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N-[1-(4-chlorophenyl)cyclobutyl]-2-(1H-imidazol-2-yl)benzamide
N-{[7-chloro-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
N-({8-[(4-chlorophenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-3-fluorobenzamide
N-methyl-N-(pyrazin-2-ylmethyl)-2-[4-(trifluoromethyl)phenyl]-1,3-benzoxazole-5-carboxamide
N-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-1-(pyrimidin-2-yl)piperidin-3-amine
4-[(1-acetylpiperidin-4-yl)oxy]-N-[(4-ethylphenyl)methyl]-3-methoxy-N-methylbenzamide
methyl 5-{[1-(3-methoxyphenyl)propan-2-yl]amino}-3-(oxolane-3-amido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-1H-1,3-benzodiazole-2-carboxamide
2-amino-6-(5-methylfuran-2-yl)-4-(2,4,5-trimethoxyphenyl)pyridine-3-carbonitrile
4-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidine-1-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
methyl 1-[(3R,5S)-1-cyclopentyl-5-{[2-(1H-indol-3-yl)ethyl]carbamoyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
4,6-dimethyl-2-oxo-N-(1,2,3,4-tetrahydronaphthalen-2-yl)-1,2-dihydropyridine-3-carboxamide
1-(2-methoxyethyl)-8-(naphthalen-1-ylmethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-ethyl-N-[2-(4-hydroxyphenyl)ethyl]-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
4-({4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}methyl)-2,6-dimethoxyphenol
2-(4-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl)ethan-1-ol
1-(3-methoxyphenyl)-2,2-dimethyl-4-{2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}piperazine
2-methyl-6-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-2,3,4,5-tetrahydropyridazin-3-one
5-(2-chloro-4-fluorophenoxymethyl)-N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1,2-oxazole-3-carboxamide
2-(3-hydroxypropyl)-8-(pyridine-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
(2S,4S)-4-[(2-amino-6-methylpyrimidin-4-yl)amino]-N-ethyl-1-[(5-methylfuran-2-yl)methyl]pyrrolidine-2-carboxamide
methyl 3-{[(2E)-3-(3-fluorophenyl)prop-2-enamido]methyl}-5-[2-(1H-pyrazol-1-yl)acetamido]benzoate
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-6-methylimidazo[1,2-a]pyridine-2-carboxamide
{[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
3-(3-phenyl-1,2,4-oxadiazol-5-yl)-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)propanamide
3,5-dichloro-N-[2-(furan-2-ylmethyl)-3-hydroxypropyl]-4-methylbenzamide
N-(cyclohexylmethyl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-({4-[benzyl(ethyl)amino]quinazolin-2-yl}methyl)-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
2-amino-8-(3-ethoxyphenyl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
6-methyl-5-{[2-(3-phenylpropyl)morpholin-4-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-(2-methoxyphenyl)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carboxamide
(1R,4S)-2-[2-(3,4-dimethylphenyl)pyridine-3-carbonyl]-2-azabicyclo[2.2.1]heptane
2-cyclopentyl-7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-(2-chloro-6-methylphenyl)-2-[2-(morpholin-4-yl)ethyl]piperidine-1-carboxamide
3-methyl-6-(5-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}-1,2,4-oxadiazol-3-yl)pyridazine
1-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
3-[(3S,4R)-1-[(4-chlorophenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]-N-[2-(2-methoxyphenyl)ethyl]propanamide
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[2-(furan-2-ylmethyl)-3-hydroxypropyl]benzamide
3-[1-(4-phenyl-1H-imidazole-5-carbonyl)azetidin-3-yl]pyridine
2-{1-[(2-ethoxyphenyl)methyl]-4-(3-phenylpropyl)piperazin-2-yl}ethan-1-ol
N,N-dimethyl-5-({3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}methyl)-1,3-thiazol-2-amine
6-cyclopentyl-2-(4-{[3-(1H-pyrazol-1-yl)azetidin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl](methyl)[2-(3-methyl-1,2-oxazol-5-yl)ethyl]amine
3-[4-(4-methoxyphenyl)-3,3-dimethylpiperazine-1-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
methyl 1-methyl-5-({8-methyl-2,8-diazaspiro[4.5]decan-2-yl}sulfonyl)-1H-pyrrole-2-carboxylate
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-4-hydroxy-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
2-{2-oxo-2-[(2S)-2-(piperidine-1-carbonyl)pyrrolidin-1-yl]ethyl}-2,3-dihydro-1,2-benzothiazol-3-one
2,3-dimethyl-5-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]benzene-1-sulfonamide
3-[(4-methylquinolin-2-yl)methyl]-1λ6-thiane-1,1-dione
1-(2-chloroprop-2-en-1-yl)-3-{[4-(2,4-dimethylphenyl)piperazin-1-yl]methyl}-6,7-dimethoxy-1,2-dihydroquinolin-2-one