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N-cyclopropyl-3-[1-(3,5-dimethyl-1H-indole-2-carbonyl)piperidin-4-yl]propanamide
N-cycloheptyl-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-({4-[4-(2-methoxyphenyl)piperazin-1-yl]quinazolin-2-yl}methyl)pyridine-4-carboxamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]benzamide
(1S,3R)-3-amino-N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]cyclopentane-1-carboxamide
N-benzyl-2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-(2-hydroxyethyl)acetamide
1-[(2-methoxypyridin-3-yl)methyl]-4-[4-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]piperazine
3-phenyl-5-[3-(prop-2-en-1-yloxy)benzoyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
2-({4-[2-(4-fluorophenyl)piperidine-1-carbonyl]phenyl}(methyl)amino)ethan-1-ol
5-(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepine-3-carbonyl)pyridin-2-amine
N-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-6-cyclopropylpyrimidin-4-amine
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-(3-oxo-2,3-dihydro-1,2-benzothiazol-2-yl)acetamide
1-(4-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-3,5-dimethyl-1H-pyrrol-2-yl)ethan-1-one
6-oxo-1-(2-phenylethyl)-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]piperidine-3-carboxamide
7-(pyridin-2-yl)-4-{[2-(trifluoromethyl)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-[1-(2-methoxyethyl)-3-(2-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-[(4-methylphenyl)methyl]acetamide
N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
2-{2-[(3S,4S)-3,4-bis(hydroxymethyl)pyrrolidin-1-yl]-4-(morpholin-4-yl)pyrimidin-5-yl}-2-methylpropanoic acid
1-(2-amino-5-ethylpyrimidin-4-yl)-4-(hydroxymethyl)piperidin-4-ol
6-{1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-{1-[(3,4-difluorophenyl)methyl]-4-[(4-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
(3S,4R)-1-(benzenesulfonyl)-N,N-dimethyl-4-(4-methylphenyl)pyrrolidin-3-amine
8-[(5-methylfuran-2-yl)methyl]-3-(2-phenylpropyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-(3-ethyl-1,2-oxazol-5-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperidine
3-[(3S,7S,8aS)-3-ethyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(4-chloro-2-methylphenyl)urea
3-[(3R,4S)-1-[2-(3-hydroxyphenyl)acetyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
(2R,6R)-4-{2-[cyclopentyl(methyl)amino]acetyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
4-methyl-2-{2-oxo-2-[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]ethyl}-1,2-dihydrophthalazin-1-one
(4aR,8aS)-6-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-1-[(3,4,5-trimethoxyphenyl)methyl]-decahydro-1,6-naphthyridin-2-one
3-[2-(dimethylamino)ethyl]-5-(3-methylbutyl)-5-[1-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
1-(carbamoylmethyl)-N-[(4-fluorophenyl)methyl]-N-(prop-2-en-1-yl)piperidine-4-carboxamide
8-(1,3-benzothiazol-2-yl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
4-({5-[({2,4-dimethyl-5H,6H-furo[2,3-d]pyrimidin-6-yl}methyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)piperidine
4-[1-(cyclohex-3-ene-1-carbonyl)piperidin-3-yl]-5-(4-methylphenyl)pyrimidine
methyl N-[1-({[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}carbamoyl)ethyl]carbamate
4-ethyl-3,5-dimethyl-1-(2-{5-[2-(methylsulfanyl)ethyl]-4-phenyl-1H-imidazol-1-yl}ethyl)-1H-pyrazole
8-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-2-(dimethylamino)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
1-methyl-6-{4-[(1-methylpiperidin-3-yl)methyl]piperazine-1-carbonyl}-1H-indole
N-{[7-(3-chlorobenzoyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}cyclopropanecarboxamide
2-[2-(3-methyl-4H-1,2,4-triazol-4-yl)ethyl]-2,3-dihydro-1,2-benzothiazol-3-one
3-cyclohexyl-N-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1H-pyrazole-4-carboxamide
N-{[7-(5-chloro-2-fluorobenzoyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}-3-(pyridin-3-yl)propanamide
2-methyl-6-[4-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-2H,3H,5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-one
2-methyl-N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-(2-{4-[(4-phenylpiperazin-1-yl)methyl]phenoxy}propyl)-4-(trifluoromethyl)benzamide
2-[4-cycloheptyl-1-(thiophen-2-ylmethyl)piperazin-2-yl]ethan-1-ol
3-(2H-1,3-benzodioxol-4-ylmethyl)-N-[1-(furan-2-yl)ethyl]-9-methoxy-N-methyl-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
4-benzoyl-6-[(3,5-dimethoxyphenyl)methoxy]-1-(propan-2-yl)-1,4-diazepan-2-one
N-[2-(7-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-1-[2-(morpholin-4-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide