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6-(1-tert-butyl-5-oxopyrrolidine-3-carbonyl)-1-methyl-1H,4H,5H,6H,7H-pyrrolo[2,3-c]pyridine-2-carboxamide
2-{9-[(3-methylthiophen-2-yl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}propanoic acid
N-(1-hydroxybutan-2-yl)-2-(methylamino)-N-(pyridin-2-ylmethyl)pyridine-3-carboxamide
4-{1-[2-(5-methylthiophen-2-yl)-1H-imidazol-1-yl]propyl}pyridine
6-chloro-N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-1-methyl-1H-indole-2-carboxamide
1-{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(pyridin-2-yl)piperazine
1-[5-(2,6-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]-4-(pyridin-4-yl)piperazine
4-ethyl-3-{1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]piperidin-3-yl}-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[3-(2-methoxyphenoxy)azetidin-1-yl]-2-(2-methyl-1H-1,3-benzodiazol-1-yl)ethan-1-one
2-(2-{[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}phenoxy)-1-(piperidin-1-yl)ethan-1-one
1-(prop-2-ene-1-sulfonyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
1-[2-(cyclopent-2-en-1-yl)acetyl]-4-(3-fluorophenoxy)piperidine-4-carboxylic acid
(3aR,5S,6S,7aS)-2-[2-methyl-6-(1H-pyrazol-1-yl)pyrimidin-4-yl]-octahydro-1H-isoindole-5,6-diol
4-[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]-N-methyl-N-(pyrazin-2-ylmethyl)pyrimidin-2-amine
N-{2-[3-(1,2-oxazolidin-2-yl)propanoyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}oxolane-2-carboxamide
7-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
[(1,5-dimethyl-1H-indazol-3-yl)methyl][1-(1H-imidazol-1-yl)propan-2-yl]amine
1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-4-phenylpiperidine-4-carbonitrile
4-[3-(3-chlorophenyl)pyrrolidine-1-carbonyl]-3-phenyl-1H-pyrazole
(2S)-2-{[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]amino}-4-(methylsulfanyl)butan-1-ol
ethyl 5-(5-ethyl-1,2-oxazole-3-carbonyl)-1-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
(2S,4R)-4-amino-1-{2-[5-(4-fluorophenyl)-2H-1,2,3,4-tetrazol-2-yl]acetyl}-N-methylpyrrolidine-2-carboxamide
(1R,5S,6R,7S)-3-(2-aminoethyl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]decane-6-carboxamide
4-[(3-fluorophenyl)methyl]-1-[4-(furan-2-yl)benzoyl]-1,4-diazepan-5-one
6-(2-fluoro-5-methoxyphenyl)pyridin-2-amine
(4aR,7aS)-1-(cyclopropylmethyl)-4-(3-hydroxypyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(2,3-dihydro-1H-inden-1-yl)-N-[2-(1H-1,2,3,4-tetrazol-5-yl)phenyl]acetamide
2-(methoxymethyl)-1-[1-(2-phenylethyl)-1H-1,2,3-triazole-4-carbonyl]piperidine
2-[(3aS,6aR)-3-[3-(4-fluorophenyl)propyl]-2-oxo-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-5-yl]pyridine-4-carboxamide
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-(2-phenylbenzoyl)piperidin-4-ol
4-(2-cyclopropylquinoline-4-carbonyl)-1,4-oxazepan-6-ol
{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}(oxolan-2-ylmethyl)amine
N-(4-chlorophenyl)-3-[1-(2,3-dimethylquinoxaline-6-carbonyl)piperidin-3-yl]propanamide
6-[(3-phenyl-1H-pyrazol-4-yl)methyl]-N-(thiophen-2-ylmethyl)-6-azaspiro[2.5]octane-1-carboxamide
1-[1-(3-benzyl-1H-1,2,4-triazol-5-yl)ethyl]-4-methylpiperidine
3-{[4-cyclopentyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}phenol
N-cyclopropyl-1-(1-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)piperidine-4-carboxamide
N-(1-{7-[(4-hydroxy-3,5-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-phenylpropanamide
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-N-(2-methoxyethyl)-1H-pyrazole-4-carboxamide
2-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}-7-methyl-2,7-diazaspiro[4.5]decan-6-one
4-(3-hydroxy-3-methylbutyl)-N-{2-[(3-methylpyridin-2-yl)amino]ethyl}benzamide
methyl({[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl})(thiophen-3-ylmethyl)amine
({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl}methyl)(methyl)(thiophen-3-ylmethyl)amine
N-[(3,4-dimethoxyphenyl)methyl]-2-[3-(2-fluorophenyl)-1-(2-methoxyethyl)-2,5-dioxopyrrolidin-3-yl]-N-methylacetamide
2-[1-(3,5-dimethylphenyl)-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-5-yl]morpholine
2-cyclopropyl-5-{2-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl}pyrimidin-4-ol
1-[1-(2,5-dimethylpyrimidin-4-yl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
5-(3-acetamidophenyl)naphthalene-1-carboxamide
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
1-{2-oxo-2-[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]ethyl}-1,2,3,4-tetrahydroquinolin-2-one