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1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
5-ethyl-5-{1-[(3-methylphenyl)methyl]piperidin-4-yl}-3-(2-methylprop-2-en-1-yl)imidazolidine-2,4-dione
N-(1-{7-[(3,4-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-phenoxyacetamide
(2S,4R)-4-[4-(4-chlorophenyl)-1H-1,2,3-triazol-1-yl]-N-methylpyrrolidine-2-carboxamide
2-(4-methylpentyl)-4-(morpholine-4-sulfonyl)morpholine
5-methyl-5-[1-(quinolin-7-ylmethyl)piperidin-4-yl]-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
N-[2-(3-chlorophenyl)ethyl]-2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
methyl 3-[(3,4-dimethylphenyl)methyl]-7-oxo-9-[2-(thiophen-3-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(1S,5R)-6-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
1-{1-[(3-chlorophenyl)methyl]piperidin-4-yl}-4-(pyrrolidine-1-carbonyl)piperidine
1-{1-[(5-methylthiophen-2-yl)methyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
methyl 6-[(3-chlorophenyl)methyl]-2-[(oxolan-2-ylmethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-[2-(4-methoxyphenyl)ethyl]-2-methyl-N-(pyridin-4-ylmethyl)-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
1-[(3aR,5S,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-3-{3-methyl-3H-imidazo[4,5-b]pyridin-2-yl}propan-1-one
2-(benzylsulfanyl)-5-[1-(pyrrolidin-3-yl)-1H-imidazol-2-yl]pyrimidine
4-(methoxymethyl)-6-[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]pyrimidine
N-[(2R,3R)-1'-[(2,5-dimethoxyphenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
(3R,4R)-1-(oxan-4-yl)-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-3-ol
1-[2-({[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}amino)ethyl]imidazolidin-2-one
1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-N-(1H-1,2,4-triazol-3-ylmethyl)piperidine-4-carboxamide
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
{[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(2-methoxyethyl)methylamine
3-(1H-indol-3-yl)-1-(4-{5-[(1E)-prop-1-en-1-yl]-2-(pyridin-3-yl)pyrimidin-4-yl}piperidin-1-yl)propan-1-one
N-methyl-N-{2-phenyl-1-[1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)piperidin-4-yl]ethyl}-2-(1H-pyrazol-1-yl)acetamide
ethyl 2-(1-{[(pyridin-2-ylmethyl)carbamoyl]methyl}piperidin-2-yl)acetate
1-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}-2-(methylamino)ethan-1-one
N-[(2-methylphenyl)methyl]-N-(prop-2-en-1-yl)oxolane-3-carboxamide
(2E)-N-{[5-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(pyridin-4-yl)prop-2-enamide
N-(2-{1-[(3-methylthiophen-2-yl)sulfonyl]piperidin-2-yl}ethyl)acetamide
N-[(3S,4R)-1-[4-(difluoromethoxy)benzoyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
methyl 6-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-2-[(oxolan-2-ylmethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
8-(3-methoxypropanoyl)-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
diethyl({5-methyl-4-[3-methyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]furan-2-yl}methyl)amine
2-[4-(2H-1,3-benzodioxol-5-yl)-2-[(3-methylpiperidin-1-yl)methyl]phenoxy]-N-[3-(dimethylamino)-2,2-dimethylpropyl]acetamide
3-(4-{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperazin-1-yl)-1,2-dihydropyrazin-2-one
(1H-imidazol-2-ylmethyl)[(8-methoxy-2H-chromen-3-yl)methyl]methylamine
9-(5-phenyl-1,3,4-thiadiazol-2-yl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
3-(3-methylphenoxymethyl)-1-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]piperidine
2-(3-acetyl-2-fluorophenyl)-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)acetic acid
N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
N-(2-methoxyethyl)-5-methyl-1-[4-(5-methylfuran-2-yl)pyrimidin-2-yl]-N-(propan-2-yl)-1H-pyrazole-4-carboxamide
3-[(4-ethoxyphenyl)methyl]-9-methoxy-10-(thiomorpholine-4-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
2-[(4-benzylpiperazin-1-yl)methyl]-N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-1,3-oxazole-4-carboxamide
1-(furan-2-carbonyl)-4-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,4-diazepane
(1H-indol-4-ylmethyl)({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})amine
1-methyl-3-phenyl-8-[1-(propan-2-yl)-1H-pyrrole-2-carbonyl]-1,8-diazaspiro[4.5]decane
methyl 3-({[7-(5-acetyl-2-fluorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}carbamoyl)propanoate
1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-4-(pyrimidin-2-yl)-1,4-diazepane
3-({4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}sulfonyl)pyridine
N-(2-{4H,5H,6H,7H,8H-cyclohepta[b]thiophene-2-carbonyl}-1,2,3,4-tetrahydroisoquinolin-7-yl)-3-methoxypropanamide