]methyl}dimethylamine
3-(3-methoxyphenyl)-N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-1H-pyrazole-5-carboxamide
3-[2-(2,6-difluorophenyl)ethyl]-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]piperidine
2-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1H-indole
2-(2-methoxyethyl)-8-[(2-methoxyphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
1-methyl-N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-1H-pyrazole-4-carboxamide
2-(4-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}piperazin-1-yl)pyrimidine
6-{3-[(2-chlorophenyl)methyl]-1,2-oxazole-5-carbonyl}-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane