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N-(2-hydroxyethyl)-3-(4-hydroxyphenyl)-N-{[4-(methylsulfanyl)phenyl]methyl}propanamide
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-(5,6-dimethylpyridine-3-carbonyl)pyrrolidine-3-carboxylic acid
3-ethoxy-1-[3-(3-fluorophenoxymethyl)piperidin-1-yl]propan-1-one
(3S,4R)-1-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}-4-methyl-3-(2-methylpropyl)piperidin-4-ol
9-(4-aminopyrimidin-2-yl)-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
N-[3-(3-chlorophenyl)phenyl]-1-(2-hydroxypropanoyl)piperidine-4-carboxamide
2-methoxy-3-[4-(1H-pyrazol-5-yl)phenyl]pyrazine
4-{[(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidin-1-yl]methyl}-1-azatricyclo[7.3.1.05,13]trideca-3,5,7,9(13)-tetraen-2-one
(1R,5R)-6-[3-(1H-1,2,3-benzotriazol-1-yl)propanoyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
[(4-fluorophenyl)methyl][(1-methyl-1H-imidazol-2-yl)methyl](prop-2-en-1-yl)amine
3-{imidazo[1,2-a]pyridin-2-yl}-1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}propan-1-one
2-[(cyclohexylmethyl)amino]-N-[(2-fluorophenyl)methyl]acetamide
[1-(1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)piperidin-4-yl]methanol
N-({8-[(4-methylphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)furan-2-carboxamide
2-(4-{[(3aR,6aS)-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrol-2-yl]methyl}-2-chlorophenoxy)acetamide
methyl 3-(5-{[(3-ethyl-1-methyl-1H-pyrazol-5-yl)formamido]methyl}-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine-2-carbonyl)benzoate
6-[3-(2,5-difluorobenzoyl)piperidine-1-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(3-chlorophenyl)-N-{[5-fluoro-7-(6-methoxypyridazin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
(1R,3s,6r,8S)-4-[5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]-4-azatricyclo[4.3.1.13,8]undecane
1-ethyl-4-[(5-ethyl-2-methylpyrimidin-4-yl)amino]pyrrolidin-2-one
4-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-N-{[(3S,4S)-3-hydroxypiperidin-4-yl]methyl}benzamide
N-{[5-fluoro-7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclopropanecarboxamide
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-(3-methoxypyrazin-2-yl)-2,8-diazaspiro[4.5]decan-3-one
1-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}-2-{2-[(4-methyl-1,4-diazepan-1-yl)methyl]-4-(pyrimidin-2-yl)phenoxy}ethan-1-one
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}-4-(1H-pyrazol-4-yl)butanamide
2-fluoro-N-[3-(1H-indazol-1-yl)propyl]-5-sulfamoylbenzamide
N-(3,4-dimethylphenyl)-1-(6-methylquinoline-4-carbonyl)piperidin-3-amine
4-[2-(3-hydroxy-3-phenylpyrrolidin-1-yl)-2-oxoethyl]-3-methyl-1-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
6-[4-hydroxy-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine-5-carbonyl]-2,3-dimethyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
1-{3-oxo-3-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
ethyl[(1-ethyl-1H-pyrazol-4-yl)methyl](oxan-2-ylmethyl)amine
methyl 5-(6-methyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
methyl 5-{[4-(1H-indol-3-yl)butan-2-yl]amino}-3-(2-methoxyacetamido)-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]propanamide
2-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]thiophene-3-sulfonamide
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-1H-pyrrole-2-carboxamide
N-(2H-1,3-benzodioxol-5-yl)-1-(5-methoxyfuran-2-carbonyl)piperidin-3-amine
5-(2,4-difluorophenoxymethyl)-N-methyl-N-[(1-methylpiperidin-2-yl)methyl]-1,2-oxazole-3-carboxamide
(2S,4S)-N-ethyl-4-[2-(4-hydroxyphenyl)acetamido]-1-(1H-imidazol-4-ylmethyl)pyrrolidine-2-carboxamide
{1-[3-(4H-1,2,4-triazol-4-yl)phenyl]-1H-1,3-benzodiazol-2-yl}methanol
5-[1-(2,3-dimethylbenzoyl)piperidin-4-yl]-5-[(3-fluorophenyl)methyl]-3-(2-methoxyethyl)imidazolidine-2,4-dione
N-(2-methoxy-2-methylpropyl)-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
4-{1-[3-(morpholin-4-yl)benzoyl]piperidin-3-yl}benzoic acid
{1-[4-(hydroxymethyl)cyclohexanecarbonyl]-3-propylpiperidin-3-yl}methanol
({4-ethyl-5-[1-(1,2-oxazole-3-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-3-propyl-N-(pyridin-2-ylmethyl)-1H-pyrazole-5-carboxamide
ethyl 4-{[(4-phenyl-1,2,3-thiadiazol-5-yl)carbamoyl]amino}piperidine-1-carboxylate
3-[(2-fluorophenyl)formamido]-N-[3-hydroxy-3-(prop-2-en-1-yl)hex-5-en-2-yl]propanamide
3,5-dimethyl-1-(2-{3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}propyl)-1H-1,2,4-triazole
N-(carbamoylmethyl)-2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}acetamide